Erica M. Haslach

Identification of Tetrapeptides from a Mixture Based Positional Scanning Library That Can Restore nM Full Agonist Function of the L106P, I69T, I102S, A219V, C271Y, and C271R Human Melanocortin-4 Polymorphic Receptors (hMC4Rs)

Clemencia Pinilla, Michael A. Walters, Richard A. Houghten, 2014, Journal of medicinal chemistry.

Structure-activity relationships (SAR) of melanocortin and agouti-related (AGRP) peptides.

C. Haskell-Luevano, Erica M. Haslach, Anamika Singh, 2010, Advances in experimental medicine and biology.

Beta-turn secondary structure and melanocortin ligands.

C. Haskell-Luevano, Erica M. Haslach, Jay W Schaub, 2009, Bioorganic & medicinal chemistry.

Human β-Defensin 1 and β-Defensin 3 (Mouse Ortholog mBD14) Function as Full Endogenous Agonists at Select Melanocortin Receptors.

Mark D. Ericson, R. Speth, B. Smeester, 2018, Journal of medicinal chemistry.

Discovery of Molecular Interactions of the Human Melanocortin-4 Receptor (hMC4R) Asp189 (D189) Amino Acid with the Endogenous G-Protein-Coupled Receptor (GPCR) Antagonist Agouti-Related Protein (AGRP) Provides Insights to AGRP's Inverse Agonist Pharmacology at the hMC4R.

Mark D. Ericson, R. Speth, K. Freeman, 2021, ACS chemical neuroscience.

Discovery of Mixed Pharmacology Melanocortin-3 Agonists and Melanocortin-4 Receptor Tetrapeptide Antagonist Compounds (TACOs) Based on the Sequence Ac-Xaa1-Arg-(pI)DPhe-Xaa4-NH2.

Radleigh G. Santos, M. Giulianotti, R. Houghten, 2017, Journal of medicinal chemistry.