A. Daïch

发表

From Conventional Lewis Acids to Heterogeneous Montmorillonite K10: Eco-Friendly Plant-Based Catalysts Used as Green Lewis Acids.

C. Waterlot, M. Hechelski, Alina Ghinet, 2018, ChemSusChem.

Synthesis of highly functionalized pyrrolidines as tunable templates for the direct access to (±)-coerulescine and the tricyclic core of martinellines.

Ronan Le Goff, A. Daïch, A. M. Lawson, 2013, Organic & biomolecular chemistry.

The CERT antagonist HPA-12: first practical synthesis and individual binding evaluation of the four stereoisomers.

F. Ausseil, L. Fleury, C. Santos, 2015, Bioorganic & medicinal chemistry.

Synthesis of novel chiral 1,4-dihydropyridinyl Schiff-base ligands, with characterization and evaluation of calcium channel blocker activity

L. Varečka, B. Lakatoš, P. Baran, 2014, Monatshefte für Chemie - Chemical Monthly.

CIAT with simultaneous epimerization at two stereocenters. Synthesis of substituted β-methyl-α-homophenylalanines

F. Považanec, A. Daïch, D. Berkeš, 2007 .

A versatile domino process for the synthesis of substituted 3-aminomethylene-chromanones and 2-pyridones catalyzed by CsF

A. Daïch, A. M. Lawson, S. Comesse, 2013 .

Oxidized isoquinolinoisoindolinone and benzazepinoisoindolinone alkaloids cores by convergent cyclisation processes : π-aromatic attack of thionium and oxonium species

Till Bousquet, A. Daïch, J. Fleury, 2006 .

Five‐Membered Nitrogen Heterocycles Synthesis through 1,3‐Dipolar Cycloaddition of Non‐Stabilized Azomethine Ylides with 2‐Pyridone Heteroaromatic Systems as Dipolarophiles

Sami Ben Salah, A. Daïch, I. Chataigner, 2020 .

Aza-heterocyclic frameworks through intramolecular π-system trapping of spiro-N-acyliminiums generated from isoindolinone

M. Knorr, C. Strohmann, Anis Romdhane, 2021, New Journal of Chemistry.

Synthesis and sequential diastereoselective incorporation of hydroxyl groups into hexahydrofuro[3,2-f]indolizin-7(2H)-one to give mono-, di- and tetra-hydroxyfuroindolizidines.

J. Moncol’, Michal Šoral, A. Daïch, 2020, Organic & biomolecular chemistry.

Synthesis and reactivity of (1S)-N-(1-phenylethyl)maleimide towards nucleophiles: an application to preparation of chiral pyrroloisothiochroman and pyrrolobenzo[d]thiepine based on π-cationic cyclization

B. Decroix, A. Daïch, A. Jilale, 2001 .

A facile fused-dioxaza-ring synthesis from N-hydroxyphthalimide

B. Decroix, A. Daïch, P. Netchitaïlo, 1999 .

Synthesis of isoindolo[1,3]benzoxazine derivatives through intramolecular arylation of N‐acyliminium ions

B. Decroix, N. Hucher, A. Daïch, 1998 .

Synthesis and reactivity of oxopyrrolidinothieno[2]azepinones: [3]Benzazepine antidepressant analogs

B. Decroix, A. Daïch, A. Mamouni, 1996 .

Highly Enantioselective Semisynthesis of (+)/(-)-Gossypol Schiff Base Derivatives from Ground Plant Material.

A. Daïch, A. M. Lawson, M. Othman, 2019, Journal of natural products.

Metal-Free Cascade Approach toward Polysubstituted Indolizines from Chromone-Based Michael Acceptors.

A. Daïch, A. M. Lawson, M. Othman, 2017, Organic letters.

Smart and concise entry to chiral spiro[cyclopentane-indolizidine]-tetraol diastereomers as a new aza-spirocyclic framework

J. Moncol’, A. Daïch, P. Šafár̆, 2021, New Journal of Chemistry.

Combined Chemical, Biological and Theoretical DFT‐QTAIM Study of Potent Glycosidase Inhibitors Based on Quaternary Indolizinium Salts

Vincent Tognetti, L. Joubert, N. Prónayová, 2012 .

