Tetsuo Takayama

发表

5-(1,3-Benzothiazol-6-yl)-4-(4-methyl-1,3-thiazol-2-yl)-1H-imidazole derivatives as potent and selective transforming growth factor-β type I receptor inhibitors.

H. Amada, Y. Sekiguchi, N. Ono, 2012, Bioorganic & medicinal chemistry.

Blocking S1P interaction with S1P₁ receptor by a novel competitive S1P₁-selective antagonist inhibits angiogenesis.

Y. Igarashi, Y. Ueda, R. Goitsuka, 2012, Biochemical and biophysical research communications.

Discovery of novel 2-[(4-hydroxy-6-oxo-2,3-dihydro-1H-pyridine-5-carbonyl)amino]acetic acid derivatives as HIF prolyl hydroxylase inhibitors for treatment of renal anemia.

H. Kakinuma, Sota Kato, Hiroki Takano, 2018, Bioorganic & medicinal chemistry letters.

Effects of the novel and potent lymphocyte-specific protein tyrosine kinase inhibitor TKM0150 on mixed lymphocyte reaction and contact hypersensitivity in mice

Masakazu Sato, Tetsuo Takayama, A. Takaoka, 2010, Arzneimittelforschung.

Isoquinoline derivatives as potent CRTH2 antagonists: design, synthesis and SAR.

Kazuhito Watanabe, Susumu Yamanobe, Y. Sekiguchi, 2013, Bioorganic & medicinal chemistry.

Isoquinoline derivatives as potent CRTH2 receptor antagonists: synthesis and SAR.

Kazuhito Watanabe, Y. Sekiguchi, T. Koami, 2012, Bioorganic & medicinal chemistry letters.

Amelioration of Collagen-Induced Arthritis by a Novel S1P1 Antagonist with Immunomodulatory Activities

Y. Igarashi, R. Goitsuka, K. Nakazawa, 2012, The Journal of Immunology.

Ring-fused pyrazole derivatives as potent inhibitors of lymphocyte-specific kinase (Lck): Structure, synthesis, and SAR.

H. Amada, T. Koami, Fumiyasu Shiozawa, 2010, Bioorganic & medicinal chemistry letters.

Pyrrole derivatives as potent inhibitors of lymphocyte-specific kinase: Structure, synthesis, and SAR.

H. Amada, Fumiyasu Shiozawa, Mayumi Endo, 2010, Bioorganic & medicinal chemistry letters.

Lymphopenia induced by a novel selective S1P(1) antagonist structurally unrelated to S1P.

Y. Igarashi, R. Goitsuka, Yasuyuki Fujii, 2012, Biochimica et biophysica acta.

Amelioration of Collagen-Induced Arthritis by a Novel S1P1 Antagonist with Immunomodulatory Activities

Y. Igarashi, R. Goitsuka, K. Nakazawa, 2012, The Journal of Immunology.

Amelioration of Collagen-Induced Arthritis by a Novel S1P1 Antagonist with Immunomodulatory Activities

R. Goitsuka, K. Nakazawa, Yasuyuki Fujii, 2012, The Journal of Immunology.

Isoquinoline derivatives as potent, selective, and orally active CRTH2 antagonists.

Kazuhito Watanabe, Y. Sekiguchi, Tetsuo Takayama, 2014, Chemical & pharmaceutical bulletin.

Effects of the novel and potent lymphocyte-specific protein tyrosine kinase inhibitor TKM0150 on mixed lymphocyte reaction and contact hypersensitivity in mice

Masakazu Sato, Tetsuo Takayama, A. Takaoka, 2010, Arzneimittelforschung.