G. Makara

发表

Synthesis of Condensed Heterocycles by the Gould–Jacobs Reaction in a Novel Three-Mode Pyrolysis Reactor

F. Darvas, G. Dormán, J. Gerencsér, 2015 .

A reagent-based strategy for the design of large combinatorial libraries: A preliminary experimental validation

E. Wintner, G. Makara, H. Nash, 2004, Molecular Diversity.

Derivatization Design of Synthetically Accessible Space for Optimization: In Silico Synthesis vs Deep Generative Design.

I. Szabó, G. Makara, G. Pőcze, 2021, ACS medicinal chemistry letters.

Synthesis, molecular modeling, and evaluation of nonphenolic indole analogs of mycophenolic acid.

R. Bernacki, G. Makara, P. Pera, 2004, Bioorganic & medicinal chemistry.

Bound conformations for ligands for G-protein coupled receptors

G. Marshall, R. Ragno, R. Arimoto, 1999, Letters in Peptide Science.

Hit discovery and hit-to-lead approaches.

György M Keseru, Gergely M Makara, G. Keserű, 2006, Drug discovery today.

Activation of carboxylic acids by Burgess reagent: an efficient route to acyl ureas and amides

P. Lan, G. Makara, J. Athanasopoulos, 2006 .

Versatile solid-phase synthesis of trisubstituted 1H-pyrido[2,3-d]pyrimidin-4-ones and related heterocycles.

G. Makara, M. Richards, P. Schell, 2005, Journal of combinatorial chemistry.

Michael addition of amines to vinyl sulfonamides on solid support

G. Makara, Yao Ma, 2001 .

Solid-phase synthesis of 3-alkylamino-1,2,4-triazoles.

G. Makara, Yao Ma, Laura Margarida, 2002, Organic letters.

On the conformation of tiazofurin analogues.

G. Keserű, G. Makara, 1997, Journal of medicinal chemistry.

Nuclear magnetic resonance and molecular modeling study on mycophenolic acid: implications for binding to inosine monophosphate dehydrogenase.

G. Keserű, G. Makara, M. Kajtár-Peredy, 1996, Journal of medicinal chemistry.

A single vessel protocol for the efficient formation of amide bonds from esters and lactones

G. Makara, N. Kawahata, Jeseca Brookes, 2002 .

A facile synthesis of 3-substituted pipecolic acids, chimeric amino acids

Garland R. Marshall, Gergely M. Makara, G. Marshall, 1997 .

Synthesis of bicyclic pyrimidine derivatives as ATP analogues.

E. Wintner, W. Ewing, G. Makara, 2001, The Journal of organic chemistry.

The influence of lead discovery strategies on the properties of drug candidates

György M. Keserü, Gergely M. Makara, G. Keserü, 2009, Nature Reviews Drug Discovery.

Rhodopsin-transducin interface: studies with conformationally constrained peptides.

G. Marshall, R. Arimoto, G. Makara, 2001, Biophysical journal.

An Improved Synthesis of 5,7-Dimethoxy-4-methylphthalide, A Key Intermediate in the Synthesis of Mycophenolic Acid

G. Makara, K. Klubek, W. Anderson, 1996 .

AN EFFICIENT SYNTHESIS OF 5,7-DIMETHOXY-4-METHYLPHTHALIDE, A KEY INTERMEDIATE IN THE SYNTHESIS OF MYCOPHENOLIC ACID

G. Makara, W. Anderson, 1995 .

An efficient method to access 2-substituted benzimidazoles under solvent-free conditions

F. A. Romero, P. Lan, G. Makara, 2008 .

Combinatorial synthesis of substituted biaryls and heterocyclic arylamines.

G. Makara, S. Berk, Yao Ma, 2004, Journal of combinatorial chemistry.

Improving success rates for lead generation using affinity binding technologies

Gergely M Makara, G. Makara, John Athanasopoulos, 2005, Current Opinion in Biotechnology.

Hit-to-Lead Optimization and Discovery of 5-((5-([1,1'-Biphenyl]-4-yl)-6-chloro-1H-benzo[d]imidazol-2-yl)oxy)-2-methylbenzoic Acid (MK-3903): A Novel Class of Benzimidazole-Based Activators of AMP-Activated Protein Kinase.

Margaret S. Wu, Q. Dang, D. Mackenna, 2017, Journal of medicinal chemistry.

Identification of a small molecule nonpeptide active site beta-secretase inhibitor that displays a nontraditional binding mode for aspartyl proteases.

M Katharine Holloway, Gergely M Makara, Zhongguo Chen, 2004, Journal of medicinal chemistry.

Label-free high-throughput screening via mass spectrometry: a single cystathionine quantitative method for multiple applications.

Claude Dufresne, Gergely M Makara, Bernard K. Choi, 2009, Assay and drug development technologies.

- Fragment-Based Methods in Drug Design

György M. Keserü, Márton Vass, Gergely M. Makara, 2015 .

On sampling of fragment space.

Gergely M Makara, G. Makara, 2007, Journal of medicinal chemistry.

An efficient solid-phase synthesis of 3-alkylamino-1,2,4-oxadiazoles

G. Makara, P. Schell, K. Hanson, 2002 .

Measuring molecular similarity and diversity: total pharmacophore diversity.

G. Makara, G M Makara, 2001, Journal of medicinal chemistry.

Synthesis and modeling studies with monocyclic analogues of mycophenolic acid.

T. Boehm, G. Makara, W. Anderson, 1996, Journal of medicinal chemistry.

Label-free high-throughput screening via mass spectrometry: a single cystathionine quantitative method for multiple applications.

Bernard K. Choi, N. Geoghagen, Kristian K. Jensen, 2009, Assay and drug development technologies.