B. Gilmour

发表

Synthesis and evaluation of 1,2,4-methyltriazines as mGluR5 antagonists.

H. Navarro, F. Carroll, Jeremy P. Olson, 2011, Organic & biomolecular chemistry.

Synthesis and Evaluation of Metabotropic Glutamate Receptor Subtype 5 Antagonists Based on Fenobam().

S. Mascarella, H. Navarro, F. Carroll, 2011, ACS medicinal chemistry letters.

Toward the Development of Bivalent Ligand Probes of Cannabinoid CB1 and Orexin OX1 Receptor Heterodimers.

B. Thomas, B. Gilmour, Yanan Zhang, 2014, ACS medicinal chemistry letters.

Effect of the 3- and 4-Methyl Groups on the Opioid Receptor Properties of N-Substituted trans-3,4-Dimethyl-4-(3-hydroxyphenyl)piperidines

James B. Thomas, S. Runyon, L. Brieaddy, 2014, Journal of medicinal chemistry.

Trace amine-associated receptor 1 is a stereoselective binding site for compounds in the amphetamine class.

G. Miller, A. Lewin, B. Gilmour, 2011, Bioorganic & medicinal chemistry.

Identification of neuropeptide S antagonists: structure-activity relationship studies, X-ray crystallography, and in vivo evaluation.

J. Deschamps, T. Fennell, R. Snyder, 2014, ACS chemical neuroscience.

Inhibition of NFκB by the natural product Withaferin A in cellular models of Cystic Fibrosis inflammation

R. Maitra, B. Gilmour, M. Porter, 2009, Journal of Inflammation.

Diarylureas as Allosteric Modulators of the Cannabinoid CB1 Receptor: Structure–Activity Relationship Studies on 1-(4-Chlorophenyl)-3-{3-[6-(pyrrolidin-1-yl)pyridin-2-yl]phenyl}urea (PSNCBAM-1)

B. Thomas, J. Wiley, B. Gilmour, 2014, Journal of medicinal chemistry.

Truncated Orexin Peptides: Structure-Activity Relationship Studies.

B. Thomas, B. Gilmour, N. German, 2013, ACS medicinal chemistry letters.

Substituted tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

B. Thomas, B. Gilmour, D. Harris, 2013, Journal of medicinal chemistry.

Synthesis, pharmacological characterization, and structure-activity relationship studies of small molecular agonists for the orphan GPR88 receptor.

Xi-Ping Huang, B. Roth, X. Zhang, 2014, ACS chemical neuroscience.

Discovery of N-{4-[(3-hydroxyphenyl)-3-methylpiperazin-1-yl]methyl-2-methylpropyl}-4-phenoxybenzamide analogues as selective kappa opioid receptor antagonists.

I. Carroll, James B. Thomas, S. Runyon, 2013, Journal of medicinal chemistry.

The importance of the 6- and 7-positions of tetrahydroisoquinolines as selective antagonists for the orexin 1 receptor.

S. Runyon, B. Thomas, B. Gilmour, 2015, Bioorganic & medicinal chemistry.

Effect of 1-substitution on tetrahydroisoquinolines as selective antagonists for the orexin-1 receptor.

S. Runyon, B. Thomas, B. Gilmour, 2015, ACS chemical neuroscience.

Diaryl urea analogues of SB-334867 as orexin-1 receptor antagonists.

S. Runyon, B. Thomas, B. Gilmour, 2011, Bioorganic & medicinal chemistry letters.

α1 and α2 Ca2+ channel subunit expression in human neuronal and small cell carcinoma cells

S. Froehner, B. Gilmour, M. Morton, 1994, FASEB journal : official publication of the Federation of American Societies for Experimental Biology.

Amiodarone and its putative metabolites fail to activate wild type hTAAR1.

