Hao Liu

发表

Efficient conversion of a nonselective norepinephrin reuptake inhibitor into a dual muscarinic antagonist-β₂-agonist for the treatment of chronic obstructive pulmonary disease.

P. Glossop, L. Jones, Rachel Osborne, 2011, Journal of medicinal chemistry.

Ibrexafungerp: an orally active β-1,3-glucan synthesis inhibitor.

P. Liberator, M. Motyl, M. Peel, 2020, Bioorganic & medicinal chemistry letters.

MK-5204: An orally active β-1,3-glucan synthesis inhibitor.

P. Liberator, M. Motyl, M. Peel, 2020, Bioorganic & medicinal chemistry letters.

Design, synthesis, and antifungal activity of novel cinnamon–pyrazole carboxamide derivatives

Xianhai Lv, Zi-Li Ren, H. Cao, 2018, Drug development research.

Discovery of a stable macrocyclic o-aminobenzamide Hsp90 inhibitor which significantly decreases tumor volume in a mouse xenograft model.

J. Levin, J. Lucas, J. Bloom, 2011, Bioorganic & medicinal chemistry letters.

Discovery of a macrocyclic o-aminobenzamide Hsp90 inhibitor with heterocyclic tether that shows extended biomarker activity and in vivo efficacy in a mouse xenograft model.

J. Levin, J. Lucas, J. Bloom, 2011, Bioorganic & medicinal chemistry letters.

Macrocyclic lactams as potent Hsp90 inhibitors with excellent tumor exposure and extended biomarker activity.

J. Levin, J. Lucas, J. Bloom, 2011, Bioorganic & medicinal chemistry letters.

Design and SAR of macrocyclic Hsp90 inhibitors with increased metabolic stability and potent cell-proliferation activity.

J. Levin, J. Bloom, Jennifer M. Golas, 2011, Bioorganic & medicinal chemistry letters.

Novel orally active inhibitors of β-1,3-glucan synthesis derived from enfumafungin.

P. Liberator, M. Motyl, M. Peel, 2015, Bioorganic & medicinal chemistry letters.

Design, synthesis, and biological evaluations of phenylpropiolic acid derivatives as novel GPR40 agonists.

Mingyao Liu, Weiqiang Lu, Hao Liu, 2018, European journal of medicinal chemistry.

A cell-based screen for inhibitors of protein folding and degradation

Roseann Petersen, Jennifer M. Golas, K. Arndt, 2010, Cell stress & chaperones (Print).

A bioactivity-oriented modification strategy for SDH inhibitors with superior activity against fungal strains.

Xianhai Lv, Hao Liu, Wei Wang, 2020, Pesticide biochemistry and physiology.

Novel coumarin-pyrazole carboxamide derivatives as potential topoisomerase II inhibitors: Design, synthesis and antibacterial activity.

Xianhai Lv, Zi-Li Ren, M. Chu, 2018, European journal of medicinal chemistry.

Design and synthesis of novel tacrine-dipicolylamine dimers that are multiple-target-directed ligands with potential to treat Alzheimer's disease.

Shan He, Bin Zhang, Ning Wang, 2021, Bioorganic chemistry.

Novel coumarin-thiazolyl ester derivatives as potential DNA gyrase Inhibitors: Design, synthesis, and antibacterial activity.

Xianhai Lv, Hao Liu, Dongguo Xia, 2020, Bioorganic chemistry.

Discovery of novel multi-substituted benzo-indole pyrazole schiff base derivatives with antibacterial activity targeting DNA gyrase.

Xianhai Lv, H. Cao, Hao Liu, 2020, Bioorganic chemistry.

Discovery of Novel Triazole-Containing Pyrazole Ester Derivatives as Potential Antibacterial Agents

Xianhai Lv, Li Wang, Zi-Li Ren, 2019, Molecules.

Design, synthesis and biological evaluation of novel flavone Mannich base derivatives as potential antibacterial agents

Xianhai Lv, Zi-Li Ren, H. Cao, 2018, Molecular Diversity.

A potential anticancer agent 1,2-di(quinazolin-4-yl)diselane induces apoptosis in non-small-cell lung cancer A549 cells

J. Qian, Yinjiu Huang, Xiaomei Hu, 2015, Medicinal Chemistry Research.

A potential anticancer agent 1,2-di(quinazolin-4-yl)diselane induces apoptosis in non-small-cell lung cancer A549 cells

Yinjiu Huang, Xiaomei Hu, Hao Liu, 2014, Medicinal Chemistry Research.

Design, Synthesis and Biological Evaluation of Novel Pyrazole Sulfonamide Derivatives as Potential AHAS Inhibitors.

Xianhai Lv, Li Wang, Zi-Li Ren, 2018, Chemical and pharmaceutical bulletin.

Preparation and In Vivo Antinociceptive Behavior of Four New 2‐Amino‐6‐trifuromethoxybenzothiazole Carboxylic Acid Derivatives

Qichun Zhang, T. Lu, Xianglong Wu, 2019, ChemistrySelect.

Design, synthesis, and biological evaluation of indole-based hydroxamic acid derivatives as histone deacetylase inhibitors.

Mingyao Liu, Xiufeng Pang, Yu Wen, 2021, European journal of medicinal chemistry.

Synthesis and biological evaluation of antifungal derivatives of enfumafungin as orally bioavailable inhibitors of β-1,3-glucan synthase.

P. Liberator, G. J. Pacofsky, M. Peel, 2012, Bioorganic & medicinal chemistry letters.

Design, synthesis and antibacterial activity of a class of novel molecular engineering analogues of Tachyplesin I

Shengnan Song, Haotian Sun, Hao Liu, 2022, Phytochemistry Letters.

Anti-oligomerization sheet molecules: Design, synthesis and evaluation of inhibitory activities against α-synuclein aggregation.

Hao Liu, S. Bai, Ji Xu, 2019, Bioorganic & medicinal chemistry.

Optimization of N-Phenylpropenoyl-l-amino Acids as Potent and Selective Inducible Nitric Oxide Synthase Inhibitors for Parkinson's Disease.

W. Ye, F. Xiong, Xiao-Qi Zhang, 2021, Journal of medicinal chemistry.