G. E. Jagdmann

发表

Discovery of allosteric potentiators for the metabotropic glutamate 2 receptor: synthesis and subtype selectivity of N-(4-(2-methoxyphenoxy)phenyl)-N-(2,2,2- trifluoroethylsulfonyl)pyrid-3-ylmethylamine.

D. Schoepp, T. Large, M. Baez, 2003, Journal of medicinal chemistry.

SAR study of a subtype selective allosteric potentiator of metabotropic glutamate 2 receptor, N-(4-phenoxyphenyl)-N-(3-pyridinylmethyl)ethanesulfonamide.

D. Schoepp, D. Barda, Michael P Johnson, 2004, Bioorganic & medicinal chemistry letters.

A Mild Efficient Procedure for the Conversion of Carboxylic Acid Esters to Primary Amides Using Formamide/Methanolic Sodium Methoxide

G. E. Jagdmann, H. R. Munson, T. Gero, 1990 .

Chemical synthesis and characterization of epicatechin glucuronides and sulfates: bioanalytical standards for epicatechin metabolite identification.

M. V. Van Zandt, P. Beckett, G. E. Jagdmann, 2013, Journal of natural products.

Enantioselective synthesis of orthogonally protected (2R,3R)-(−)-epicatechin derivatives, key intermediates in the de novo chemical synthesis of (−)-epicatechin glucuronides and sulfates

P. Beckett, G. E. Jagdmann, H. Schroeter, 2013 .

Two efficient syntheses of (±)-anti-N-benzyl-3-amino-4-hydroxyhexahydroazepine

P. Hughes, G. E. Jagdmann, Hongdan Hu, 1995 .

Discovery of (R)-2-amino-6-borono-2-(2-(piperidin-1-yl)ethyl)hexanoic acid and congeners as highly potent inhibitors of human arginases I and II for treatment of myocardial reperfusion injury.

E. Howard, A. Mitschler, M. V. Van Zandt, 2013, Journal of medicinal chemistry.

.alpha.-Amino carbanions. Preparation, metalation, and alkylation of enamidines. Synthesis of piperidine and pyrrolidine natural products and homologation of carbonyl compounds

A. Meyers, P. Edwards, G. E. Jagdmann, 1985 .

Enamidines. Versatile vehicles for homologation of carbonyl compounds

A. Meyers, G. E. Jagdmann, 1982 .

Thallium in organic synthesis. 60. 2,6-Diaryl-3,7-dioxabicyclo[3.3.0]octane-4,8-dione lignans by oxidative dimerization of 4-alkoxycinnamic acids with thallium(III) trifluoroacetate or cobalt(III) trifluoride

A. Mckillop, G. E. Jagdmann, K. Steliou, 1981 .

Discovery of N-substituted 3-amino-4-(3-boronopropyl)pyrrolidine-3-carboxylic acids as highly potent third generation inhibitors of human arginase I and II.

A. Pyle, O. Potapova, E. Howard, 2019, Journal of medicinal chemistry.

Metabotropic glutamate 2 receptor potentiators: receptor modulation, frequency-dependent synaptic activity, and efficacy in preclinical anxiety and psychosis model(s)

E. Nisenbaum, D. McKinzie, D. Schoepp, 2005, Psychopharmacology.

Small Molecule Antagonists of the RIG-I Innate Immune Receptor.

A. Pyle, O. Potapova, G. E. Jagdmann, 2020, ACS chemical biology.

Synthesis and biological evaluation of conformationally constrained bicyclic and tricyclic balanol analogues as inhibitors of protein kinase C

J. Mendoza, G. E. Jagdmann, P. Gosnell, 1995 .

RING SIZE EFFECT IN THE PKC INHIBITORY ACTIVITIES OF PERHYDROAZEPINE ANALOGS OF BALANOL

S. Hall, Y. Lai, G. E. Jagdmann, 1995 .

Increasing the cellular PKC inhibitory activity of balanol: A study of ester analogs

G. E. Jagdmann, James W. Darges, Heidi M. Crane, 1995 .

Potent and selective PKC inhibitory 5-membered ring analogs of balanol with replacement of the carboxamide moiety

J. Lampe, G. E. Jagdmann, J. Darges, 1996 .

Synthesis and protein kinase inhibitory activity of balanol analogues with modified benzophenone subunits.

M. G. Johnson, M. P. Lynch, Philip F. Hughes, 2002, Journal of medicinal chemistry.

Thallium in organic synthesis. 53. Simple procedures for the replacement of a phenolic OH group by N = NAr, N = O, H, NH2, and C substituents

A. Mckillop, G. E. Jagdmann, E. Taylor, 1978 .

Small molecules that target group II introns are potent antifungal agents

R. L. Adams, A. Pyle, M. V. Van Zandt, 2018, Nature Chemical Biology.

Novel PKC inhibitory analogs of balanol with replacement of the ester functionality

S. Hall, Hong Hu, Y. Lai, 1995 .