T. Herpin

发表

Solid-phase synthesis of α-hydroxy phosphonates and hydroxystatine amides. Transition-state isosteres derived from resin-bound amino acid aldehydes

R. Dolle, T. Herpin, Y. Shimshock, 2001 .

Synthesis and diversity analysis of lead discovery piperazine-2-carboxamide libraries

P. Menard, R. Labaudinière, J. Salvino, 2004, Molecular Diversity.

2-Arylbenzoxazoles as novel cholesteryl ester transfer protein inhibitors: optimization via array synthesis.

David S. Taylor, David S Nirschl, C. Weigelt, 2008, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of novel pyrrolidine acid analogs as potent dual PPARα/γ agonists.

Weiqi Wang, A. Doweyko, T. Harrity, 2015, Bioorganic & medicinal chemistry letters.

beta-alanine dipeptides as MC4R agonists.

J. Macor, R. Ruel, D. Shi, 2003, Bioorganic & medicinal chemistry letters.

Discovery of 2-(phenoxypyridine)-3-phenylureas as small molecule P2Y1 antagonists.

J. Y. Roberge, D. Schnur, A. Cacace, 2013, Journal of medicinal chemistry.

Directed sorting approach for the synthesis of large combinatorial libraries of discrete compounds.

T. Herpin, George C. Morton, 2003, Methods in enzymology.

Novel solid-phase synthesis of 1,5-benzothiazepine-4-one derivatives

R. Labaudinière, T. Herpin, M. SalvinoJoseph, 2000 .

Allylindium and allylboronic acid pinacolate: Mild reagents for the allylation of resin-bound aldehydes. Application to the solid-phase synthesis of hydroxypropylamines

C. Cavallaro, R. Dolle, T. Herpin, 1999 .

Deprotection of N-Alloc amines by Pd(0)/DABCO—an efficient method for in situ peptide coupling of labile amino acids

O. Reiser, T. Herpin, Sunnhild Salmen, 2001 .

Novel safety-catch linker and its application with a Ugi/De-BOC/Cyclization (UDC) strategy to access carboxylic acids, 1,4-benzodiazepines, diketopiperazines, ketopiperazines and dihydroquinoxalinones

C. Hulme, R. Labaudinière, J. Salvino, 1998 .

Synthesis of a 10,000 member 1,5-benzodiazepine-2-one library by the directed sorting method.

R. Labaudinière, J. Salvino, T. Herpin, 2000, Journal of combinatorial chemistry.

Polymer-supported tetrafluorophenol: a new activated resin for chemical library synthesis.

R. Labaudinière, J. Salvino, D. Engers, 2000, Journal of combinatorial chemistry.

Discovery of tyrosine-based potent and selective melanocortin-1 receptor small-molecule agonists with anti-inflammatory properties.

J. Tokarski, J. Macor, A. Khanna, 2003, Journal of medicinal chemistry.

2-hydroxy-N-arylbenzenesulfonamides as ATP-citrate lyase inhibitors.

Dong Cheng, Ramesh Padmanabha, Kristen Pike, 2007, Bioorganic & medicinal chemistry letters.

β-Alanine dipeptides as MC4R agonists

R. Ruel, D. Shi, I. Zimanyi, 2003 .

A selective small molecule agonist of the melanocortin‐1 receptor inhibits lipopolysaccharide‐induced cytokine accumulation and leukocyte infiltration in mice

J. Haycock, K. McIntyre, J. Macor, 2006, Journal of leukocyte biology.

Australian biotech companies: Navigating the maze

J. E. Foley, T. Herpin, H. Karuso, 2005 .