Simple access to highly functional bicyclic γ- and δ-lactams: origins of chirality transfer to contiguous tertiary/quaternary stereocenters assessed by DFT.

Ronan Le Goff, A. Daïch, A. M. Lawson, 2015, Chemistry.

Sulfonation of Polyvinylidene fluoride: Investigation of the Microstructure by {1H, 13C, 19F} NMR Spectroscopy and Mechanisms

L. Truong, K. Fatyeyeva, H. Oulyadi, 2022, ACS Applied Polymer Materials.

Synthesis of a new pyrrolo[1,3]diazepine: 4H‐pyrrolo[1,2‐a]thieno[2,3‐e][1,3]diazepine

B. Decroix, A. Daïch, P. Ohier, 1995 .

Toward new camptothecins. Part 6: Synthesis of crucial ketones and their use in Friedländer reaction

P. Gautret, J. Hénichart, B. Rigo, 2010 .

Unexpected reversible nitrogen atom transfer in the synthesis of polysubstituted imides and 7-aza-hexahydroindolones via enaminonitrile γ-lactams

H. Oulyadi, A. Daïch, S. Comesse, 2009 .

Expedious and practical synthesis of the bioactive alkaloids rutaecarpine, euxylophoricine A, deoxyvasicinone and their heterocyclic homologues

A. Daïch, A. Elomri, A. Hamid, 2006 .

The Reactivity of Enantiopure (S )-6-Oxopipecolic Acid and Corresponding Pyridoisoquinolines Under Acidic Conditions

J. Moncol’, B. Balónová, Michal Šoral, 2018, European Journal of Organic Chemistry.

An expedient synthesis of 7(S)-ethyl-8(R or S)-indolizidinols based on a thiophene reductive desulfurization

P. Baran, A. Daïch, P. Šafár̆, 2007 .

Access to substituted thiapyrrolizidinones and fused pyridones using the domino N-acyliminium-thionium equilibrium/1,3-dipolar cycloaddition/desulfurization cyclization cascade

H. Oulyadi, A. Daïch, A. Hamid, 2006 .

A Versatile Domino Process for the Synthesis of Substituted 3-Aminomethylene-chromanones and 2-Pyridones Catalyzed by CsF.

A. Daïch, A. M. Lawson, S. Comesse, 2013 .

Competitive Intramolecular C—C vs. C—O Bond Coupling Reactions Toward C6 Ring-Fused 2-Pyridone Synthesis.

A. Rebbaa, A. Daïch, A. M. Lawson, 2016 .

A domino N-amidoacylation/aldol-type condensation approach to the synthesis of the topo-I inhibitor Rosettacin and derivatives.

A. Daïch, S. Comesse, M. Sanselme, 2008, The Journal of organic chemistry.

2.17 Addition to N -Acyliminium Ions of Heteroatoms such as Oxygen, Nitrogen, Sulfur, and Selenium as Internal Nucleophiles

Alina Ghinet, B. Rigo, A. Daïch, 2014 .

Reactivity of N‐benzyl‐3‐nitrophthalimide: A facile access to isoindolo[1,2‐d][3,5]benzothiazocine derivatives

B. Decroix, A. Daïch, A. Jilale, 2000 .

Intramolecular N-aza-amidoalkylation in association with Witkop–Winterfeldt oxidation as the key step to synthesize Luotonin-A analogues

A. Daïch, S. Comesse, Frédéric Pin, 2011 .

Expeditious Synthesis of the Topoisomerase I Inhibitors Isoindolo[2,1-b]isoquinolin-7(5H)-one and the Alkaloid Rosettacin Based on Aryl Radical Cyclization of Enamide Generated by Using N-Acyliminium Chemistry

A. Bridoux, Lahssen El Blidi, A. Daïch, 2015 .

Studies on (1S)-N-(1-Phenylethyl)-phthalimide: Synthesis of Both Chiral Spiro Indane and Benzazepine Derivatives

B. Decroix, A. Daïch, A. Jilale, 2002 .

Synthesis of benzo(or furo)[5,6]azepino[2,1-a]isoindolone derivatives: π-cyclisations of N-acyliminium ions

