J. Scherkenbeck

发表

Small Molecules Antagonise the MIA-Fibronectin Interaction in Malignant Melanoma

R. Gasper, E. Hofmann, R. Stoll, 2016, Scientific Reports.

Anthelmintic PF1022A: stepwise solid-phase synthesis of a cyclodepsipeptide containing N-methyl amino acids

F. Sondermann, J. Scherkenbeck, Sebastian Lüttenberg, 2011, Tetrahedron.

Structures of some moenomycin antibiotics - inhibitors of peptidoglycan biosynthesis

J. Heijenoort, J. Scherkenbeck, M. Limbert, 1993 .

Cyclodepsipeptides: A Rich Source of Biologically Active Compounds for Drug Research

J. Scherkenbeck, Sivatharushan Sivanathan, 2014, Molecules.

Segment Solid-Phase Total Synthesis of the Anthelmintic Cyclooctadepsipeptides PF1022A and Emodepside

K. Brücher, J. Scherkenbeck, Sebastian Lüttenberg, 2012 .

Syntheses of analogues of the insect neuropeptide proctolin containing an oxazole ring as an amide bond replacement.

F. Stieber, J. Scherkenbeck, A. Plant, 2001, Organic letters.

Sequence-selective molecular recognition of the C-terminal CaaX-boxes of Rheb and related Ras-proteins by synthetic receptors.

R. Stoll, K. T. Yip, Jasmin Autzen, 2014, ACS chemical biology.

A highly efficient synthesis of the anthelmintic cyclooctadepsipeptide PF1022A

N. Mencke, J. Scherkenbeck, A. Harder, 1995 .

The Bisphenol A analogue Bisphenol S binds to K‐Ras4B – implications for ‘BPA‐free’ plastics

C. Herrmann, R. Stoll, J. Scherkenbeck, 2016, FEBS letters.

Enantiomerically pure 3-aryl- and 3-hetaryl-2-hydroxypropanoic acids by chemoenzymatic reduction of 2-oxo acids.

J. Tent, J. Scherkenbeck, Sivatharushan Sivanathan, 2015, The Journal of organic chemistry.

Isolation, total synthesis and quantification of caffeoylisocitric acid, a characteristic ingredient of the superfood amaranth

Benedikt Ringbeck, N. Schebb, J. Scherkenbeck, 2019, Tetrahedron.

Chimeric cyclodepsipeptides as mimetics for the anthelmintic PF1022A.

J. Scherkenbeck, A. Harder, H. Dyker, 2004, Bioorganic & medicinal chemistry letters.

Macrocyclic analogues of the diuretic insect neuropeptide helicokinin I show strong receptor-binding.

J. Scherkenbeck, Chien Tran Van, D. Nennstiel, 2015, Bioorganic & medicinal chemistry.

Enantioselective Reduction of 3-Aryl-2-oxo-propanoic Acids: A Comparison of Enzymatic and Transition-Metal-Catalyzed Methods

J. Scherkenbeck, Sebastian Lüttenberg, J. Heyden, 2013 .

Asymmetric total synthesis of the indole alkaloid cyclopiazonic acid and first structure–activity data

M. Schindler, J. Scherkenbeck, H. Antonicek, 2011 .

The Natural Plant Product Rottlerin Activates Kv7.1/KCNE1 Channels

S. Meuth, F. Lang, G. Seebohm, 2016, Cellular Physiology and Biochemistry.

Structural Prerequisites for Receptor Binding of Helicokinin I, a Diuretic Insect Neuropeptide from Helicoverpa zea

G. Seebohm, O. Zerbe, J. Scherkenbeck, 2014 .

Receptor assay guided structure‐activity studies of helicokinin insect neuropeptides and peptidomimetic analogues

K. Brücher, J. Scherkenbeck, H. Antonicek, 2009, Journal of peptide science : an official publication of the European Peptide Society.

Syntheses of analogues of the insect neuropeptide proctolin containing an oxazole ring as an amide bond replacement.

F. Stieber, J. Scherkenbeck, A. Plant, 2001, Organic letters.

Model studies directed toward forskolin: Synthesis of a tricyclic model compound from farnesol

J. Scherkenbeck, P. Welzel, Karl-Heinz Metten, 1988 .

Syntheses of depsipeptide analogues of the insect neuropeptide proctolin.

F. Stieber, J. Scherkenbeck, A. Plant, 2002, Bioorganic & medicinal chemistry letters.

Synthesis and SERCA activities of structurally simplified cyclopiazonic acid analogues.

M. Schindler, J. Scherkenbeck, K. Wölfel, 2011, Bioorganic & medicinal chemistry.

Semisynthetic routes to PF1022H--A precursor for new derivatives of the anthelmintic cyclooctadepsipeptide PF1022A.

J. Scherkenbeck, Sivatharushan Sivanathan, Florian Körber, 2016, Bioorganic & medicinal chemistry.

The Knight route to cyclopiazonic acid: enantioselective synthesis of a key intermediate

F. Sondermann, J. Scherkenbeck, C. Beyer, 2010 .

1,9-Dideoxyforskolin : Enolate formation - oxidation

J. Scherkenbeck, P. Welzel, D. Böttger, 1987 .

Sequence‐Selective Covalent CaaX‐Box Receptors Prevent Farnesylation of Oncogenic Ras Proteins and Impact MAPK/PI3 K Signaling

D. Wolters, U. Koch, B. Klebl, 2021, ChemMedChem.

Applications of combinatorial chemistry in the agrosciences.

