Celine Valant

Accelerated structure-based design of chemically diverse allosteric modulators of a muscarinic G protein-coupled receptor

J. Andrew McCammon, Arthur Christopoulos, Patrick M. Sexton, 2016, Proceedings of the National Academy of Sciences.

A Novel Mechanism of G Protein-coupled Receptor Functional Selectivity

Arthur Christopoulos, Nathan E Hall, Patrick M Sexton, 2008, Journal of Biological Chemistry.

Orthosteric/allosteric bitopic ligands: going hybrid at GPCRs.

Arthur Christopoulos, Patrick M Sexton, P. Sexton, 2009, Molecular interventions.

Allosteric modulators of the adenosine A1 receptor: synthesis and pharmacological evaluation of 4-substituted 2-amino-3-benzoylthiophenes.

Arthur Christopoulos, Patrick M Sexton, P. Sexton, 2009, Journal of medicinal chemistry.

Endogenous Allosteric Modulators of G Protein–Coupled Receptors

Arthur Christopoulos, Patrick M Sexton, P. Sexton, 2015, The Journal of Pharmacology and Experimental Therapeutics.