B. Decroix, P. Pigeon, A. Daïch, 1998 .

Acid-mediated intramolecular cationic cyclization using an oxygen atom as internal nucleophile: synthesis of substituted oxazolo-, oxazino- and oxazepinoisoindolinones ☆ ☆☆

B. Decroix, A. Daïch, S. Marchalin, 2002 .

Diastereoselective access to chiral non‐racemic [1,3]oxazolo‐[2,3‐a]isoindol‐5‐one ring systems viaO‐cationic cyclization

A. Daïch, S. Marchalin, Abderrahim Chihab-Eddine, 2002 .

Diastereoselective Alkylation of Aromatic Enamidone Functionality in Isoindole Series:A Convenient Route to Chiral Aza-analogues of Senkyunolide-E

B. Decroix, A. Daïch, A. Jilale, 1999 .

Tetracyclic Systems: An Efficient and Rapid Synthesis of New Pyrrolothieno[1,3]Thiazocines

B. Decroix, A. Daïch, A. Mamouni, 1997 .

Access to 3-spiroindolizines containing an isoindole ring through intra-molecular arylation of spiro-N-acyliminium species: a new family of potent farnesyltransferase inhibitors.

M. Knorr, C. Strohmann, J. Dubois, 2019, Organic & biomolecular chemistry.

Palladium(II) Catalyzed Cyclization: A Facile Access to New Difunctionalized Thieno[3,2-f]indolizine

B. Decroix, A. Daïch, A. Mamouni, 1998 .

Toward the improvement of the tandem halide displacement/amide coupling spiro-cyclization as a new route to γ-lactam and pyrroloisoquinoline templates

A. Daïch, S. Comesse, D. Berkeš, 2009 .

Benzo[7,8]indolizinoquinoline scaffolds based on Mg(ClO4)2-promoted regiospecific imide reduction and π-cyclization of N-acyliminium species. Analogues of the topo-1 poison rosettacin and 22-hydroxyacuminatine alkaloids

A. Souizi, Alina Ghinet, B. Rigo, 2019, Arabian Journal of Chemistry.

Kinetic versus thermodynamic access to imidazoisoindolones, benzimidazoisoindolones, and [1,4]diazepinoisoindolones: intramolecular nitrogen and π-aromatic trapping of N-acyliminium cation

B. Decroix, A. Daïch, L. Hijfte, 2004 .

Evaluation of N-Hydroxymethylphthalimide in alkaline medium: Novel entry to the tricyclic [1,3]oxazepine core via an intramolecular π and o-cationic cyclization

A. Daïch, S. Marchalin, Abderrahim Chihab-Eddine, 2003 .

Reactivity of N-Benzyl-3-nitrophthalimide: A Facile Access to Isoindolo[1,2-d][3,5]benzothiazocine Derivatives.

B. Decroix, A. Daïch, A. Jilale, 2001 .

An innovative and efficient method to synthesize meloxicam in one-step procedure with respect to the green chemistry

C. Waterlot, M. Hechelski, Alina Ghinet, 2018, Journal of the Iranian Chemical Society.

A new process for Na2Ca(HPO4)2 synthesis and its application as a heterogeneous catalyst in Knoevenagel condensation

S. Boukhris, A. Hassikou, A. Souizi, 2018 .

Diastereoselective Access to Tri‐ and Pentacyclic Spiro‐γ‐lactam‐oxindole Cores through a Tandem Aza‐Michael Initiated Ring Closure Sequence

A. Daïch, S. Comesse, M. Sanselme, 2011 .

π-Aromatic and Sulfur Nucleophilic Partners in Cationic π-Cyclizations: Intramolecular Amidoalkylation and Thioamidoalkylation Cyclization via ω-Carbinol Lactams1,2

B. Decroix, N. Hucher, A. Daïch, 2001 .

Highly Stereoselective Domino Oxa‐Michael/Aza‐Michael/Cyclization: Synthesis of Bicyclic Lactams and Spirooxindole Skeleton

A. Daïch, A. M. Lawson, S. Comesse, 2015 .

Domino process optimized via ab initio study for an alternative access to bicyclic lactams.

