J. Prasad

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Structure of a quinolone-stabilized cleavage complex of topoisomerase IV from Klebsiella pneumoniae and comparison with a related Streptococcus pneumoniae complex

I. Laponogov, J. Narasimhan, G. Skamrova, 2016, Acta crystallographica. Section D, Structural biology.

Nonpeptidic HIV protease inhibitors possessing excellent antiviral activities and therapeutic indices. PD 178390: a lead HIV protease inhibitor.

G. Zeikus, C. Humblet, E. Lunney, 1999, Bioorganic & medicinal chemistry.

A new class of anti-HIV-1 agents targeted toward the nucleocapsid protein NCp7: the 2,2'-dithiobisbenzamides.

J. Domagala, D. Hupe, R. Schultz, 1997, Bioorganic & medicinal chemistry.

Structure-activity and modeling studies of tryptophan-modified peptidyl antagonists of endothelin

A. Doherty, J. Dunbar, T. Sawyer, 1994 .

4-Hydroxy-2-pyridones: Discovery and evaluation of a novel class of antibacterial agents targeting DNA synthesis.

J. Narasimhan, A. Branstrom, Josephine Sheedy, 2017, Bioorganic & medicinal chemistry letters.

Hydroboration. LXXII: Hydroboration-oxidation of 1,4-epoxy-1,4-dihydronaphthalene with and without ring opening

H. Brown, J. Prasad, 1985 .

2,2′-dithiobisbenzamides derived from α-, β- and γ-amino acids possessing anti-HIV activities: synthesis and structure–activity relationship

D. P. Mack, W. J. Turner, J. Domagala, 1998 .

Novel Series of Achiral, Low Molecular Weight, and Potent HIV-1 Protease Inhibitors

James B. Dunbar, Daniel F. Ortwine, Donna Ferguson, 1994 .

Chiral synthesis via organoboranes. 17. Preparation of .alpha.-chiral .alpha.'-alkynyl ketones of high enantiomeric excess from optically pure organyl(1-alkynyl)borinic esters

M. Srebnik, H. Brown, A. Gupta, 1988 .

Hydroboration. 80. Preparation of trans-2-phenylcyclopentyl- and trans-2-phenylcyclohexylboronates of very high enantiomeric purities

R. Bakshi, H. Brown, A. Gupta, 1987 .

Chiral synthesis via organoboranes. 9. Crystalline chelates from borinic and boronic esters. A simple procedure for upgrading borinates and boronates to materials approaching 100% optical purity

H. Brown, J. Prasad, 1986 .

Chiral synthesis via organoboranes. 6. Hydroboration. 74. Asymmetric hydroboration of representative heterocyclic olefins with diisopinocampheylborane. Synthesis of heterocyclic boronates and heterocyclic alcohols of very high enantiomeric purity

H. Brown, J. Prasad, 1986 .

Synthesis of E- and Z-alkene dipeptide isosteres

D. Rich, J. Prasad, A. C. Bohnstedt, 1993 .

Addition of Allylic Metals to α-Aminoaldehydes. Application to the Synthesis of Statine, Ketomethylene and Hydroxyethylene Dipeptide Isosteres

D. Rich, J. Prasad, 1990 .

Thiocyanation of alkylanilines. A simple and efficient synthesis of thiosulfonates containing 2-aminobenzothiazole

J. Rubin, J. Prasad, A. Panapoulous, 2000 .

Synthesis of 5,6-dihydro-4-hydroxy-2-pyrones as HIV-1 protease inhibitors: the profound effect of polarity on antiviral activity.

E. Lunney, S. Hagen, J. Domagala, 1997, Journal of medicinal chemistry.

Synthesis of hydroxyethylene dipeptide isosteres that mimic A cyclic amino acid at the P1' subsite

D. Rich, J. Prasad, 1991 .

Mass spectra of some 2‐ and 3‐cycloalkenylfurans and ‐cycloalkenylthiophenes and their oxyderivatives

K. Wood, A. Gupta, J. Prasad, 1987 .

Hydroboration. 83. Asymmetric hydroboration of representative cis disubstituted and heterocyclic olefins with dicaranylboranes of high enantiomeric purity

H. Brown, J. Prasad, M. Zaidlewicz, 1988 .

Hydroboration of Heterocycles Olefins — A Versatile Route for the Synthesis of Both Racemic and Optically Active Heterocyclic Compounds

H. Brown, J. Prasad, 1987 .

Hydroboration. 75. Directive effects in the hydroboration of vinyl and propenyl heterocycles with representative hydroborating agents

H. Brown, J. Prasad, S. Zee, 1986 .

Hydroboration. 71. Hydroboration of representative heterocyclic olefins with borane-methyl sulfide, 9-borabicyclo[3.3.1]nonane, dicyclohexylborane, and disiamylborane. Synthesis of heterocyclic alcohols

H. Brown, J. Prasad, S. Zee, 1985 .

Vinylic organoboranes. 9. A general stereospecific synthesis of (Z)- and (E)-disubstituted alkenes via organoboranes

H. Brown, J. Prasad, D. Basavaiah, 1988 .

Chiral Synthesis via Organoboranes. 11. Hydroboration. 82. Asymmetric Hydroboration of 1-Heteroarylcycloalkenes with Monoisopinocampheylborane. Synthesis of trans-2-Heteroarylcycloalkyl Boronates and Derived Alcohols of Very High Enantiomeric Purity

H. Brown, A. Gupta, J. Prasad, 1988 .

Chiral Synthesis via Organoboranes. Part 9. Crystalline “Chelates” from Borinic and Boronic Esters. A Simple Procedure for Upgrading Borinates and Boronates to Materials Approaching 100% Optical Purity.

