E. Perrone

发表

Synthesis and evaluation of new elastase inhibitors. I: 1,1-Dioxocephem-4-thiolesters

A. Baici, G. Franceschi, P. Carminati, 1992 .

Bicyclopyrazoles actifs comme inhibiteurs de la kinase

A. Borgia, T. Bandiera, P. Pevarello, 2007 .

Cephem sulfones as inactivators of human leukocyte elastase. II. Keto-enol tautomerish in cephem-4-ketones.

M. Alpegiani, P. Bissolino, S. D. Nero, 1992 .

Synthesis of Penems

G. Franceschi, E. Perrone, 1990 .

2-(Heteroaroma-substituted)methyl Penems. III. Nitrogen Derivatives

A. Bedeschi, G. Franceschi, M. Alpegiani, 1988 .

Synthesis and biological properties of sodium (5R, 6S, 8R)-6 alpha-hydroxyethyl-2-carbamoyloxymethyl-2-penem-3-carboxylate (FCE 22101) and its orally absorbed esters FCE 22553 and FCE 22891.

A. Bedeschi, F. Arcamone, G. Franceschi, 1983, The Journal of antibiotics.

2-(Heteroatom-substituted)methyl penems. IV, Oxygen derivatives

A. Bedeschi, G. Franceschi, M. Alpegiani, 1990 .

Cyclic thiosulfinates and thiosulfonates from oxidation of the 2-thiacephem ring system. Synthesis of (5R)-penems by stereospecific sulfur dioxide extrusion

D. Borghi, A. Bedeschi, G. Franceschi, 1986 .

2‐Selenacephems and 1‐Dethia‐1‐selenapenems.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1986 .

Structure determination of the primary renal metabolite of the penem FCE 22101.

A. Bedeschi, G. Franceschi, G. Cassinelli, 1988, The Journal of antibiotics.

Synthesis and structure-activity relations in the class of 2-(pyridyl)penems.

A. Bedeschi, G. Franceschi, E. Perrone, 1990, The Journal of antibiotics.

Novel quaternary ammonium penems: the [(pyridinio)methyl]-phenyl derivatives.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1987, The Journal of antibiotics.

2-(quaternary ammonio)-methyl penems.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1986, The Journal of antibiotics.

Activity of new penems against defined MRSA strains

B. P. Andreini, G. Franceschi, M. Alpegiani, 1993 .

Synthesis and biological properties of FCE 25199, a new oral penem.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1992, The Journal of antibiotics.

Dual-action penems.

B. P. Andreini, G. Franceschi, M. Alpegiani, 1992, The Journal of antibiotics.

A new reductive acylation of azetidinone disulphide in the route to penems

G. Franceschi, E. Perrone, C. Battistini, 1986 .

A new class of penems, the 2-heterocyclyl(thio)methyl derivatives.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1984, The Journal of antibiotics.

Desulphurative approaches to penem antibiotics. V. 2-(Functionalized methyl)penems from 3-methylenecepham-1-oxides

A. Bedeschi, G. Franceschi, M. Alpegiani, 1984 .

Desulphurative approaches to penem antibiotics. VI. From penam methyl esters to penem acetonyl esters: A fully conservative conversion

A. Bedeschi, G. Franceschi, M. Alpegiani, 1984 .

The carbonyl-carbonyl coupling route to penems : a stepwise analysis

A. Bedeschi, G. Franceschi, M. Alpegiani, 1984 .

SOLID STATE PHOTOREACTIVITY OF A DIOXOLENONEMETHYL ESTER

D. Borghi, E. Fasani, A. Albini, 1995 .

Desulphurative approaches to penem antibiotics. I. 4-acyldithioazetidin-2-ones via thermolysis of penicillin-derived sulphoxides

A. Bedeschi, M. Alpegiani, E. Perrone, 1983 .

A new reductive acetylation of sulphinic acids and its application to the synthesis of 2-acetylthio-4-oxoazetidines

E. Perrone, J. Irving, R. J. Stoodley, 1983 .

Contrasting thermal behaviour of diastereoisomeric 4-acetylthio-3-acylamino-1-(α-triphenylphosphoranylidene)alkoxycarbonylmethylazetidin-2-ones

E. Perrone, J. Irving, R. J. Stoodley, 1983 .

Desulphurative approaches to penem antibiotics. III. Synthesis and desulphurisation of 3-methyl-2-thiacephem-4-carboxylates

A. Bedeschi, G. Franceschi, M. Alpegiani, 1983 .

Desulphurative approaches to penem antibiotics. II. 4-acyldithioazetidin-2-ones from penicillin derived sulphenimides, thiolsulphonates and disulphides.

