M. Lasne

发表

(-)-Cytisine and derivatives: synthesis, reactivity, and applications.

J. Baudoux, J. Rouden, M. Lasne, 2014, Chemical reviews.

Microspheres based on inulin for the controlled release of serine protease inhibitors: preparation, characterization and in vitro release.

M. Prud'homme, I. Dez, M. Lasne, 2003, Journal of controlled release : official journal of the Controlled Release Society.

Synthesis of a cytisine/epibatidine hybrid: a radical approach

P. Lestage, R. Bureau, J. Rouden, 2010 .

Synthesis of a [2-pyridinyl-18F]-labelled fluoro derivative of (-)-cytisine as a candidate radioligand for brain nicotinic alpha4beta2 receptor imaging with PET.

J. Bénavidès, F. Dollé, H. Valette, 2003, Bioorganic & medicinal chemistry.

2- and 4-[18F]Fluorophenols from Baeyer-Villiger Oxidation of [18F]Fluorophenylketones and [18F]Fluorobenzaldehydes

L. Barré, M. Lasne, F. Gourand, 1995 .

New trends in molecular imaging of tumor angiogenesis.

G. Déléris, T. Berthelot, M. Lasne, 2008, Anti-cancer agents in medicinal chemistry.

Synthesis of no carrier added [1-11C]propenoic acid and derivatives.

L. Barré, M. Lasne, P. Cairon, 1992, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

Syntheses of piperidine and perhydroazepine derivatives, precursors of two selective antagonists of muscarinic M2 receptors: AF-DX 384 and its perhydroazepine isomer

M. Lasne, Cécile Perrio-Huard, C. Ducandas, 1996 .

Rapid synthesis of aliphatic amides by reaction of carboxylic acids, Grignard reagent and amines: application to the preparation of [11C]amides

C. Aubert, M. Lasne, Cécile Huard-Perrio, 1997 .

Synthesis and biological evaluation of novel fluoro and iodo quinoline carboxamides as potential ligands of NK-3 receptors for in vivo imaging studies.

L. Barré, I. Bennacef, M. Lasne, 2004, Bioorganic & medicinal chemistry.

Synthesis of P,N-2,2′-biphenyl derivatives with central chirality

L. Jean, J. Rouden, M. Lasne, 2010 .

Reactivity of (-)-cytisine and derivatives towards palladium salts. X-ray characterization of a new palladium complex of (-)-cytisine

M. Hervieu, B. Tinant, J. Muzart, 2006 .

The rotational constants of acetylene-d

J. Burie, G. Wlodarczak, J. Demaison, 1989 .

Oxidation of aromatic lithium thiolates into sulfinate salts: an attractive entry to aryl sulfones labeled with carbon-11.

M. Lasne, C. Perrio, S. Perrio, 2006, The Journal of organic chemistry.

Debenzylation of tertiary amines using phosgene or triphosgene: an efficient and rapid procedure for the preparation of carbamoyl chlorides and unsymmetrical ureas. Application in carbon-11 chemistry.

M. Ibazizène, J. Rouden, M. Lasne, 2003, The Journal of organic chemistry.

Synthesis of analogues of (-)-cytisine for in vivo studies of nicotinic receptors using positron emission tomography.

J. Rouden, M. Lasne, V. Tadino, 2000, Organic letters.

Reductive amination of carboxylic acids and [11C]magnesium halide carboxylates

C. Aubert, M. Lasne, Cécile Perrio-Huard, 2000 .

Palladium-mediated N-arylation of heterocyclic diamines: insights into the origin of an unusual chemoselectivity.

L. Jean, J. Maddaluno, J. Rouden, 2007, The Journal of organic chemistry.

Synthesis of [11C]‐S21007 a novel 5HT3 partial agonist as a potential tracer for PET studies

L. Barré, S. Rault, S. Guillouet, 1996 .

Identification of 9-fluoro substituted (-)-cytisine derivatives as ligands with high affinity for nicotinic receptors.

P. Lestage, J. Rouden, M. Lasne, 2010, Bioorganic & medicinal chemistry letters.

Chemistry of β +-Emitting Compounds Based on Fluorine-18

C. Crouzel, L. Barré, F. Dollé, 2002 .

Efficient Deracemization of Pipecolic Acid Amides through Enantioselective Protonation of Their Lithium Enolates: Insights into the Origin of the Transferred Proton

J. Maddaluno, J. Rouden, M. Lasne, 2009 .

Enantioselective decarboxylation–reprotonation of an α-amino malonate derivative as a route to optically enriched cyclic α-amino acid

J. Rouden, M. Lasne, L. Rogers, 2003 .

Lithiation of functionalized fluoroquinolines: synthesis of dihalo-2-phenylquinoline-4-carboxamides and in vitro evaluation as NK-3 receptor ligands for medical imaging studies.

