G. Koether

4-aryl piperazine and piperidine amides as novel mGluR5 positive allosteric modulators.

J. McCauley, Minli Zhang, James Kang, 2010, Bioorganic & medicinal chemistry letters.

Discovery of novel, orally active dual NK1/NK2 antagonists.

W. Rumsey, P. Bernstein, J. Albert, 2001, Bioorganic & medicinal chemistry letters.

Design and optimization of cyclized NK1 antagonists with controlled atropisomeric properties

J. Evenden, W. Rumsey, B. Masek, 2004 .

Design, synthesis, and SAR of tachykinin antagonists: modulation of balance in NK(1)/NK(2) receptor antagonist activity.

W. Rumsey, P. Bernstein, J. Albert, 2002, Journal of medicinal chemistry.

Application of fragment-based lead generation to the discovery of novel, cyclic amidine beta-secretase inhibitors with nanomolar potency, cellular activity, and high ligand efficiency.

Gianni Chessari, Mark Sylvester, Rutger H A Folmer, 2007, Journal of medicinal chemistry.

Naphtho[2,1-b][1,5] and [1,2-f][1,4]oxazocines as selective NK1 antagonists.

W. Rumsey, B. Masek, P. Bernstein, 2004, Bioorganic & medicinal chemistry.