H. Navarro, A. Lewin, B. Gilmour, 2009, Bioorganic & medicinal chemistry letters.

Validation of a High-Throughput Calcium Mobilization Assay for the Human Trace Amine-Associated Receptor 1

B. Blough, B. Gilmour, A. Decker, 2020, SLAS discovery : advancing life sciences R & D.

A Rapid Functional Assay for the Human Trace Amine-Associated Receptor 1 Based on the Mobilization of Internal Calcium

H. Navarro, A. Lewin, B. Gilmour, 2006, Journal of biomolecular screening.

Synthesis and pharmacological evaluation of phenylethynyl[1,2,4]methyltriazines as analogues of 3-methyl-6-(phenylethynyl)pyridine.

S. Mascarella, H. Navarro, F. Carroll, 2007, Journal of medicinal chemistry.

Identification of N-[(5-{[(4-Methylphenyl)sulfonyl]amino}-3-(trifluoroacetyl)-1H-indol-1-yl)acetyl]-l-leucine (NTRC-824), a Neurotensin-like Nonpeptide Compound Selective for the Neurotensin Receptor Type 2

L. Gendron, James B. Thomas, S. Runyon, 2014, Journal of medicinal chemistry.

A new synthesis of the ORL-1 antagonist 1-[(3R,4R)-1-cyclooctylmethyl-3-hydroxymethyl-4-piperidinyl]-3-ethyl-1,3-dihydro-2H-benzimidazol-2-one (J-113397) and activity in a calcium mobilization assay.

J. Deschamps, James B. Thomas, H. Navarro, 2008, Bioorganic & medicinal chemistry.

Multiple binding sites for myogenic regulatory factors are required for expression of the acetylcholine receptor gamma-subunit gene.

G. Fanger, P. Gardner, B. Gilmour, 1991, The Journal of biological chemistry.

A biomimetic multicellular model of the airways using primary human cells.

Sonia Grego, Scott H Randell, Katelyn L Sellgren, 2014, Lab on a chip.

The amide linker in nonpeptide neurotensin receptor ligands plays a key role in calcium signaling at the neurotensin receptor type 2.

James B. Thomas, S. Runyon, R. Wiethe, 2015, Bioorganic & medicinal chemistry letters.

Identification of N-{[6-chloro-4-(2,6-dimethoxyphenyl)quinazolin-2-yl]carbonyl}-l-leucine (NTRC-808), a novel nonpeptide chemotype selective for the neurotensin receptor type 2.

James B. Thomas, S. Runyon, R. Wiethe, 2015, Bioorganic & medicinal chemistry letters.

Identification of 1-({[1-(4-Fluorophenyl)-5-(2-methoxyphenyl)-1H-pyrazol-3-yl]carbonyl}amino)cyclohexane Carboxylic Acid as a Selective Nonpeptide Neurotensin Receptor Type 2 Compound

L. Gendron, James B. Thomas, S. Runyon, 2014, Journal of medicinal chemistry.

Kappa opioid mediation of cannabinoid effects of the potent hallucinogen, salvinorin A, in rodents

J. Warner, H. Navarro, F. Carroll, 2010, Psychopharmacology.

Synthetic studies of neoclerodane diterpenes from Salvia divinorum: semisynthesis of salvinicins A and B and other chemical transformations of salvinorin A.

W. Harding, P. Kannan, H. Navarro, 2006, Journal of natural products.

Identifying structural features on 1,1-diphenyl-hexahydro-oxazolo[3,4-a]pyrazin-3-ones critical for Neuropeptide S antagonist activity.

S. Runyon, H. Navarro, B. Gilmour, 2008, Bioorganic & medicinal chemistry letters.

The effect of 1-substitution on tetrahydroisoquinolines as selective antagonists for the Orexin-1 receptor

S. Runyon, B. Thomas, B. Gilmour, 2015 .

Electrical Activity Suppresses Nicotinic Acetylcholine Receptor γ Subunit Promoter Activity

K. Chahine, P. Gardner, D. Goldman, 1995 .

The identification of nonpeptide neurotensin receptor partial agonists from the potent antagonist SR48692 using a calcium mobilization assay.

James B. Thomas, H. Navarro, B. Gilmour, 2009, Bioorganic & medicinal chemistry letters.

Journal of Inflammation Inhibition of Nfκb by the Natural Product Withaferin a in Cellular Models of Cystic Fibrosis Inflammation

R. Maitra, B. Gilmour, Melissa A. Porter, 2022 .