E. Pitsinos

发表

DNA Binding and Cleavage Modes of Shishijimicin A.

K. Nicolaou, Hao Zhang, Tianhu Li, 2019, Journal of the American Chemical Society.

Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics.

K. Nicolaou, M. Aujay, J. Lyssikatos, 2020, Journal of the American Chemical Society.

Diaryl Ether Formation in the Synthesis of Natural Products

Veroniki P. Vidali, E. Couladouros, E. Pitsinos, 2011 .

Streamlined Total Synthesis of Uncialamycin and Its Application to the Synthesis of Designed Analogues for Biological Investigations.

K. Nicolaou, D. Mandal, G. Vite, 2016, Journal of the American Chemical Society.

Tumor necrosis factor-alpha promotes malignant pleural effusion.

C. Roussos, I. Kalomenidis, T. Blackwell, 2007, Cancer research.

Identification of Gli-mediated transcription inhibitors through synthesis and evaluation of taepeenin D analogues

M. Chatzopoulou, A. Giannis, E. Pitsinos, 2016 .

Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates.

K. Nicolaou, V. Sisodiya, Qifeng Chen, 2020, Journal of the American Chemical Society.

Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating Reagents.

K. Nicolaou, M. Aujay, Christina Lee, 2018, Journal of the American Chemical Society.

Heterofunctional Linking Agents for the Synthesis of Well-Defined Block Copolymers of Dimethylsiloxane and tert-Butyl Methacrylate or 2-Vinylpyridine

N. Hadjichristidis, H. Iatrou, V. Bellas, 2001 .

Synthesis and biological evaluation of novel steroid-modified ether phospholipids.

E. Couladouros, Smaragdi Antonopoulou, H. Karantonis, 2005, Chemistry and physics of lipids.

Total synthesis of calicheamicin .gamma.1I

K. Nicolaou, H. Saimoto, C. W. Hummel, 1992 .

Influence of the Scyphostatin Side Chain on the Mode of Inhibition of Neutral Sphingomyelinase

A. Giannis, E. Pitsinos, V. Wascholowski, 2006, ChemMedChem.

Synthetic calicheamicin mimics with novel initiation mechanisms: DNA cleavage, cytotoxicity, and apoptosis.

K. Nicolaou, H. Saimoto, E. Theodorakis, 1994, Chemistry & biology.

Synthesis and characterization of novel natural product-Gd(III) MRI contrast agent conjugates.

L. Leondiadis, M. Fardis, D. Vourloumis, 2008, Bioorganic & medicinal chemistry letters.

A novel 2'-(N-methylpyridinium acetate) prodrug of paclitaxel induces superior antitumor responses in preclinical cancer models.

G. Gaedicke, K. Nicolaou, R. Guy, 2002, Bioconjugate chemistry.

Open-chain half-bastadins mimic the effects of cyclic bastadins on calcium homeostasis in cultured neurons.

E. Couladouros, E. Pitsinos, J. Lazarewicz, 2008, Bioorganic & medicinal chemistry letters.

A fast entry to furanoditerpenoid-based Hedgehog signaling inhibitors: identifying essential structural features.

M. Chatzopoulou, S. Haroutounian, A. Giannis, 2014, Organic letters.

Total synthesis of calicheamicin .gamma.1I. 3. The final stages

K. Nicolaou, H. Saimoto, K. Baldenius, 1993 .

Enantioselective Synthesis of Cassane-Type Furanoditerpenoids: Total Synthesis of Sucutiniranes C and D

Veroniki P. Vidali, E. Pitsinos, Ioannis Mavridis, 2020 .

Total Synthesis and Full Structural Assignment of Namenamicin.

K. Nicolaou, Ruofan Li, Zhaoyong Lu, 2018, Journal of the American Chemical Society.

Diels–Alder reaction between 1,3,3-trisubstituted-2-vinylcyclohexenes and quinones under exceptionally mild conditions: a concise entry to the cassane-type furanoditerpenoid skeleton

Veroniki P. Vidali, E. Pitsinos, Ioannis Mavridis, 2016 .

Enantioselective total synthesis of (-)-calicheamicinone

K. Nicolaou, E. Pitsinos, A. Smith, 1992 .

Total synthesis of calicheamicin .gamma.1I. 2. Development of an enantioselective route to (-)-calicheamicinone

K. Nicolaou, T. Suzuki, H. Saimoto, 1993 .

Total synthesis of (+)-scyphostatin featuring an enantioselective and highly efficient route to the side-chain via Zr-catalyzed asymmetric carboalumination of alkenes (ZACA).

