P. Mainkar

发表

Expanding the tetrahydroquinoline pharmacophore.

R. Ummanni, S. Chandrasekhar, Navya Goli, 2017, Bioorganic & medicinal chemistry letters.

S. Chandrasekhar, S. Ghosh, P. Mainkar, 2021, Tetrahedron Letters.

Strategies towards the synthesis of anti-tuberculosis drugs.

S. Chandrasekhar, R. Grée, P. Mainkar, 2019, Organic & biomolecular chemistry.

In vitro and in vivo studies reveal α-Mangostin, a xanthonoid from Garcinia mangostana, as a promising natural antiviral compound against chikungunya virus

S. Cherian, Manish Kumar Jeengar, P. Mainkar, 2021, Virology journal.

HDAC inhibitor misprocesses bantam oncomiRNA, but stimulates hid induced apoptotic pathway

B. Parida, U. Bhadra, P. Das, 2015, Scientific Reports.

The Ireland-Claisen rearrangement strategy towards the synthesis of the schizophrenia drug, (+)-asenapine.

S. Chandrasekhar, B. Sridhar, P. Mainkar, 2016, Organic & biomolecular chemistry.

Cell-autonomous and non-cell-autonomous mechanisms of transformation by amplified FGFR1 in lung cancer.

Roman K. Thomas, T. Zander, M. Peifer, 2014, Cancer discovery.

Identification of New Molecular Entities (NMEs) as Potential Leads against Tuberculosis from Open Source Compound Repository

R. Ummanni, Tanmay Banerjee, P. Mainkar, 2015, PloS one.

More Twins in the Scientific Literature of the 21st Century

S. Chandrasekhar, P. Mainkar, Ambica Vankamamidi, 2020, Angewandte Chemie International Edition.

Click reaction on in situ generated β-azidostyrenes from cinnamic acid using CAN–NaN3: synthesis of N-styryl triazoles

S. Chandrasekhar, P. Mainkar, M. Kavitha, 2011 .

Synthesis of O-spiro-C-aryl glycosides using organocatalysis.

S. Chandrasekhar, T. Rao, P. Mainkar, 2012, The Journal of organic chemistry.

Intermolecular trifluoromethyl-alkenylation of alkenes enabled by metal-free photoredox catalysis.

P. Mainkar, Srirama Murthy Akondi, Arun D. Kulthe, 2021, Chemical communications.

In Vitro Antiviral Activity of α-Mangostin against Dengue Virus Serotype-2 (DENV-2)

S. Cherian, P. Mainkar, M. Agrawal, 2021, Molecules.

21st Century, More Twins in Scientific Literature: Intentional or Accidental?

S. Chandrasekhar, P. Mainkar, Ambica V, 2020, Angewandte Chemie.

Total synthesis of (±)-galanthamine from GABA through regioselective aryne insertion.

S. Chandrasekhar, P. Mainkar, Telugu Venkatesh, 2019, Organic & biomolecular chemistry.

Synthesis of Asthma Drug Zafirlukast (Accolate) Using Intramolecular Oxidative Coupling via sp3 C–H Bond Activation

S. Chandrasekhar, P. Mainkar, Srinu Paladugu, 2018, ACS omega.

Synthesis and biological evaluation of strained unusual amino acid containing tetrapeptides as potential antidepressant agents.

S. Chakravarty, P. Mainkar, B. N. Babu, 2015, Bioorganic chemistry.

sp3‐Rich Glycyrrhetinic Acid Analogues Using Late‐Stage Functionalization as Potential Breast Tumor Regressing Agents

S. Chandrasekhar, P. Mainkar, Mohana Krishna Reddy Mudiam, 2020, ChemMedChem.

Ruthenium-catalyzed benzimidazoisoquinoline synthesis via oxidative coupling of 2-arylbenzimidazoles with alkynes

S. Chandrasekhar, P. Mainkar, N. Kavitha, 2013 .

Mn-catalyzed radical initiated domino transformation of alkynylated cyclohexadienones with TMSN3 and O2 to bicyclic azido alcohols.

