D. Lin

Citric acid cycle intermediates as ligands for orphan G-protein-coupled receptors

Jinhai Gao, Zhulun Wang, W. He, 2004, Nature.

Identification and Molecular Characterization of Two Closely Related G Protein-coupled Receptors Activated by Prokineticins/Endocrine Gland Vascular Endothelial Growth Factor*

Qun Zhou, C. Bullock, F. Ehlert, 2002, The Journal of Biological Chemistry.

GPR40 Is Necessary but Not Sufficient for Fatty Acid Stimulation of Insulin Secretion In Vivo

T. Alquier, V. Poitout, M. Latour, 2007, Diabetes.

A Potent Class of GPR40 Full Agonists Engages the EnteroInsular Axis to Promote Glucose Control in Rodents

Sean P. Brown, S. Wong, B. Shan, 2012, PloS one.

Discovery of AM-6226: A Potent and Orally Bioavailable GPR40 Full Agonist That Displays Efficacy in Nonhuman Primates.

Sean P. Brown, S. Wong, Liusheng Zhu, 2018, ACS medicinal chemistry letters.

Discovery of AM-1638: A Potent and Orally Bioavailable GPR40/FFA1 Full Agonist.

Sean P. Brown, S. Wong, J. Medina, 2012, ACS medicinal chemistry letters.

AMG 837: a potent, orally bioavailable GPR40 agonist.

Ying Sun, J. Reagan, Rajiv Sharma, 2012, Bioorganic & medicinal chemistry letters.