A. Daïch, S. Comesse, Arnaud Martel, 2011, Organic letters.

Asymmetric Synthesis and Binding Study of New Long-Chain HPA-12 Analogues as Potent Ligands of the Ceramide Transfer Protein CERT.

F. Ausseil, L. Fleury, C. Santos, 2016, Chemistry.

Pyrrolo[1,4]diazepines, via thermolyse of carbonylazides, and [3,2,2]cyclazines, via Diels-Alder reaction of [f]indolizines, annelated to [1]benzothiophene

B. Decroix, A. Daïch, P. Ohier, 1996 .

Bi(OTf)3‐Catalysed Access to 2,3‐Substituted Isoindolinones and Tricyclic N,O‐Acetals by Trapping of Bis‐N‐Acyliminium Species in a Tandem Process

Vincent Tognetti, L. Joubert, A. Daïch, 2016 .

Novel syntheses of densely functionalized indolizines, di- and tetrahydroindolizines from 2-formyl-1,4-dihydropyridine systems based on cascade process

I. Svoboda,, A. Daïch, J. Kožíšek, 2001 .

Regioselective ring opening of the chiral non-racemic furoindolizidinols. New entry to alkylindolizidinediol derivatives

N. Prónayová, A. Daïch, S. Comesse, 2010 .

1,3,5‐Oxadiazine Framework by Oxygen vs. Nitrogen Trapping of an N‐Acyliminium Ion Derived from N,O‐bis‐TMS Pyroglutamic Acid

J. Dubois, Alina Ghinet, B. Rigo, 2017 .

Original Mitsunobu-Triggered Sequence Involved in a One-Pot Domino Process toward Tetracyclic Systems Bearing a Bis-N,O-acetal Junction.

A. Daïch, A. M. Lawson, C. Denhez, 2016, The Journal of organic chemistry.

Intermolecular and intramolecular alpha-amidoalkylation reactions using bismuth triflate as the catalyst.

A. Daïch, S. Comesse, B. Garrigues, 2007, The Journal of organic chemistry.

Phenyliodine(III) Diacetate/I2 -Mediated Domino Approach for Pyrrolo[1,4]Thiazines and 1,4-Thiazines by a One-Pot Morin Rearrangement of N,S-Acetals.

J. Moncol’, Alina Ghinet, B. Rigo, 2019, Chemistry.

Tandem Michael addition/amino-nitrile cyclization from 2-formyl-1,4-DHP in the synthesis of novel dihydroindolizine-based compounds.

H. Oulyadi, P. Baran, A. Daïch, 2006, The Journal of organic chemistry.

Tandem Michael addition/amino-nitrile cyclization from 2-formyl-1,4-DHP in the synthesis of novel dihydroindolizine-based compounds.

H. Oulyadi, P. Baran, A. Daïch, 2006, The Journal of organic chemistry.

Chemistry and Biology of HPAs: A Family of Ceramide Trafficking Inhibitors.

C. Santos, S. Ballereau, Y. Génisson, 2016, Chemistry.

General and versatile entry to 4,5-fused polycyclic imidazolones systems. Use of the tandem transposition/pi-cyclization of N-acyliminium species.

L. van Hijfte, A. Daïch, Anthony Pesquet, 2006, The Journal of organic chemistry.

Synthesis and reductive desulfurization of chiral non-racemic benzothienoindolizines. An efficient approach to a novel bioactive tylophorine alkaloid analogue and 6-phenylindolizidine

N. Prónayová, A. Daïch, S. Comesse, 2009 .

Indolylglycines Backbones in the Synthesis of Enantiopure 3,3-Spiroindolenines, Indolyl Tetracyclic Hemiaminals, and 3-Indolyl-maleimides Frameworks

J. Moncol’, A. Daïch, A. M. Lawson, 2019, European Journal of Organic Chemistry.

Acid-catalysed formation of tricyclic N,S-acetals in imidazolinone series based on the use of the unprecedented N-acyliminium ion cascade reaction involving transposition, heterocyclisation and pi-cyclisation.

