A. Chollet

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Probing the Structure and Function of the Tachykinin Neurokinin-2 Receptor through Biosynthetic Incorporation of Fluorescent Amino Acids at Specific Sites*

Manuel Peitsch, Horst Vogel, André Chollet, 1996, The Journal of Biological Chemistry.

Characterization of Non-peptide Antagonist and Peptide Agonist Binding Sites of the NK1 Receptor with Fluorescent Ligands*

G. Turcatti, J. Lowe, T. Schwartz, 1997, The Journal of Biological Chemistry.

Selective Attachment of Oligonucleotides to Interleukin-1β and Targeted Delivery to Cells

A. Chollet, 1990 .

Optimizing the expression in E. coli of a synthetic gene encoding somatomedin-C (IGF-I).

E. Kawashima, G. Buell, N. Movva, 1985, Nucleic acids research.

Preparation, application and biological characterization of interleukin-1 beta mutant protein biotinylated at a single site.

J. Bonnefoy, A. Chollet, N. Odermatt, 1990, Journal of immunological methods.

Effects of the Oral Oxytocin Receptor Antagonist Tocolytic OBE001 on Reproduction in Rats

Jon Rhodes, O. Pohl, P. Baldrick, 2016, Reproductive Sciences.

Oxytocin Receptor Antagonists, Atosiban and Nolasiban, Inhibit Prostaglandin F2α-induced Contractions and Inflammatory Responses in Human Myometrium

Sung Hye Kim, A. Hanyaloglu, P. Bennett, 2019, Scientific Reports.

Identification of the extracellular loop 2 as the point of interaction between the N terminus of the chemokine MIP-1alpha and its CCR1 receptor.

J. Galzi, A. Chollet, S. Zoffmann, 2002, Molecular pharmacology.

Fluorescent pseudo-peptide linear vasopressin antagonists: design, synthesis, and applications.

G. Turcatti, R. Seyer, T. Durroux, 1999, Journal of medicinal chemistry.

JPET #49395 1 PHARMACOLOGY OF (2S,4Z)-N-[(2S)-2-HYDROXY-2-PHENYLETHYL]-4- (METHOXYIMINO)-1-[(2’-METHYL[1,1’-BIPHENYL]-4-YL)CARBONYL]-2- PYRROLIDINECARBOXAMIDE, A NEW POTENT AND SELECTIVE NON- PEPTIDE ANTAGONIST OF THE OXYTOCIN RECEPTOR

C. Giachetti, A. Nichols, C. Barberis, 2003 .

Pharmacology of (2S,4Z)-N-[(2S)-2-Hydroxy-2-phenylethyl]-4-(methoxyimino) -1-[(2′-methyl[1,1′-biphenyl]-4-yl)carbonyl]-2-pyrrolidinecarboxamide, a New Potent and Selective Nonpeptide Antagonist of the Oxytocin Receptor

C. Giachetti, M. Schwarz, A. Scheer, 2003, Journal of Pharmacology and Experimental Therapeutics.

Molecular cloning of mouse tumour necrosis factor cDNA and its eukaryotic expression.

J. Tavernier, L. Fransen, R. Müller, 1985, Nucleic acids research.

Tocolytic effect of a selective FP receptor antagonist in rodent models reveals an innovative approach to the treatment of preterm labor

A. Chollet, R. Cirillo, E. G. Tos, 2007, BMC pregnancy and childbirth.

Arrest of preterm labor in rat and mouse by an oral and selective nonprostanoid antagonist of the prostaglandin F2alpha receptor (FP).

M. Schwarz, A. Scheer, A. Chollet, 2007, American journal of obstetrics and gynecology.

Synthesis and characterization of fluorescent and photoactivatable MIP-1alpha ligands and interactions with chemokine receptors CCR1 and CCR5.

G. Turcatti, J. Galzi, A. Chollet, 2001, Journal of medicinal chemistry.

Pharmacokinetic interactions of OBE001 and betamethasone in healthy female volunteers

A. Patat, O. Pohl, A. Chollet, 2015, Journal of clinical pharmacy and therapeutics.

Synthesis and characterization of selective fluorescent ligands for the neurokinin NK2 receptor.

