R. Heckendorn

发表

2-Methyl-6-(phenylethynyl)-pyridine (MPEP), a potent, selective and systemically active mGlu5 receptor antagonist

Roland Heckendorn, Hans Allgeier, Fabrizio Gasparini, 1999, Neuropharmacology.

Synthesis and preliminary pharmacological evaluation of the four stereoisomers of (2S)-2-(2'-phosphono-3'-phenylcyclopropyl)glycine, the first class of 3'-substituted trans C1'-2'-2-(2'-phosphonocyclopropyl)glycines.

F. Gasparini, P. Flor, G. Costantino, 2007, Bioorganic & medicinal chemistry.

Addition of phenylmagnesium bromide to an amino-cyano-thiophene

R. Heckendorn, A. Gagneux, 1973 .

[Oxetane from A-nor-steroides: 2-alpha, 5-oxido-A-nor-5-alpha-cholestane, 2-beta, 5-oxido-A-nor-5-beta-cholestane and 2-alpha-ethyl-2-beta,2'-oxido-A-nor-5-alpha-cholestane].

R. Heckendorn, C. Tamm, 1968, Helvetica chimica acta.

SYNTHESIS OF (1,2,4)TRIAZOLO)1,5‐A)QUINAZOLINES. EFFECT OF SUBSTITUENT ORIENTATION ON CARBON‐13 CHEMICAL SHIFT. PART III. DEDUCTION OF THE CONFORMATION OF SUBSTITUENTS BY CARBON‐13 NMR SPECTROSCOPY

T. Winkler, R. Heckendorn, 1980 .

Azomalonate Syntheses Part II. Synthesis and Reactivity of Novel 1,2,4‐Triazin‐5‐one Derivatives

R. Heckendorn, 1990 .

Novel Heterocycles by the Malonic Ester Variation of the Japp‐Klingemann Reaction

R. Heckendorn, 2010 .

Azomalonic Ester Syntheses. Part I. One‐Step Synthesis of Triazolo[1,4]benzodiazepines from Azomalonates. Preparation of Novel Polyaza Tricycles from Diethyl (2‐Chloroacetamido)malonate

R. Heckendorn, 1987 .

Photoreactions of benzonitrile with cyclic enol ethers

J. Mattay, R. Heckendorn, Jan Runaink, 1987 .

Synthesis of trans-10,11-dihydro-10,11-dihydroxy-5H-dibenz[b,f]azepine-5-carboxamide, a major metabolite of carbamazepine

R. Heckendorn, 1987 .

Perhydro-1,3-diazepine-2,4-diones by cyclization of 4-ureidobutyric acids with thionyl chloride: A reinvestigation

T. Winkler, R. Heckendorn, 2000 .

[3H]CGP 61594, the first photoaffinity ligand for the glycine site of NMDA receptors

M. Honer, H. Mohler, M. Pozza, 1999, Neuropharmacology.

CGP 37849 and CGP 39551: novel and potent competitive N‐methyl‐d‐aspartate receptor antagonists with oral activity

G. Fagg, M. Pozza, M. Schmutz, 1990, British journal of pharmacology.

Synthese der 2,5‐Diole des A‐nor‐5α‐Cholestans und A‐nor‐5β‐Cholestans

R. Heckendorn, C. Tamm, 1967 .

Differentiation of glycine antagonist sites of N-methyl-D-aspartate receptor subtypes. Preferential interaction of CGP 61594 with NR1/2B receptors.

H. Monyer, P. Seeburg, M. Honer, 1998, The Journal of biological chemistry.

The competitive NMDA receptor antagonists CGP 37849 and CGP 39551 are potent, orally-active anticonvulsants in rodents

G. Fagg, H. Riezen, K. Klebs, 1990, Naunyn-Schmiedeberg's Archives of Pharmacology.

Molecular distinction of three N-methyl-D-aspartate-receptor subtypes in situ and developmental receptor maturation demonstrated with the photoaffinity ligand 125I-labeled CGP 55802A.

D. Laurie, P. Seeburg, T. Marti, 1993, Proceedings of the National Academy of Sciences of the United States of America.

Synthesis, Structure, and Reactivity of Secosteroids Containing a Medium‐Sized Ring. Part 36. Transannular photocyclization of some unsaturated 5,10‐secosteroidal ketones: A reevaluation

R. Heckendorn, J. Kalvoda, H. Fuhrer, 1995 .

CGP 37849 / CGP 39551: The First Competitive NMDA Receptor Antagonists Suitable for Oral Antiepileptic Therapy

G. Fagg, K. Klebs, M. Schmutz, 1991 .

Photoaffinity labeling of the NMDA receptor.

T. Marti, H. Mohler, D. Benke, 1993, European journal of pharmacology.