L. Bornaghi

发表

Design, synthesis, and biological evaluation of novel carbohydrate-based sulfamates as carbonic anhydrase inhibitors.

C. Supuran, A. Innocenti, D. Vullo, 2011, Journal of medicinal chemistry.

Sulfonamide linked neoglycoconjugates--a new class of inhibitors for cancer-associated carbonic anhydrases.

C. Supuran, A. Innocenti, D. Vullo, 2010, Journal of medicinal chemistry.

Orthogonally Protected Monosaccharide Building Blocks for Solid Phase Production of Diversity Oriented Libraries

W. Meutermans, M. West, N. Wimmer, 2010 .

A novel amino protecting group: DTPM

G. Dékány, L. Bornaghi, J. Papageorgiou, 2001 .

Anti-mycobacterial activity of a bis-sulfonamide.

Brendan L Wilkinson, A. Wright, T. Houston, 2007, Bioorganic & medicinal chemistry letters.

Microwave-accelerated cross-metathesis reactions of N-allyl amino acid substrates

S. Poulsen, L. Bornaghi, 2005 .

Structural Insights into Carbonic Anhydrase IX Isoform Specificity of Carbohydrate-Based Sulfamates

C. Supuran, D. Vullo, B. Mahon, 2014, Journal of medicinal chemistry.

A prodrug approach toward cancer-related carbonic anhydrase inhibition.

C. Supuran, D. Vullo, S. Charman, 2013, Journal of medicinal chemistry.

Synthesis of acylated glycoconjugates as templates to investigate in vitro biopharmaceutical properties.

David M. Shackleford, S. Charman, Marie Lopez, 2013, Bioorganic & medicinal chemistry letters.

Design and synthesis of thiourea compounds that inhibit transmembrane anchored carbonic anhydrases.

Brendan L Wilkinson, C. Supuran, A. Innocenti, 2012, Bioorganic & medicinal chemistry.

Inhibition of carbonic anhydrase isozymes with benzene sulfonamides incorporating thio, sulfinyl and sulfonyl glycoside moieties.

C. Supuran, A. Innocenti, D. Vullo, 2009, Bioorganic & medicinal chemistry letters.

Synthetic utility of glycosyl triazoles in carbohydrate chemistry

Brendan L Wilkinson, T. Houston, S. Poulsen, 2006 .

Synthesis and structure-activity relationships of novel benzene sulfonamides with potent binding affinity for bovine carbonic anhydrase II.

P. Healy, S. Poulsen, L. Bornaghi, 2005, Bioorganic & medicinal chemistry letters.

Microwave-accelerated Fischer glycosylation

S. Poulsen, L. Bornaghi, 2005 .

Carbonic anhydrase inhibitors: inhibition of isozymes I, II, and IX with triazole-linked O-glycosides of benzene sulfonamides.

Brendan L Wilkinson, C. Supuran, A. Innocenti, 2007, Journal of medicinal chemistry.

Targeting hypoxic tumor cell viability with carbohydrate-based carbonic anhydrase IX and XII inhibitors.

C. Supuran, J. Pouysségur, Marie Lopez, 2011, Journal of medicinal chemistry.

Synthesis of sulfonamide-bridged glycomimetics.

Sally-Ann Poulsen, H. Driguez, Marie Lopez, 2011, The Journal of organic chemistry.

Dde as a Protecting Group for Carbohydrate Synthesis

M. West, I. Toth, L. Bornaghi, 2006 .

Transfer reactions catalyzed by cyclodextrin glucosyltransferase using 4-thiomaltosyl and C-maltosyl fluorides as artificial donors.

H. Driguez, J. Mallet, J. Utille, 1997, Carbohydrate research.

Synthesis of cyclic oligomers of a modified sugar amino acid utilising dynamic combinatorial chemistry

Brendan L Wilkinson, M. Kiefel, S. Poulsen, 2004 .

Methyl 2,3,4-tri-O-acetyl-1-azido-1-deoxy-β-d-glucopyranuronate at room temperature

Brendan L Wilkinson, P. Healy, T. Houston, 2005 .

Synthesis of N-Propargyl Iminosugar Scaffolds for Compound Library Generation using Click Chemistry

Brendan L Wilkinson, P. Healy, Marie Lopez, 2010 .

A novel class of carbonic anhydrase inhibitors: glycoconjugate benzene sulfonamides prepared by "click-tailing".

Brendan L Wilkinson, C. Supuran, A. Innocenti, 2006, Journal of medicinal chemistry.

Fragment-based drug discovery of carbonic anhydrase II inhibitors by dynamic combinatorial chemistry utilizing alkene cross metathesis.

Sally-Ann Poulsen, Laurent F Bornaghi, S. Poulsen, 2006, Bioorganic & medicinal chemistry.

Stereoselective Synthesis of Highly Functionalized Arabinosyl Nucleosides through Application of an N-Nitro Protecting Group.

S. Poulsen, L. Bornaghi, D. Hilko, 2018, The Journal of organic chemistry.

Synthesis of 5‐Alkynyl Substituted 2ʹ‐Arabinosyl 2ʹ‐Halogenated Uridine Nucleosides

S. Poulsen, L. Bornaghi, D. Hilko, 2019, Current protocols in nucleic acid chemistry.

Galactan biosynthesis in snails: a comparative study of β-(1 → 6) galactosyltransferases from Helix pomatia and Biomphalaria glabrata

L. Kröger, J. Thiem, L. Bornaghi, 2000, Journal of Comparative Physiology B.

Cyclic secondary sulfonamides: unusually good inhibitors of cancer-related carbonic anhydrase enzymes.

C. Supuran, T. Peat, D. Vullo, 2014, Journal of medicinal chemistry.

Synthesis of S-glycosyl primary sulfonamides.

Marie Lopez, S. Poulsen, L. Bornaghi, 2009, The Journal of organic chemistry.

Carbonic anhydrase inhibitors with dual-tail moieties to match the hydrophobic and hydrophilic halves of the carbonic anhydrase active site.

C. Supuran, T. Peat, D. Vullo, 2015, Journal of medicinal chemistry.

Inhibition of membrane-associated carbonic anhydrase isozymes IX, XII and XIV with a library of glycoconjugate benzenesulfonamides.

Brendan L Wilkinson, C. Supuran, A. Innocenti, 2007, Bioorganic & medicinal chemistry letters.

Regioselective Fucosylation Using L-Galactosyltransferase from Helix pomatia

L. Keating, J. Thiem, L. Bornaghi, 1998 .

Enzymic synthesis of cyclothiomaltins

G. Schulz, L. Dijkhuizen, H. Driguez, 1997 .

Selective Monoesterification of Malonic Acid Catalyzed by Boric Acid

Stephan M Levonis, T. Houston, L. Bornaghi, 2007 .

Synthesis of sulfonamide-conjugated glycosyl-amino acid building blocks.

Marie Lopez, S. Poulsen, L. Bornaghi, 2014, Carbohydrate research.

N-Cinnamoyl-l-phenylalanine methyl ester

P. Healy, S. Poulsen, L. Bornaghi, 2007, Acta crystallographica. Section E, Structure reports online.

Targeting hypoxic tumor cell viability with carbohydrate-based carbonic anhydrase IX and XII inhibitors.

C. Supuran, J. Pouysségur, Marie Lopez, 2011, Journal of medicinal chemistry.

Methyl 2,3,4-tri-O-acetyl-1-azido-1-deoxy-β-d-glucopyranuronate at room temperature

Brendan L Wilkinson, P. Healy, T. Houston, 2005 .