K. Washizuka

发表

Discovery of a novel series of biphenyl benzoic acid derivatives as potent and selective human beta3-adrenergic receptor agonists with good oral bioavailability. Part I.

M. Sakurai, Y. Matsumura, M. Imanishi, 2008, Journal of medicinal chemistry.

Discovery of Novel Spiroindoline Derivatives as Selective Tankyrase Inhibitors.

T. Umehara, M. Shirouzu, H. Seimiya, 2019, Journal of medicinal chemistry.

Novel generation and cycloaddition of N-silylated azomethine ylides from α-silylimidates and trifluorosilane

I. Ryu, S. Minakata, M. Komatsu, 1999 .

Discovery of a novel, potent and selective human beta3-adrenergic receptor agonist.

H. Kayakiri, Y. Tomishima, H. Hamashima, 2005, Bioorganic & medicinal chemistry letters.

Synthesis and biological activity of a novel squalene epoxidase inhibitor, FR194738.

K. Washizuka, M. Sawada, H. Okumura, 2004, Bioorganic & Medicinal Chemistry Letters.

Novel generation of azomethine imines from α-silylnitrosamines by 1,4-silatropic shift and their cycloaddition

I. Ryu, S. Minakata, M. Komatsu, 1999 .

Generation and cycloaddition of polymer-supported azomethine imines: traceless synthesis of pyrazole derivatives from α-silylnitrosoamide derivatives bound to resin

I. Ryu, S. Minakata, M. Komatsu, 2000 .

Palladium-Catalyzed Double and Single Carbonylations of β-Amino Alcohols. Selective Synthesis of Morpholine-2,3-diones and Oxazolidin-2-ones and Applications for Synthesis of α-Oxo Carboxylic Acids

K. Washizuka, Y. Imada, S. Murahashi, 1996 .

Synthesis and antibacterial activity of novel 4-pyrrolidinylthio carbapenems. Part III:

M. Sakurai, T. Kamimura, K. Washizuka, 1999 .

Design and Discovery of an Orally Efficacious Spiroindolinone-based Tankyrase Inhibitor for the Treatment of Colon Cancer.

T. Umehara, M. Shirouzu, H. Seimiya, 2020, Journal of medicinal chemistry.

Discovery of novel series of benzoic acid derivatives containing biphenyl ether moiety as potent and selective human beta(3)-adrenergic receptor agonists: Part IV.

Nobuhiro Yamamoto, Minoru Sakurai, Yutaka Nakajima, 2008, Bioorganic & medicinal chemistry letters.

Effect of FR194738, a potent inhibitor of squalene epoxidase, on cholesterol metabolism in HepG2 cells.

J Seki, J. Seki, K. Washizuka, 2001, European journal of pharmacology.

Discovery of highly potent and selective biphenylacylsulfonamide-based beta3-adrenergic receptor agonists and evaluation of physical properties as potential overactive bladder therapies: part 5.

M. Sakurai, Y. Matsumura, M. Imanishi, 2009, Journal of medicinal chemistry.

Discovery of a novel series of benzoic acid derivatives as potent and selective human beta3 adrenergic receptor agonists with good oral bioavailability. 3. Phenylethanolaminotetraline (PEAT) skeleton containing biphenyl or biphenyl ether moiety.

M. Sakurai, Y. Matsumura, M. Imanishi, 2008, Journal of medicinal chemistry.

Discovery of a novel series of biphenyl benzoic acid derivatives as highly potent and selective human beta3 adrenergic receptor agonists with good oral bioavailability. Part II.

M. Sakurai, Y. Matsumura, M. Imanishi, 2008, Journal of medicinal chemistry.