Valeria Famiglini

发表

Inhibition of dengue virus replication by novel inhibitors of RNA-dependent RNA polymerase and protease activities

A. Coluccia, R. Silvestri, G. La Regina, 2017, Journal of enzyme inhibition and medicinal chemistry.

New Inhibitors of Indoleamine 2,3-Dioxygenase 1: Molecular Modeling Studies, Synthesis, and Biological Evaluation.

A. Coluccia, R. Silvestri, G. La Regina, 2016, Journal of medicinal chemistry.

New 6- and 7-heterocyclyl-1H-indole derivatives as potent tubulin assembly and cancer cell growth inhibitors.

C. Martini, A. Coluccia, R. Silvestri, 2018, European journal of medicinal chemistry.

Discovery of 1,1'-Biphenyl-4-sulfonamides as a New Class of Potent and Selective Carbonic Anhydrase XIV Inhibitors.

C. Supuran, A. Coluccia, D. Vullo, 2015, Journal of medicinal chemistry.

Focus on Chirality of HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors

R. Silvestri, Valeria Famiglini, 2016, Molecules.

Toward highly potent cancer agents by modulating the C-2 group of the arylthioindole class of tubulin polymerization inhibitors.

Y. Ni, E. Novellino, B. Maresca, 2013, Journal of medicinal chemistry.

Indolylarylsulfones, a fascinating story of highly potent human immunodeficiency virus type 1 non-nucleoside reverse transcriptase inhibitors

R. Silvestri, Valeria Famiglini, 2018, Antiviral chemistry & chemotherapy.

Exploring the first Rimonabant analog-opioid peptide hybrid compound, as bivalent ligand for CB1 and opioid receptors

E. Novellino, A. Mollica, R. Silvestri, 2017, Journal of enzyme inhibition and medicinal chemistry.

Arylsulfone-based HIV-1 non-nucleoside reverse transcriptase inhibitors.

A. Coluccia, A. Brancale, R. Silvestri, 2013, Future medicinal chemistry.

Venting-while-heating microwave-assisted synthesis of 3-arylthioindoles.

R. Silvestri, G. La Regina, F. Piscitelli, 2012, ACS combinatorial science.

Design, synthesis, and biological evaluation of 1-phenylpyrazolo[3,4-e]pyrrolo[3,4-g]indolizine-4,6(1H,5H)-diones as new glycogen synthase kinase-3β inhibitors.

E. Novellino, A. Coluccia, A. Brancale, 2013, Journal of medicinal chemistry.

New Indole Tubulin Assembly Inhibitors Cause Stable Arrest of Mitotic Progression, Enhanced Stimulation of Natural Killer Cell Cytotoxic Activity, and Repression of Hedgehog-Dependent Cancer.

E. Novellino, L. Di Marcotullio, C. Martini, 2015, Journal of medicinal chemistry.

New pyrrole derivatives with potent tubulin polymerization inhibiting activity as anticancer agents including hedgehog-dependent cancer.

Ettore Novellino, Andrea Brancale, Ruoli Bai, 2014, Journal of medicinal chemistry.

Indolylarylsulfones carrying a heterocyclic tail as very potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors.

E. Novellino, A. Coluccia, A. Brancale, 2014, Journal of Medicinal Chemistry.

New indolylarylsulfones as highly potent and broad spectrum HIV-1 non-nucleoside reverse transcriptase inhibitors.

E. Novellino, B. Clotet, A. Coluccia, 2014, European journal of medicinal chemistry.

N-Pyrrylarylsulfones with High Therapeutic Potential

R. Silvestri, S. Castellano, Valeria Famiglini, 2017, Molecules.

Mitotic cell death induction by targeting the mitotic spindle with tubulin-inhibitory indole derivative molecules

E. Cundari, A. Coluccia, R. Silvestri, 2017, Oncotarget.

Chiral Indolylarylsulfone Non-Nucleoside Reverse Transcriptase Inhibitors as New Potent and Broad Spectrum Anti-HIV-1 Agents.

C. Limatola, E. Novellino, A. Coluccia, 2017, Journal of medicinal chemistry.

An High-Throughput In Vivo Screening System to Select H3K4-Specific Histone Demethylase Inhibitors

E. Cundari, A. Coluccia, R. Silvestri, 2014, PloS one.

3-Aroyl-1,4-diarylpyrroles Inhibit Chronic Myeloid Leukemia Cell Growth through an Interaction with Tubulin.

A. Coluccia, A. Brancale, R. Silvestri, 2017, ACS medicinal chemistry letters.

New 1-phenyl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamides inhibit hepatitis C virus replication via suppression of cyclooxygenase-2.

A. Coluccia, C. Zamperini, M. Botta, 2015, European journal of medicinal chemistry.

β-catenin knockdown promotes NHERF1-mediated survival of colorectal cancer cells: implications for a double-targeted therapy

I. Fournier, A. Coluccia, R. Silvestri, 2018, Oncogene.

New nitrogen containing substituents at the indole-2-carboxamide yield high potent and broad spectrum indolylarylsulfone HIV-1 non-nucleoside reverse transcriptase inhibitors.

E. Novellino, B. Clotet, A. Coluccia, 2012, Journal of medicinal chemistry.

Chiral Indolylarylsulfone Non-Nucleoside Reverse Transcriptase Inhibitors as New Potent and Broad Spectrum Anti-HIV-1 Agents.

C. Limatola, E. Novellino, A. Coluccia, 2017, Journal of medicinal chemistry.

New pyrrole derivatives with potent tubulin polymerization inhibiting activity as anticancer agents including hedgehog-dependent cancer.

E. Novellino, L. Di Marcotullio, A. Brancale, 2014, Journal of medicinal chemistry.

Toward highly potent cancer agents by modulating the C-2 group of the arylthioindole class of tubulin polymerization inhibitors.

Y. Ni, E. Novellino, B. Maresca, 2013, Journal of medicinal chemistry.

3-Aroyl-1-arylpyrroles: a New Class of Potent Inhibitors of Tubulin Polymerization.

E. Novellino, R. Silvestri, E. Hamel, 2014 .