V. Garaj

发表

The inhibitory potency of local anesthetics on NMDA receptor signalling depends on their structural features.

M. Hollmann, C. Gronwald, K. Hahnenkamp, 2012, European journal of pharmacology.

QSAR ANALYSES OF BENZENESULFONAMIDE INHIBITORS OF CARBONIC ANHYDRASE INHIBITORS WITH 1,3,5-TRIAZINE MOIETY

V. Garaj, Tomus Lv, 2008 .

Photoswitching hydrazones based on benzoylpyridine.

A. Marini, J. Filo, V. Garaj, 2019, Physical chemistry chemical physics : PCCP.

Effect of dielectric medium on angiotensin converting enzyme inhibitors binding to Zn2+

V. Garaj, Martin Šramko, Július Šille, 2010 .

ORIGINAL PAPER Effect of dielectric medium on angiotensin converting enzyme inhibitors binding to Zn 2

V. Garaj, 2010 .

7-Dialkylaminocoumarin Oximates: Small Molecule Fluorescent “Turn-On” Chemosensors for Low-Level Water Content in Aprotic Organic Solvents

A. Gáplovský, J. Filo, V. Garaj, 2017, Molecules.

Synthesis and Antimicrobial Evaluation of 6‐Alkylamino‐N‐phenylpyrazine‐2‐carboxamides

L. Naesens, P. Jílek, M. Doležal, 2015, Chemical biology & drug design.

Optimal detection of cholinesterase activity in biological samples: modifications to the standard Ellman's assay.

E. Krejci, V. Garaj, D. Dingová, 2014, Analytical biochemistry.

Novel sulfonamides incorporating 1,3,5-triazine and amino acid structural motifs as inhibitors of the physiological carbonic anhydrase isozymes I, II and IV and tumor-associated isozyme IX.

C. Supuran, A. Angeli, Silvia Bua, 2018, Bioorganic chemistry.

Novel 1,3,5-Triazinyl Aminobenzenesulfonamides Incorporating Aminoalcohol, Aminochalcone and Aminostilbene Structural Motifs as Potent Anti-VRE Agents, and Carbonic Anhydrases I, II, VII, IX, and XII Inhibitors

C. Supuran, M. Brázdová, J. Jampílek, 2021, International journal of molecular sciences.

Carbonic anhydrase inhibitors: novel sulfonamides incorporating 1,3,5-triazine moieties as inhibitors of the cytosolic and tumour-associated carbonic anhydrase isozymes I, II and IX.

Giuseppe Fasolis, Alessio Innocenti, Vladimir Garaj, 2005, Bioorganic & medicinal chemistry letters.

Sulfonamides incorporating 1,3,5-triazine moieties selectively and potently inhibit carbonic anhydrase transmembrane isoforms IX, XII and XIV over cytosolic isoforms I and II: Solution and X-ray crystallographic studies.

Vladimir Garaj, Andrea Scozzafava, Alfonso Maresca, 2011, Bioorganic & medicinal chemistry.

Isatinphenylsemicarbazones as efficient colorimetric sensors for fluoride and acetate anions - anions induce tautomerism.

A. Gáplovský, V. Garaj, M. Cigáň, 2014, Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy.

Coumarin phenylsemicarbazones: sensitive colorimetric and fluorescent “turn-on” chemosensors for low-level water content in aprotic organic solvents

J. Gašpar, H. Stankovičová, V. Garaj, 2016 .

Venlafaxine Chiral Separation by Capillary Electrophoresis Using Cyclodextrin Derivatives as Chiral Selector and Experimental Design Method Optimization

Andreea Milan, Gabriel Hancu, Daniela Lupu, 2020, Symmetry.

Enantioseparation of citalopram enantiomers by capillary electrophoresis: Method development through experimental design and computational modeling.

V. Garaj, D. Muntean, G. Hancu, 2020, Chirality.

Thermodynamics of binding of angiotensin-converting enzyme inhibitors to enzyme active site model

Milan Remko, M. Remko, Martin Šramko, 2008 .

Thermodynamics of binding of Zn2+ to carbonic anhydrase inhibitors

M. Remko, V. Garaj, 2003 .

Novel sulfonamide incorporating piperazine, aminoalcohol and 1,3,5-triazine structural motifs with carbonic anhydrase I, II and IX inhibitory action.

C. Supuran, D. Vullo, J. Csöllei, 2018, Bioorganic chemistry.

Small-molecule coumarin fluorescent pH probes for extremely acidic conditions

H. Stankovičová, J. Filo, V. Garaj, 2020 .

Carbonic anhydrase inhibitors: synthesis and inhibition of cytosolic/tumor-associated carbonic anhydrase isozymes I, II, and IX with sulfonamides incorporating 1,2,4-triazine moieties.

C. Supuran, A. Scozzafava, J. Winum, 2004, Bioorganic & medicinal chemistry letters.

Virtual screening of combinatorial library of novel benzenesulfonamides on mycobacterial carbonic anhydrase II

V. Garaj, F. Dikant, F. Gáplovský, 2016 .

Alkylamino derivatives of N-benzylpyrazine-2-carboxamide: synthesis and antimycobacterial evaluation

L. Naesens, Jana Korduláková, M. Doležal, 2015 .

Synthesis and antimycobacterial evaluation of 5-alkylamino-N-phenylpyrazine-2-carboxamides.

M. Doležal, M. Vejsová, J. Zítko, 2015, Bioorganic & medicinal chemistry.

[Conformational study of drugs which affect I1-imidazoline receptors].

M. Remko, V. Garaj, 2002, Ceska a Slovenska farmacie : casopis Ceske farmaceuticke spolecnosti a Slovenske farmaceuticke spolecnosti.

Theoretical Study of Gas-Phase Acidities of Selected Angiotensin-Converting Enzyme Inhibitors

M. Remko, V. Garaj, Martin Šramko, 2005 .

Gas phase and solution state stability of complexes L…M, where M = Cu2+, Ni2+, or Zn2+ and L = R−C(O)NHOH (R = H, NH2, CH3, CF3, or Phenyl)

M. Remko, V. Garaj, Martin Šramko, 2009 .