L. Barré, I. Bennacef, M. Lasne, 2004, The Journal of organic chemistry.

Fluorine‐18 Chemistry for Molecular Imaging with Positron Emission Tomography

F. Dollé, B. Kuhnast, M. Lasne, 2008 .

Rapid synthesis of quinoline-4-carboxylic acid derivatives from arylimines and 2-substituted acrylates or acrylamides under indium(III) chloride and microwave activations. Scope and limitations of the reaction.

O. Parisel, M. Lasne, C. Perrio, 2005, Organic & biomolecular chemistry.

Synthesis of a-fluorinated-a,a-difunctionalized sulfides and sulfones

M. Lasne, J. Pommelet, C. Jouen, 1996 .

Palladium‐Mediated Cross‐Coupling Reaction of an Heteroaryl‐Imidoyl Chloride and Primary Amines — Preparation of a New Ligand of Serotoninergic Receptors.

A. Bernard, J. Rouden, M. Lasne, 1999 .

Metal-Free SN2′ Decarboxylative Rearrangement of β-Keto Esters

J. Baudoux, X. Franck, J. Rouden, 2011 .

Palladium-mediated arylation of 3-aminopiperidines and 3-aminopyrrolidines.

L. Jean, J. Maddaluno, J. Rouden, 2004, Journal of Organic Chemistry.

Asymmetric Malonic and Acetoacetic Acid Syntheses – A Century of Enantioselective Decarboxylative Protonations

J. Baudoux, J. Rouden, M. Lasne, 2008 .

Organocatalyzed route to enantioenriched pipecolic esters: decarboxylation of an aminomalonate hemiester

T. Seitz, J. Baudoux, J. Rouden, 2006 .

Preparation of tertiary amides from carbamoyl chlorides and organocuprates.

T. Seitz, J. Rouden, M. Lasne, 2004, Organic letters.

Cross-coupling reactions of carbamoyl chlorides and Grignard reagents: a new rapid synthesis of tertiary amides

J. Rouden, M. Lasne, Laurent Lemoucheux, 2000 .

Studies toward labeling cytisine with [11C]phosgene: rapid synthesis of a delta-lactam involving a new chemoselective lithiation-annulation method.

T. Seitz, J. Rouden, M. Lasne, 2004, The Journal of organic chemistry.

(9R)‐9‐Amino‐9‐Deoxyquinidine

J. Rouden, M. Lasne, 2009 .

Highly enantioselective decarboxylative protonation of alpha-aminomalonates mediated by thiourea cinchona alkaloid derivatives: access to both enantiomers of cyclic and acyclic alpha-aminoacids.

J. Rouden, M. Lasne, Mukkanti Amere, 2007, Organic letters.

Synthesis of BINOL derived phosphorodithioic acids as new chiral Brønsted acids and an improved synthesis of 3,3′-disubstituted H8-BINOL derivatives

J. Rouden, M. Lasne, J. Blanchet, 2009 .

A NMR and theoretical study of the aggregates between alkyllithium and chiral lithium amides: control of the topology through a single asymmetric center.

C. Giessner-Prettre, A. Harrison-Marchand, J. Valnot, 2002, Journal of the American Chemical Society.

New Synthetic Developments of the [4π + 2π]Cycloreversion

M. Lasne, J. Ripoll, 1985 .

Enantioselective tautomerization of a new metastable enol

M. Lasne, L. Duhamel, Ruediger Henze, 1997 .

Environmentally benign metal-free decarboxylative aldol and Mannich reactions

Rémi Legay, J. Baudoux, J. Rouden, 2010 .

3-trifluoromethanesulfonamido-pyrrolidine: a general organocatalyst for anti-selective mannich reactions.

J. Rouden, M. Lasne, J. Blanchet, 2008, Organic letters.

Chiral 3-aminopyrrolidines as a rigid diamino scaffold for organocatalysis and organometallic chemistry

J. Maddaluno, J. Rouden, M. Lasne, 2010 .

A convenient route to 1-benzyl 3-aminopyrrolidine and 3-aminopiperidine

L. Jean, J. Maddaluno, J. Rouden, 2001 .

A rapid and convenient synthesis of β-proline

J. Rouden, M. Lasne, J. Blanchet, 2007 .

NMR in chiral polypeptide liquid crystals: the problem of amines

J. Courtieu, A. Meddour, L. Jean, 2007 .

4-Toluenesulfonic acid: an environmentally benign catalyst for Nazarov cyclizations

J. Rouden, M. Lasne, J. Blanchet, 2008 .

The radiosynthesis of No‐carrier added [1‐11C]allyl alcohol evidence for the formation of a new reducing species: Lithium aluminium hydride — vinylmagnesium bromide