E. Negishi, Guangwei Wang, Zhao-Qin Xu, 2010, Chemical communications.

Synthesis and Evaluation of Three Novel Scyphostatin Analogues as Neutral Sphingomyelinase Inhibitors

E. Couladouros, A. Giannis, E. Pitsinos, 2003, Chembiochem : a European journal of chemical biology.

A general method for the synthesis of bastaranes and isobastaranes: first total synthesis of bastadins 5, 10, 12, 16, 20, and 21.

E. Couladouros, E. Pitsinos, V. Moutsos, 2004, Chemistry.

Enantioselective Total Synthesis of (‐)‐Calicheamicinone.

K. Nicolaou, E. Pitsinos, A. Smith, 1992 .

Enantioselective total synthesis of (-)-laurenditerpenol.

Veroniki P. Vidali, E. Pitsinos, Nikolaos Athinaios, 2012, Organic letters.

Total Synthesis of Calicheamicin γI 1. Part 2. Development of an Enantioselective Route to (-)-Calicheamicinone.

K. Nicolaou, T. Suzuki, H. Saimoto, 1993 .

Short and efficient route to the fully functionalized polar core of scyphostatin.

E. Pitsinos, A. Cruz, 2005, Organic letters.

Inhibition of topoisomerase I by naphthoquinone derivatives.

A. Assimopoulou, E. Couladouros, V. Papageorgiou, 1998, Bioorganic & medicinal chemistry letters.

Bioefficacy of acyclic monoterpenes and their saturated derivatives against the West Nile vector Culex pipiens.

Veroniki P. Vidali, A. Kimbaris, M. Polissiou, 2014, Chemosphere.

Stereostructural Determination by a Synthetic and NMR‐Based Approach of Three Oxazinins Isolated from Adriatic Mussels

C. Dell’Aversano, P. Ciminiello, L. Tartaglione, 2007 .

Oxazinins from toxic mussels : isolation of a novel oxazinin and reassignment of the C-2 configuration of oxazinin-1 and -2 on the basis of synthetic models

C. Dell’Aversano, P. Ciminiello, M. Forino, 2006 .

Stereoselective Syntheses of 2,6-disubstituted Piperidin-3-oles (alkaloid lipids)

S. Haroutounian, E. Pitsinos, S. Koulocheri, 2008 .

Synthetic studies towards oxazinins. An expedient first total synthesis and proof of the absolute stereochemistry of oxazinin-3

E. Couladouros, E. Pitsinos, V. Moutsos, 2004 .

Uncialamycin-based antibody–drug conjugates: Unique enediyne ADCs exhibiting bystander killing effect

M. Aujay, M. Pysz, H. Karsunky, 2021, Proceedings of the National Academy of Sciences.

Tumor Necrosis Factor-α Promotes Malignant Pleural Effusion

C. Roussos, I. Kalomenidis, T. Blackwell, 2007 .

Synthetic Bastadins Modify the Activity of Ryanodine Receptors in Cultured Cerebellar Granule Cells

E. Couladouros, E. Pitsinos, J. Lazarewicz, 2007, Neurosignals.

A Water‐Soluble Prodrug of Taxol with Self‐Assembling Properties

K. Nicolaou, R. Guy, W. Wrasidlo, 1994 .

Synthesis of enantiopure (S)-7-hydroxy-3-amino-3,4-dihydro-2H-1-benzopyran en route to (+)-scyphostatin

E. Pitsinos, V. Moutsos, Olga Vageli, 2007 .

Total synthesis of (+)-scyphostatin featuring an enantioselective and highly efficient route to the side-chain via Zr-catalyzed asymmetric carboalumination of alkenes (ZACA).

E. Negishi, Guangwei Wang, Zhao-Qin Xu, 2010, Chemical communications.

DNA Binding and Cleavage Modes of Shishijimicin A.

Hao Zhang, Tianhu Li, Ruofan Li, 2019, Journal of the American Chemical Society.

K. Nicolaou, M. Aujay, Christina Lee, 2018, Journal of the American Chemical Society.

Biomimetic Explorations Towards the Bisorbicillinoids: Total Synthesis of Bisorbicillinol, Bisorbibutenolide, and Trichodimerol.

Baran, Veroniki P. Vidali, K. Nicolaou, 1999, Angewandte Chemie.