G. Turcatti, I. Beresford, A. Chollet, 1994, Journal of medicinal chemistry.

Optical surface methods for detection of nucleic acid binding

I. Lundström, C. Mandenius, K. Mosbach, 1989 .

Discovery of a new class of potent, selective, and orally bioavailable CRTH2 (DP2) receptor antagonists for the treatment of allergic inflammatory diseases.

G. Bernardinelli, Y. Filinchuk, C. Giachetti, 2008, Journal of medicinal chemistry.

Expression and characterization of human D4 dopamine receptors in baculovirus‐infected insect cells

E. Kawashima, B. Allet, A. Bernard, 1993, FEBS letters.

Optimization of the Central Core of Indolinone-Acetic Acid-Based CRTH2 (DP2) Receptor Antagonists.

Gordon Campbell, C. Jorand-Lebrun, Z. Johnson, 2011, ACS medicinal chemistry letters.

Palmitoylation but not the extreme amino‐terminus of Gqα is required for coupling to the NK2 receptor

S. Arkinstall, M. Edgerton, A. Chollet, 1994, FEBS letters.

The Effects of Homoconjugated Cyclopropane and Oxirane Rings on the Diels-Alder Reactivity of 2,3-bis (methylidene)norbornane†‡§

P. Vogel, A. Chollet, O. Pilet, 1979 .

Screening for interactions between suitably labelled proteins and an immobilised cyclic peptide library

A. Chollet, E. Magnenat, C. Bradshaw, 1995 .

Iron and ruthenium carbonyls of 6,7-dimethylene-exo-3-oxatricyclo[3.2.1.02.4]octane. Protic acid additions to an epoxide ring homoconjugated to a η4-(diene)Fe(CO)3 function. Crystal structures of (C9H10O)Fe(CO)3 and (C10H14O2)Fe(CO)3

P. Vogel, T. Boschi, D. Schwarzenbach, 1979 .

A Single Mutation of the Neurokinin-2 (NK2) Receptor Prevents Agonist-induced Desensitization

K. Nemeth, A. Chollet, 1995, The Journal of Biological Chemistry.

Fluorescent labeling of NK2 receptor at specific sites in vivo and fluorescence energy transfer analysis of NK2 ligand-receptor complexes.

G. Turcatti, J. Knowles, H. Vogel, 1997, Receptors & channels.

Improved Synthesis of Oligodeoxyribonucleotides by Solid-Phase Phosphotriester Method Utilizing O6-[2-(p-Nitrophenyl)ethyl]-2′-deoxyguanosine Derivatives†

E. Kawashima, E. Ayala, A. Chollet, 1984 .

High-level expression of G protein-coupled receptors with the aid of the Semliki Forest virus expression system.

K. Lundstrom, A. Chollet, G. Agudo, 1995, Journal of receptor and signal transduction research.

Probing the binding domain of the NK2 receptor with fluorescent ligands: evidence that heptapeptide agonists and antagonists bind differently.

G. Turcatti, H. Vogel, A. Chollet, 1995, Biochemistry.

Selective Hydrogen-Chloride Elimination from Primary Chlorides Induced by the Fluoride Anion - Anchimeric Participation of the Chloromethyl Group in the Heterolytic Opening of an Epoxide Stereospecific Syntheses of 5,6-Bis(Methylidene)-Syn-2-Norbornen-7-Ol and 5,6-Bis(Methylidene)-Endo-3-Chloro-Exo-

P. Vogel, A. Chollet, J. Hagenbuch, 1979 .

Carbon-13 n.m.r. spectra of 2,3-dimethylenebicyclo[2.2.1]heptanes and 2,3-dimethylene-7-oxabicyclo[2.2.1]heptanes

P. Vogel, A. Chollet, Daniel Quarroz, 1977 .

Discovery and development of a new class of potent, selective, orally active oxytocin receptor antagonists.