B. Decroix, L. van Hijfte, A. Daïch, 2005, Organic & biomolecular chemistry.

Use of chiral-pool approach into epi-thieno analogues of the scarce bioactive phenanthroquinolizidine alkaloids

N. Prónayová, A. Daïch, A. M. Lawson, 2016, Tetrahedron.

Highly diastereoselective approach to novel tetrahydrofuran-fused indolizidinols: a one-step formation of three contiguous stereocenters

N. Prónayová, A. Daïch, P. Šafár̆, 2008 .

An enantioselective approach to synthesis of advanced chiral templates for the construction of indolic and indolizidinic alkaloids

A. Daïch, S. Comesse, Radouane Affani, 2009 .

New Efficient Eco‐Friendly Supported Catalysts for the Synthesis of Amides with Antioxidant and Anti‐Inflammatory Properties

C. Waterlot, Rogatien Charlet, M. Hechelski, 2020, ChemMedChem.

Biomass of ryegrass from field experiments: toward a cost-effective and efficient biosourced catalyst for the synthesis of Moclobemide

C. Waterlot, M. Hechelski, Alina Ghinet, 2020, Green Chemistry Letters and Reviews.

Tandem aza-Michael/spiro-ring closure sequence: access to a versatile scaffold and total synthesis of (±)-coerulescine

A. Daïch, A. M. Lawson, S. Comesse, 2013 .

En-route to scarce furo[3,2-f]indolizidines, -indolizidin-9-ols and their stable quaternary ammonium salts based on the stereoselective catalytic hydrogenation of furan nucleus

N. Prónayová, A. Daïch, A. M. Lawson, 2014 .

Expedient and practical synthesis of CERT-dependent ceramide trafficking inhibitor HPA-12 and its analogues.

P. Baran, A. Daïch, Daniela Moravčíková, 2011, Organic letters.

An easy access to the exocyclic lactams analogous of the central nervous system active tricyclic nitroxapine, mianserine and chlothiapine agents using N-acyliminium chemistry

A. Daïch, A. Hamid, A. Hadou, 2008 .

Diastereoselective access to hexahydro- and octahydrofuro[f]indolizines analogues of phenanthro[f]indolizidines alkaloids

F. Szemes, A. Daïch, V. Dalla, 2004 .

Exocyclic–Endocyclic N‐Acyliminium Ion Equilibration via an Intramolecular α‐Thioamidoalkylation in the Synthesis of Fused N,S‐Heterocyclic Systems: Some New Parameters

N. Hucher, A. Daïch, P. Netchitaïlo, 2005 .

Cazolobine, a New Sesquiterpene from Isolona hexaloba (Annonaceae)

E. Seguin, H. Oulyadi, A. Daïch, 2004 .

An alkaloid, two conjugate sesquiterpenes and a phenylpropanoid from Pachypodanthium confine Engl. and Diels.

P. Vérité, A. Daïch, Hilarion Mathouet, 2007, Phytochemistry.

Eaton's reagent-mediated domino π-cationic arylations of aromatic carboxylic acids to Iasi-red polymethoxylated polycyclic aromatic hydrocarbons: products with unprecedented biological activities as tubulin polymerization inhibitors.

P. Gautret, J. Hénichart, E. Bîcu, 2014, Chemistry.

Identification of Novel CERT Ligands as Potential Ceramide Trafficking Inhibitors

T. Levade, C. Santos, S. Ballereau, 2014, Chembiochem : a European journal of chemical biology.

Highly diastereoselective approach to novel phenylindolizidinols via benzothieno analogues of tylophorine based on reductive desulfurization of benzo[b]thiophene

N. Prónayová, A. Daïch, Ľ. Švorc, 2009 .

Quinoxalines,Bezodiazepines and Bezodiazocines Fused to Pyrrole and Isoindole via N-Acyliminium Ion Aromatic Cyclization

B. Decroix, P. Pigeon, A. Daïch, 2000 .

REGIOSELECTIVE CONVERSION OF LACTAM TO CORRESPONDING THIOLACTAM IN TETRAHYDROPYRROLO[1,2-A]THIENO[3,2-E] [1,3]DIAZEPINE

B. Decroix, A. Daïch, P. Netchitaïlo, 1996 .

Synthesis of a New Pyrrolo(1,3)diazepine: 4H‐Pyrrolo(1,2‐a)thieno(2,3‐ e) (1,3)diazepine.