A. Bedeschi, M. Alpegiani, E. Perrone, 1983 .

2-(Heteroatom-Substituted)methyl Penems. Part 3. Nitrogen Derivatives.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1988 .

Rearrangement of unsym-azetidinone disulphides to 2β-(thio-substituted methyl) penams

D. Borghi, M. Alpegiani, E. Perrone, 1990 .

Silver-assisted 1,2-cleavage of penicillins. A three-step synthesis of optically active penems

A. Bedeschi, G. Franceschi, M. Alpegiani, 1985 .

Synthesis and β-lactamase inhibitory activity of 6-hydroxyethyl thiaclavulanic acid

W. Cabri, A. Bedeschi, E. Perrone, 1993 .

On the Preparation of 4-Hydroxymethyl-5-Methyl-1,3-Dioxol-2-One

M. Alpegiani, E. Perrone, F. Zarini, 1992 .

Synthesis and antimicrobial spectrum of FCE 22101 and its orally available ester FCE 22891.

A. Bedeschi, G. Franceschi, M. Alpegiani, 1989, The Journal of antimicrobial chemotherapy.

Ring nitrogen functionalization of 2‐aminothiazol‐4‐acetic acid derivatives. I. Synthesis and properties of novel 2‐aminothiazole N‐oxides

G. Nannini, A. Bedeschi, M. Alpegiani, 1984 .

6‐Substituted Pyrrolo[3,4‐c]pyrazoles: An Improved Class of CDK2 Inhibitors

C. Mercurio, A. Vulpetti, D. Ballinari, 2007, ChemMedChem.

Discovery of Entrectinib: A New 3-Aminoindazole As a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.

A. Isacchi, G. Canevari, E. Felder, 2016, Journal of medicinal chemistry.

Synthesis of novel cephem-4-ketones. A new series of human leukocyte elastase inhibitors

G. Franceschi, M. Alpegiani, P. Bissolino, 1991 .

Cephalosporins. III. Synthesis and structure-activity relationships of 7-vinylenethioacetamid:o cephalosporins with a tetrazolo-pyridazine at the 3-position.

G. Nannini, A. Bedeschi, D. Severino, 1981, Journal of antibiotics (Tokyo. 1968).

Tricyclic cephems as inhibitors of human leukocyte elastase. thieno[3,4-c]cepham sulfones and pyrrolo[3,4-c]cepham sulfones

M. Alpegiani, P. Bissolino, E. Perrone, 1995 .

Synthesis of Novel Cephem 4-Ketones. A New Series of Human Leukocyte Elastase Inhibitors.

G. Franceschi, M. Alpegiani, P. Bissolino, 1992 .

Cephalosporins. VII. Synthesis and antibacterial activity of new cephalosporins bearing a 2-imino-3-hydroxythiazoline (2-aminothiazole N-oxide) in the C-7 acylamino side chain.

G. Nannini, M. Alpegiani, E. Perrone, 1984, The Journal of antibiotics.

Cephalosporins. VI. Synthesis and structure-activity relationships of new 7 beta-[(Z)-2-alkoxyimino-2-(2-aminothiazol-4-yl)acetamido]cephalosporins with a tetraxolopyridazine at the 3-position.

G. Nannini, M. Alpegiani, E. Perrone, 1983, The Journal of antibiotics.

Cephalosporins. V. Synthesis and in vitro activity of some 7-[2-methoxyimino-(substituted thio)alkanoyl]amino cephalosporanic acid derivatives.

G. Nannini, A. Bedeschi, E. Perrone, 1982, The Journal of antibiotics.

Cephalosporins. II. Synthesis and structure-activity relationships of new 7-vinylenethioacetamido and thioacrylamido cephalosporins.

G. Nannini, A. Bedeschi, D. Severino, 1981, The Journal of antibiotics.

Studies on cephem sulfones as mechanism-based inactivators of human leukocyte elastase. III: Reactions ensuing from chemical β-lactam cleavage

D. Borghi, M. Alpegiani, P. Bissolino, 1993 .

Stereoselective alkoxy-de-amination of 7β-Amino-3-Deacetoxy cephalosporanic acid

D. Borghi, M. Alpegiani, E. Perrone, 1991 .

Stereoselective Alkoxy‐De‐Amination of 7β‐Amino‐3‐ deacetoxycephalosporanic Acid.

D. Borghi, M. Alpegiani, P. Bissolino, 1992 .

Correction to Discovery of Entrectinib: A New 3-Aminoindazole as a Potent Anaplastic Lymphoma Kinase (ALK), c-ros Oncogene 1 Kinase (ROS1), and Pan-Tropomyosin Receptor Kinases (Pan-TRKs) inhibitor.

A. Isacchi, G. Canevari, E. Felder, 2019, Journal of medicinal chemistry.