H. Brown, J. Prasad, 1987 .

Hydroboration. Part 74. Chiral Synthesis via Organoboranes. Part 6. Asymmetric Hydroboration of Representative Heterocyclic Olefins with Diisopinocampheylborane. Synthesis of Heterocyclic Boronates and Heterocyclic Alcohols of Very Hi

H. Brown, J. Prasad, 1986 .

Hydroboration. Part 80. Preparation of (trans-2-Phenylcyclopentyl)- and (trans-2-Phenylcyclohexyl)boronates of Very High Enantiomeric Purities.

R. Bakshi, H. Brown, A. Gupta, 1987 .

Chiral Synthesis via Organoboranes. Part 17. Preparation of α-Chiral α′-Alkynyl Ketones of High Enantiomeric Excess from Optically Pure Organyl(1-alkynyl)borinic Esters.

M. Srebnik, H. Brown, A. Gupta, 1988 .

Studies on the isomerization of substituted allyl alcohols over Raney nickel

J. Prasad, C. N. Pillai, 1984 .

Synthesis of E- and Z-Alkene Dipeptide Isosters.

D. Rich, J. Prasad, A. C. Bohnstedt, 2010 .

Isomerization of allyl alcohol in the presence of Raney nickel

A. Samuelson, J. Prasad, C. N. Pillai, 1982 .

Carbometallation: addition of organometallic compounds to isolated multiple bonds in functionally substituted compounds

J. Prasad, C. N. Pillai, 1983 .

Synthesis of heterocyclic thiosulfonates

J. Prasad, J. Vara Prasad, 2000 .

Addition of Allylic Metals to α-Amino Aldehydes. Application to the Synthesis of Statine, Ketomethylene, and Hydroxyethylene Dipeptide Isosteres.

D. Rich, J. Prasad, 1990 .

Nonpeptidic HIV protease inhibitors: 3-(S-benzyl substituted)-4-hydroxy-6-(phenyl substituted)-2H-pyran-2-one with an inverse mode of binding

D. Ferguson, E. Ellsworth, A. Pavlovsky, 1996 .

Nonpeptide inhibitors of HIV protease

S. Hagen, B. Tait, J. Prasad, 2000 .

New hydroxyethylamine HIV protease inhibitors that suppress viral replication.

R. Mueller, D. Rich, J. Green, 1992, Journal of medicinal chemistry.

4-hydroxy-5,6-dihydro-2H-pyran-2-ones.3. Bicyclic and hetero-aromatic ring systems as 3-position scaffolds to bind to S1' and S2' of the HIV-1 protease enzyme.

G. Zeikus, E. Lunney, S. Hagen, 1999, Bioorganic & medicinal chemistry letters.

Antibacterial oxazolidinones possessing a novel C-5 side chain. (5R)-trans-3-[3-Fluoro-4- (1-oxotetrahydrothiopyran-4-yl)phenyl]-2- oxooxazolidine-5-carboxylic acid amide (PF-00422602), a new lead compound.

J. Brieland, Ji-Young Kim, M. Huband, 2007, Journal of medicinal chemistry.

Effect of hydroxyl group configuration in hydroxyethylamine dipeptide isosteres on HIV protease inhibition. Evidence for multiple binding modes.

G. Marshall, R. Mueller, D. Rich, 1991, Journal of medicinal chemistry.

Chiral synthesis via organoboranes. XIX: The successful one-carbon homologation of heterocyclic boronate esters with high optical purity

H. Brown, A. Gupta, J. Prasad, 1989 .

Chiral Synthesis via Organoboranes. Part 19. The Successful One-Carbon Homologation of Heterocyclic Boronate Esters with High Optical Purity.

H. Brown, A. Gupta, J. Prasad, 1989 .

Hydroboration. 78. Reinvestigation of the hydroboration of N-substituted 3-pyrrolines. Preparation of N-benzyl-3-pyrrolidinol and N-benzyl-3-pyrrolidinylboronate of very high enantiomeric purity

H. Brown, A. Gupta, J. Prasad, 1986 .

A topliss tree analysis of the HIV-protease inhibitory activity of 6-phenyl-4-hydroxy-pyran-2-ones

Donna Ferguson, Elizabeth A. Lunney, C. J. Blankley, 1996 .