B. Decroix, A. Daïch, P. Ohier, 1996 .

First synthesis and Diels-Alder reaction of thieno[2,3(3,2)-f]indolizines

B. Decroix, A. Daïch, P. Ohier, 1995 .

Development of SECheM Concept for Isolation and Chemical Modification of Gossypol Directly from Cienfuegosia digitata.

A. Daïch, M. Othman, M. V. Sidi Boune, 2017, Phytochemical analysis : PCA.

Structure-Based Kinetic Control in a Domino Process: A Powerful Tool Toward Molecular Diversity in Chromone Series.

J. Moncol’, A. Daïch, C. Denhez, 2017, The Journal of organic chemistry.

Structure and Mechanism Revision of a Catalyzed Cyclization of Benzaldehyde Bearing Alkyne-Nitrile.

J. Moncol’, Michal Šoral, A. Daïch, 2017, Organic letters.

Synthesis of 5-chloropyrrole carboxaldehydes from 5-oxopyrrolidine carboxamides

B. Decroix, A. Daïch, M. Othman, 1997 .

New and expeditious tandem sequence aza-Michael/intramolecular nucleophilic substitution route to substituted gamma-lactams: synthesis of the tricyclic core of (+/-)-martinellines.

A. Daïch, S. Comesse, M. Sanselme, 2008, The Journal of organic chemistry.

A Facile Access to 2-Ethynyl-1,4- dihydropyridines via Hantzsch Three- Component Reaction

F. Szemes, N. Prónayová, A. Daïch, 2003 .

New septanoside and 20-hydroxyecdysone septanoside derivative from Atriplex portulacoides roots with preliminary biological activities.

A. Daïch, H. Ben Jannet, M. Hamza, 2015, Bioorganic & medicinal chemistry letters.

An Easy Access to the Exocyclic Lactams Analogous of the Central Nervous System Active Tricyclic Nitroxapine, Mianserine and Chlothiapine Agents Using N‐Acyliminium Chemistry.

A. Daïch, A. Hamid, A. Hadou, 2009 .

Benefits of Ryegrass on Multicontaminated Soils Part 2: A Green Process to Provide Idrocilamide

C. Waterlot, M. Hechelski, B. Louvel, 2019, Sustainability.

Conformationally constrained 1,4-DHPs. A convenient route to bis-1,4-DHPs as a novel class of nitrogen compounds

A. Daïch, J. Kožíšek, M. Chudík, 2002 .

Facile access to 6‐substituted 1,4,5,7‐tetrahydropyrrolo[3,4‐b]‐pyridines via hantzsch type dimethyl 4‐aryl‐2‐formyl‐6‐methyl‐1,4‐dihydropyridine‐3,5‐dicarboxylates

B. Decroix, A. Daïch, S. Marchalin, 2000 .

Conformationally Constrained 1,4‐DHPs. A Convenient Route to Bis‐1,4‐DHPs as a Novel Class of Nitrogen Compounds.

A. Daïch, J. Kožíšek, M. Chudík, 2002 .

Facile Access to 6-Substituted 1,4,5,7-Tetrahydropyrrolo[3,4-b]pyridines via Hantzsch Type Dimethyl 4-Aryl-2-formyl-6-methyl-1,4-dihydropyridine-3,5-dicarboxylates.

B. Decroix, A. Daïch, S. Marchalin, 2001 .

From Conventional Lewis Acids to Heterogeneous Montmorillonite K10: Eco-Friendly Plant-Based Catalysts Used as Green Lewis Acids.

C. Waterlot, M. Hechelski, B. Louvel, 2018, ChemSusChem.

Novel Oleanolic Acid-Phtalimidines Tethered 1,2,3 Triazole Hybrids as Promising Antibacterial Agents: Design, Synthesis, In Vitro Experiments and In Silico Docking Studies

A. Harrath, Anis Romdhane, A. Daïch, 2023, Molecules.

Dichotomic Dearomatizations of Benzene vs Pyridine Rings of Sulfonyloxypyridine via (3 + 2) Cycloaddition.

Sami Ben Salah, A. Daïch, I. Chataigner, 2023, The Journal of organic chemistry.