S. Masada

发表

Synthesis, structure-activity relationship, and pharmacological studies of novel melanin-concentrating hormone receptor 1 antagonists 3-aminomethylquinolines: reducing human ether-a-go-go-related gene (hERG) associated liabilities.

J. Kunitomo, Masaharu Nakayama, Koki Kato, 2012, Journal of medicinal chemistry.

Melanin-concentrating hormone receptor 1 antagonists. Synthesis and structure-activity relationships of novel 3-(aminomethyl)quinolines.

Koki Kato, Y. Nakano, Toshio Tanaka, 2012, Journal of medicinal chemistry.

Application of Continuous Flow-Flash Chemistry to Scale-up Synthesis of 5-Cyano-2-formylbenzoic Acid

K. Fukuda, S. Masada, H. Usutani, 2019, Organic Process Research & Development.

Discovery of 3,5-Diphenyl-4-methyl-1,3-oxazolidin-2-ones as Novel, Potent, and Orally Available Δ-5 Desaturase (D5D) Inhibitors.

Tomohiro Andou, Rei Okamoto, Ikuo Miyahisa, 2017, Journal of medicinal chemistry.

Rapid and efficient synthesis of a novel cholinergic muscarinic M1 receptor positive allosteric modulator using flash chemistry.

K. Fukuda, S. Masada, H. Usutani, 2019, Organic & biomolecular chemistry.

A new cytotoxic compound from a water extract of corn.

M. Takahashi, S. Masada, K. Uenakai, 1996, Bioscience, biotechnology, and biochemistry.

Direct and practical synthesis of 2'-O,4'-C-aminomethylene-bridged nucleic acid purine derivatives by transglycosylation

N. Cho, K. Ogi, S. Masada, 2017 .

Discovery of [ cis-3-({(5 R)-5-[(7-Fluoro-1,1-dimethyl-2,3-dihydro-1 H-inden-5-yl)carbamoyl]-2-methoxy-7,8-dihydro-1,6-naphthyridin-6(5 H)-yl}carbonyl)cyclobutyl]acetic Acid (TAK-828F) as a Potent, Selective, and Orally Available Novel Retinoic Acid Receptor-Related Orphan Receptor γt Inverse Agonis

Biching Sang, T. Imada, R. Skene, 2018, Journal of medicinal chemistry.

Discovery of orally efficacious RORγt inverse agonists, part 1: Identification of novel phenylglycinamides as lead scaffolds.

Biching Sang, Masaharu Nakayama, R. Skene, 2018, Bioorganic & medicinal chemistry.