S. Chandrasekhar, P. Mainkar, Pranesh Pal, 2020, Chemical communications.

Diastereoselective synthesis of CF3-dihydrobenzofurans by [4+1] annulation of in situ-generated CF3-o-quinone methides and sulfur ylides

S. Chandrasekhar, P. Mainkar, Nagender Punna, 2020, RSC advances.

Total synthesis of a thromboxane receptor antagonist, terutroban.

S. Chandrasekhar, W. Ahmed, Srihari Pabbaraja, 2015, Organic & biomolecular chemistry.

Synthesis and Self‐Assembly of Bolaamphiphiles Based on β‐Amino Acids or an Alcohol

S. Chandrasekhar, P. Mainkar, A. Sudhakar, 2013 .

Organocatalytic Asymmetric Synthesis of Tetrahydrofuran and 1,2-Dihydrobenzofuran Scaffolds

S. Chandrasekhar, P. Mainkar, L. N. Chavan, 2019, European Journal of Organic Chemistry.

Synthesis of 2-Amino-2'-hydroxy-1,1'-biaryls via Cascade Benzannulation and C-N Bond Cleavage Sequence.

S. Chandrasekhar, P. Mainkar, Raju Adepu, 2020, Organic letters.

Ruthenium(II)-Catalyzed Hydration of Terminal Alkynes in PEG-400

S. Chandrasekhar, P. Mainkar, Rambabu Chegondi, 2016, Synlett.

Synthesis and Biological Evaluation of Naphthopyranopyrimidines Derivatives as Potential Antifungal and Antibacterial Activities

P. Dubey, P. Mainkar, V. Harikrishna, 2016 .

Rapid and one-pot synthesis of tri- to tetradeca-deutero nicotines

S. Chandrasekhar, P. Mainkar, Pashikanti Gouthami, 2020 .

Epoxy-Tethered Diels-Alder Reaction toward the Tricyclic Core of Kalihinols.

S. Chandrasekhar, Shrabani Dinda, P. Mainkar, 2020, Organic letters.

Chemoenzymatic Process for the Preparation of (S)-7-((tert-Butyldiphenylsilyl)oxy)hept-1-yn-4-ol in a Continuous Packed-Bed Reactor, a Key Intermediate for Eribulin Synthesis

S. Chandrasekhar, S. Ghosh, Srihari Pabbaraja, 2020 .

Peptidomimetic organocatalysts: efficient Michael addition of ketones onto nitroolefins with very low catalyst loading

S. Chandrasekhar, B. Jagadeesh, P. Mainkar, 2014 .

High Performance Liquid Chromatography Method for Determination of Trace Amount of Ibutilide Fumarate in Pharmaceutical Manufacturing Environments

Y. Anjaneyulu, P. Mainkar, M. Babu, 2009 .

Caveat in the stereochemical outcome of the organocatalytic Diels–Alder reaction in PEG-400

S. Chandrasekhar, C. S. Reddy, P. Mainkar, 2016 .

Access to Spiroindanolactones/lactams through an Aryne Insertion/Spirocyclization Strategy.

S. Chandrasekhar, P. Mainkar, Palash Ghosh, 2022, Organic letters.

Synthesis of the ‘southern’ tripeptide of Cyclomarins A and C having novel anti-tuberculocidal mode of action

S. Chandrasekhar, P. Mainkar, G. P. Reddy, 2011 .

Convergent synthesis of fully functionalized decalin skeleton of (+)-fusarisetin A

S. Chandrasekhar, P. Mainkar, Karre Nagaraju, 2015 .

Brønsted Acid Catalyzed Domino Aza‐Piancatelli Rearrangement/Michael Reaction: Construction of 1,4‐Benzodiazepin‐5‐ones in One Pot

S. Chandrasekhar, P. Mainkar, Kiranmai Nayani, 2017 .

Stereoselective Synthesis of Northern Fragment of Eribulin Mesylate from d-Mannose

