Nigel A Swain

Novel indazole non-nucleoside reverse transcriptase inhibitors using molecular hybridization based on crystallographic overlays.

Catherine Burt, Chris Phillips, T. Knöchel, 2009, Journal of medicinal chemistry.

Highly potent and selective NaV1.7 inhibitors for use as intravenous agents and chemical probes.

Brian E Marron, Neil A Castle, Rubben Torella, 2017, Bioorganic & medicinal chemistry letters.

Discovery of Clinical Candidate 4-[2-(5-Amino-1H-pyrazol-4-yl)-4-chlorophenoxy]-5-chloro-2-fluoro-N-1,3-thiazol-4-ylbenzenesulfonamide (PF-05089771): Design and Optimization of Diaryl Ether Aryl Sulfonamides as Selective Inhibitors of NaV1.7.

P. A. Bradley, Brian E Marron, Ian K Gurrell, 2017, Journal of medicinal chemistry.

Voltage gated sodium channels as drug discovery targets

Sharan K Bagal, Brian E Marron, R. M. Owen, 2015, Channels.

Recent progress in sodium channel modulators for pain.

Sharan K Bagal, Brian E Marron, S. Bagal, 2014, Bioorganic & medicinal chemistry letters.