L. Barré, M. Lasne, P. Cairon, 1994 .

Retrodienic reactions. Part 2. Vinyl- and propenyl-phosphines: synthesis by flash vacuum thermolysis and characterization

M. Lasne, J. Ripoll, A. Thuillier, 1988 .

5,6-dihydropyridine: synthesis and characterization

J. Guillemin, M. Lasne, J. Ripoll, 1985 .

Construction of functionalized/substituted bipyridines by means of Negishi cross-coupling reactions. Formal synthesis of (±)-cytisine

J. Rouden, M. Lasne, P. Nshimyumukiza, 2001 .

Pyrrolidines bearing a quaternary α-stereogenic center. Part 1: Synthesis of analogs of ABT-418, a powerful nicotinic agonist

T. Giard, M. Lasne, J. Plaquevent, 1999 .

Syntheses of R and S isomers of AF-DX 384, a selective antagonist of muscarinic M2 receptors.

F. Dauphin, P. Desbène, C. Morin, 2000, Bioorganic & Medicinal Chemistry.

Enantioselective protonation of amide enolates derived from piperidine-2-carboxylic acid

M. Lasne, Juliette Martin, J. Plaquevent, 1997 .

Determination of the moment of inertia of methyl groups: analysis of the millimeterwave spectra of cis-propanal and methylthioethyne

G. Wlodarczak, J. Demaison, B. P. Eijck, 1987 .

Rapid Synthesis of α,β Unsaturated Iodides: Iodination Under Vacuum with Solid Diphosphorus Tetraiodide

D. Villemin, M. Lasne, P. Cairon, 1990 .

Cooked mussels contaminated by Dinophysis sp.: a source of okadaic acid.

J. Vernoux, M. Lasne, J. Frémy, 1994, Natural toxins.

Functionalization through lithiation of (S)-N-(1-phenylpropyl)-2-phenylquinoline-4-carboxamide. Application to the labeling with carbon-11 of NK-3 receptor antagonist SB 222200.

L. Barré, I. Bennacef, M. Lasne, 2007, The Journal of organic chemistry.

International Isotope Society. Abstracts of the Xth I.I.S. (UK Group) Symposium. Current themes in Isotopic chemistry.

D. F. White, G. Antoni, B. Långström, 2001 .

Regio- and diastereoselective functionalization of (−)-cytisine

J. Rouden, M. Lasne, Nicolas Houllier, 2006 .

Regio- and diastereoselective functionalization of (−)-cytisine: an unusual N–C acyl migration

J. Rouden, M. Lasne, D. Cahard, 2002 .

Rapid synthesis of N,N′-disubstituted piperazines. Application to the preparation of No carrier added 1-(4-[18F]fluorophenyl)piperazine and of an [18F]-selective ligand of serotoninergic receptors (5HT2 antagonist)

L. Barré, M. Lasne, M. Collins, 1992 .

Synthesis and regional rat brain distribution of [11C]MDL 72222: a 5HT3 receptor antagonist.

J. Baron, G. Bonvento, L. Barré, 1992, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

[11C]Carbamoyl chlorides: An easy access from [11C]phosgene and tertiary amines

M. Ibazizène, J. Rouden, M. Lasne, 2001 .

Synthesis and biological evaluation of halogenated naphthyridone carboxamides as potential ligands for in vivo imaging studies of substance P receptors.

L. Barré, D. Guilloteau, P. Emond, 2003, Bioconjugate chemistry.

Synthesis and radiosynthesis with a positron emitter of EP 00652218, a potent antagonist of NK1 receptor, and of a fluoro analog for in vivo evaluation of the substance P receptor by pet

L. Barré, D. Guilloteau, F. Dauphin, 2001 .

Radioiodinated analogs of EP 00652218 for the exploration of the tachykinin NK1 receptor by spect

L. Barré, D. Guilloteau, F. Dauphin, 2001 .

The radiosynthesis of [N-methyl-11C]-sertraline.

V. Pike, D. Turton, M. Lasne, 1989, International journal of radiation applications and instrumentation. Part A, Applied radiation and isotopes.

Preparation of [18F]RP 62203, a selective ligand for the study of serotonin receptors (5-HT2) by rapid “in situ” piperazine formation

L. Barré, M. Lasne, M. Collins, 1994 .

Specific in vivo binding in the rat brain of [18F]RP 62203: a selective 5-HT2A receptor radioligand for positron emission tomography.

J. Baron, F. Dauphin, P. Mickala, 1996, Nuclear medicine and biology.

Origin of the detrimental effect of lithium halides on an enantioselective nucleophilic alkylation of aldehydes.

A. Harrison-Marchand, J. Valnot, N. Duguet, 2007, The Journal of organic chemistry.