S. Chandrasekhar, P. Mainkar, V. Gaddam, 2018, Synthesis.

A practical synthesis of C14–C26 fragment of anticancer drug, eribulin mesylate

S. Chandrasekhar, P. Mainkar, N. Kiranmai, 2015 .

Total Synthesis of Desmethyl Jahanyne and Its Lipo-Tetrapeptide Conjugates Derived from Parent Skeleton as BCL-2-Mediated Apoptosis-Inducing Agents

S. Chandrasekhar, S. S. Jadav, P. Mainkar, 2018, ACS omega.

Tetrahydrothiopyran-4-one as Five-Carbon Source for Scalable Synthesis of (±)-Tapentadol

S. Chandrasekhar, P. Mainkar, Rambabu Chegondi, 2019, Organic Process Research & Development.

Benzoisothiazolone (BIT): A Fast, Efficient, and Recyclable Redox Reagent for Solid Phase Peptide Synthesis

P. Mainkar, P. Gangireddy, Kiranmai Nayani, 2020 .

Total syntheses of arenamides A, B and C

S. Chandrasekhar, P. Mainkar, G. P. Reddy, 2014 .

Synthesis of α,α-dideutero-β-amino esters

S. Chandrasekhar, P. Mainkar, Srirama Murthy Akondi, 2012 .

Total synthesis of antiviral drug, nirmatrelvir (PF-07321332)

S. Chandrasekhar, Srihari Pabbaraja, P. Mainkar, 2022, Tetrahedron Chem.

Development of Synthetic Approaches Towards HIV Integrase Strand Transfer Inhibitors (INSTIs)

S. S. Jadav, P. Mainkar, Kiranmai Nayani, 2022, ChemistrySelect.

Phenyl 1,2,3-Triazole-Thymidine Ligands Stabilize G-Quadruplex DNA, Inhibit DNA Synthesis and Potentially Reduce Tumor Cell Proliferation over 3′-Azido Deoxythymidine

M. Idris, N. Nagesh, Vuppalapaty Meghah, 2013, PloS one.

"Pruning of biomolecules and natural products (PBNP)": an innovative paradigm in drug discovery.

S. Chandrasekhar, S. R. Bathula, P. Mainkar, 2015, Organic & biomolecular chemistry.

Chiron approach to fully functionalized cyclohexane frame of (+)-Resiniferatoxin

S. Chandrasekhar, P. Mainkar, Y. Rao, 2019, Tetrahedron Letters.

Scalable Synthesis of l-allo-Enduracididine: The Unusual Amino Acid Present in Teixobactin

S. Chandrasekhar, P. Mainkar, Kiranmai Nayani, 2021, Synlett.

A Novel Strategy for 2,6-Dideoxy-L-Hexoses: An Application to 3-Amino-2,3,6-Trideoxy-L-Lyxo-Hexopyranose (L-Daunosamine)

M. K. Gurjar, P. Mainkar, S. M. Pawar, 1989 .

Synthesis of methyl 3-O-(2-O-methyl-α-l-fucopyranosyl)-α-l-rhamnopyranoside, methyl 3-O-α-l-rhamnopyranosyl-α-d-glucopyranoside, and methyl 3-O-[3-O-(2-O-methyl-α-l-fucopyranosyl)-α-l-rhamnopyranosyl]-α-l-rhamnopyranoside: di- and tri-saccharide segments of a lipo-oligosaccharide (LOS-1) of Mycobact

M. K. Gurjar, P. Mainkar, 1993 .

Synthesis and biological evaluation of 5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one structural derivatives as anti-cancer and apoptosis inducing agents.

R. Shukla, S. Chandrasekhar, V. Bansal, 2016, European journal of medicinal chemistry.

A perspective on medicinal chemistry approaches towards adenomatous polyposis coli and Wnt signal based colorectal cancer inhibitors.

R. Gundla, S. S. Jadav, P. Mainkar, 2021, European journal of medicinal chemistry.

A novel isothiocyanate derivative inhibits HIV-1 gene expression and replication by modulating the nuclear matrix associated protein SMAR1.