Jürgen Scherkenbeck, Stephen Lindell, J. Scherkenbeck, 2005, Combinatorial chemistry & high throughput screening.

Prospects for combinatorial chemistry in the agrosciences.

Stephen D Lindell, Jürgen Scherkenbeck, J. Scherkenbeck, 2005, Combinatorial chemistry & high throughput screening.

P. Jeschke, J. Scherkenbeck, A. Harder, 2002, Current topics in medicinal chemistry.

Moenomycin a: Minimum structural requirements for biological activity

Frithjof Kruggel, Peter Welzel, G. Seibert, 1987 .

Spatial discrimination of pheromones and behavioural antagonists by the tortricid moths Cydia pomonella and Adoxophyes orana

R. Potting, R. P. J. Potting, P. M. Lösel, 1999, Journal of Comparative Physiology A.

Factors affecting the field performance of an attracticide against the codling moth Cydia pomonella.

R. Potting, J. Scherkenbeck, P. Lösel, 2002, Pest management science.

Appeal: efficacy and mode of action of attract and kill for codling moth control

J. Romeis, J. Scherkenbeck, R. Olszak, 2001 .

Laboratory and field experiments towards the development of an attract and kill strategy for the control of the codling moth, Cydia pomonella

R. Potting, A. Elbert, J. Scherkenbeck, 2000 .

The potential of semiochemicals for control of Phorodon humuli (Homoptera: Aphididae)

L. Wadhams, J. Pickett, J. Hardie, 1996 .

Effect of primary‐host kairomones on the attractiveness of the hop‐aphid sex pheromone to Phorodon humuli males and gynoparae

L. Wadhams, J. Pickett, J. Hardie, 1996 .

Insect neuropeptides: structures, chemical modifications and potential for insect control.

J. Scherkenbeck, Tino Zdobinsky, 2009, Bioorganic & medicinal chemistry.

Aggregation Agents in German Cockroach Blattella germanica: Examination of Efficacy

G. Wendler, M. Dambach, J. Lenz, 1999, Journal of Chemical Ecology.

Rottlerin: Structure Modifications and KCNQ1/KCNE1 Ion Channel Activity

G. Seebohm, N. Strutz‐Seebohm, J. Scherkenbeck, 2020, ChemMedChem.

A practical method for the regeneration of Kaiser-oxime resin

F. Sondermann, J. Scherkenbeck, Sebastian Lüttenberg, 2013 .

Bisphenol A binds to Ras proteins and competes with guanine nucleotide exchange: implications for GTPase-selective antagonists.

R. Heumann, C. Herrmann, S. Ince, 2013, Journal of medicinal chemistry.

Detection of major and minor sex pheromone components by the male codling moth Cydia pomonella (Lepidoptera: Tortricidae).

C. Zebitz, J. Scherkenbeck, P. Lösel, 1997, Journal of insect physiology.

Synthesis, conformational studies and anthelmintic activity of a constrained PF1022A analogue

J. Scherkenbeck, F. Reichel, D. Gondol, 1999 .

Synthesis, Biological Evaluation, and Binding Mode of a New Class of Oncogenic K‐Ras4b Inhibitors

U. Koch, B. Klebl, A. Choidas, 2022, ChemMedChem.

Factors Accounting for the Variability in the Behavioral Response of the Onion Fly (Delia antiqua) to n-Dipropyl Disulfide

J. Romeis, J. Scherkenbeck, D. Ebbinghaus, 2003, Journal of Chemical Ecology.

Structures of Micelle‐Bound Selected Insect Neuropeptides and Analogues: Implications for Receptor Selection

O. Zerbe, J. Scherkenbeck, H. Antonicek, 2009, Chembiochem : a European journal of chemical biology.

Synthesis and structure-activity relationships of some milbemycin E analogues

J. Scherkenbeck, U. Wachendorff-Neumann, 1991 .

PF1022A--a novel anthelmintic cyclooctadepsipeptide. Modification and exchange of the N-methyl leucine residues.

J. Scherkenbeck, A. Harder, A. Plant, 1998, Bioorganic & medicinal chemistry letters.

Allosteric Activation of GDP-Bound Ras Isoforms by Bisphenol Derivative Plasticisers

C. Herrmann, I. Helfrich, H. Bachmann, 2018, International journal of molecular sciences.

Modern trends in agrochemistry

J. Scherkenbeck, 2009 .

Azadepsipeptides: synthesis and evaluation of a novel class of peptidomimetics.

J. Scherkenbeck, D. Gondol, A. Harder, 2001, The Journal of organic chemistry.

Compounds for the treatment of melanoma

R. Stoll, K. T. Yip, Jasmin Autzen, 2015 .

The Bisphenol A analogue Bisphenol S binds to K‐Ras4B – implications for ‘BPA‐free’ plastics

C. Herrmann, R. Stoll, J. Scherkenbeck, 2016, FEBS letters.