C. Giachetti, M. Schwarz, A. Scheer, 2005, Journal of medicinal chemistry.

Reduction of 5,6‐Dimethylidene‐exo‐2,3‐epoxynorbornane with Metal Hydrides. Efficient syntheses of 6‐methyl‐5‐methylidene‐anti‐3‐ nortricyclanol and of 2,3‐dimethylidene‐anti‐7‐norbornanol

P. Vogel, A. Chollet, 1978 .

Characterisation, CNS distribution and function of NK2 receptors studied using potent NK2 receptor antagonists

E. Kawashima, A. Mcelroy, R. Hagan, 1993, Regulatory Peptides.

DNA containing the base analogue 2-aminoadenine: preparation, use as hybridization probes and cleavage by restriction endonucleases

André Chollet, E. Kawashima, E. Kawashima, 1988, Nucleic Acids Res..

Synthesis of Oligodeoxyribonucleotides Containing the Base 2-Aminoadenine.

E. Kawashima, A. Chollet, A. Chollet-Damerius, 1986 .

Biotin-labeled synthetic oligodeoxyribonucleotides: chemical synthesis and uses as hybridization probes.

E. Kawashima, A. Chollet, 1985, Nucleic acids research.

Differential Effects of Oxytocin Receptor Antagonists, Atosiban and Nolasiban, on Oxytocin Receptor–Mediated Signaling in Human Amnion and Myometrium

Sung Hye Kim, P. Bennett, J. Gotteland, 2017, Molecular Pharmacology.

Biotin-Labeled Synthetic Oligodeoxyribonucleotides: Chemical Synthesis and Uses as Hybridization Probes

E. Kawashima, A. Chollet, 1985 .

Conformational properties of four peptides corresponding to alpha-helical regions of Rhodospirillum cytochrome c2 and bovine calcium binding protein.

S. Wodak, M. Rooman, A. Chaffotte, 1994, Biochemistry.

Subcellular Compartmentalization of Activation and Desensitization of Responses Mediated by NK2 Neurokinin Receptors*

J. Galzi, K. Takeda, A. Chollet, 1999, The Journal of Biological Chemistry.

OBE022, an Oral and Selective Prostaglandin F2α Receptor Antagonist as an Effective and Safe Modality for the Treatment of Preterm Labor

Sung Hye Kim, P. Bennett, P. Guillaume, 2018, The Journal of Pharmacology and Experimental Therapeutics.

Interaction between Non‐Conjugated Chromophores: 5,6‐Dimethylidene‐exo‐2‐norborneol, 5,6‐Dimethylidene‐exo, exo‐2,3‐norbornanediol and 5,6‐Dimethylidene‐2‐norbornanone

P. Vogel, A. Chollet, C. Mahaim, 1977 .

INTERACTION BETWEEN NON-CONJUGATED CHROMOPHORES- 5,6-DIMETHYLIDENE-EXO-2-NORBORNEOL, 5,6-DIMETHYLIDENE-EXO, EXO-2,3-NORBORNANEDIOL AND 5,6-DIMETHYLIDENE-2-NORBORNANONE

P. Vogel, A. Chollet, C. Mahaim, 1977 .

Calcium influx and protein kinase Cα activation mediate arachidonic acid mobilization by the human NK‐2 receptor expressed in Chinese Hamster ovary cells

E. Kawashima, S. Arkinstall, A. Chollet, 1994, FEBS letters.

Sequence determination of the Sendai virus HN gene and its comparison to the influenza virus glycoproteins

C. Giorgi, D. Kolakofsky, R. Raju, 1985, Cell.

Synthesis and characterisation of an immobilised random library of cyclic peptides

T. Wells, A. Chollet, C. Bradshaw, 1993 .

Biophysical approaches to G protein-coupled receptors: Structure, function and dynamics

André Chollet, Gerardo Turcatti, G. Turcatti, 1999, J. Comput. Aided Mol. Des..

Synthesis of fluoresceinyl-neurokinin-A, a biologically active probe for NK2 receptors

A. Chollet, K. Ceszkowski, 1992 .

Stimulation of atrial natriuretic peptide release by neurokinins in neonatal rat ventricular cardiomyocytes.

E. Kawashima, S. Arkinstall, M. Vallotton, 1996, American Journal of Physiology.

Thermodynamic studies of base pairing involving 2,6-diaminopurine.

I. Tinoco, C. Cheong, A. Chollet, 1988, Nucleic acids research.