A. Alam, S. Chattopadhyay, S. Chandrasekhar, 2019, Antiviral research.

Continuous flow process for preparing budesonide

R. Gundla, S. S. Jadav, P. Mainkar, 2022, Journal of Flow Chemistry.

Visible light-promoted Selectfluor-mediated quinone functionalization with unactivated Csp3-H components

P. Mainkar, Maheshwara Reddy Nadiveedhi, Srirama Murthy Akondi, 2021 .

Design principles and functional basis of enantioselectivity of alanyl-tRNA synthetase and a chiral proofreader during protein biosynthesis

R. Sankaranarayanan, P. Mainkar, Shobha P. Kruparani, 2023, Nucleic acids research.

Metal free domino β-azidation/[3+2] cycloaddition reaction for the synthesis of 1,2,3-triazole-fused dihydrobenzoxazinones.

S. Chandrasekhar, P. Mainkar, Kiranmai Nayani, 2019, The Journal of organic chemistry.

Metal-Free Dearomative 2,3-Difunctionalization of Indoles via Radical Cascade

S. Chandrasekhar, B. Sridhar, P. Mainkar, 2023, Tetrahedron Letters.

Functionalization of Tyrosine Containing Short Peptides Via Oxidative Dearomatization Strategy

S. Chandrasekhar, P. Mainkar, Babli K. Jha, 2023, Social Science Research Network.

Diastereoselective Formal Synthesis of Polycyclic Meroterpenoid (±)-Cochlearol A.

S. Chandrasekhar, P. Mainkar, Telugu Venkatesh, 2021, The Journal of organic chemistry.

Synthesis of complete carbon framework of baulamycin A

S. Chandrasekhar, P. Mainkar, Srinu Paladugu, 2017 .

Total Synthesis of Lamellarin D Trimethyl Ether, Lamellarin D, and Lamellarin H.

S. Chandrasekhar, P. Mainkar, Dhanaji M. Lade, 2017, The Journal of organic chemistry.

Research Article Synthetic Studies Towards (-)-(15R)-Hydroxycryptopleurine

S. Chandrasekhar, P. Mainkar, Sanjida Khatun, 2015 .

Formal total synthesis of ( )-rhazinal and its B-ring carbamate analogue

Amitava Das, S. Chandrasekhar, P. Mainkar, 2015 .

Benzyne Insertion onto β-Keto Esters of Polycyclic Natural Products: Synthesis of Benzo Octacyclo Scaffolds.

S. Chandrasekhar, P. Mainkar, Rambabu Chegondi, 2018, Organic Letters.

Construction of Octahydro-4H-cyclopenta[b]pyridin-6-one Skeletons using Pot, Atom, and Step Economy (PASE) Synthesis.

S. Chandrasekhar, B. Sridhar, P. Mainkar, 2023, Chemistry.

Synthesis and biological evaluation of 5,10-dihydro-11H-dibenzo[b,e][1,4]diazepin-11-one structural derivatives as anti-cancer and apoptosis inducing agents.

R. Shukla, S. Chandrasekhar, V. Bansal, 2016, European journal of medicinal chemistry.

Synthesis of cis-fused cyclopentenone-pyrrolidine scaffolds via sequential aza-Piancatelli and Conia-ene type reactions in one pot.

S. Chandrasekhar, P. Mainkar, Kiranmai Nayani, 2024, Chemical Communications.

A formal total synthesis of (6S,7S,9R,10R)-6,9-epoxynonadec-18-ene-7,10-diol from D-glucose

M. K. Gurjar, P. Mainkar, 1990 .

Organocatalytic Asymmetric Synthesis of Tetrahydrofuran and 1,2-Dihydrobenzofuran Scaffolds

S. Chandrasekhar, P. Mainkar, L. N. Chavan, 2019, European Journal of Organic Chemistry.

An Experimental Toolbox for Structure‐Based Hit Discovery for P. aeruginosa FabF, a Promising Target for Antibiotics

R. Brenk, B. Haug, J. Underhaug, 2021, ChemMedChem.