Yun He

发表

Toward the Total Synthesis of Scabrosins: Synthesis of a Desulfur-scabrosin Skeleton and Its Stereoisomers.

Zhi-Peng Wang, Yuyin Liu, Sreenivas Banne, 2019, The Journal of organic chemistry.

Design and synthesis of arylaminoethyl amides as noncovalent inhibitors of cathepsin S. Part 1.

Jennifer L. Harris, R. Epple, B. Bursulaya, 2005, Bioorganic & medicinal chemistry letters.

Pillar[5]arene-based, dual pH and enzyme responsive supramolecular vesicles for targeted antibiotic delivery against intracellular MRSA.

Yun He, Xiaohong Yang, Haibo Peng, 2020, Chemical communications.

Anti‐lung cancer activity and inhibitory mechanisms of a novel Calothrixin A derivative

Jian Guo, Yun He, Xiaohong Yang, 2019, Life sciences.

Synthesis of Carbazolequinones by Formal [3 + 2] Cycloaddition of Arynes and 2-Aminoquinones.

Yuyin Liu, Jian Guo, Yun He, 2016, Organic letters.

Total synthesis of calothrixins and their analogues via formal [3+2] cycloaddition of arynes and 2-aminophenanthridinedione

Jian Guo, Yun He, İ. Kıran, 2016 .

A SERS aptasensor based on porous Au-NC nanoballoons for Staphylococcus aureus detection.

Zhi-Peng Wang, Yun He, Beibei Xie, 2021, Analytica chimica acta.

Synthesis and biological evaluations of sulfanyltriazoles as novel HIV-1 non-nucleoside reverse transcriptase inhibitors.

K. Kuhen, D. Nguyen, B. Bursulaya, 2006, Bioorganic & medicinal chemistry letters.

Transition-Metal-Free Cascade Synthesis of 4-Quinolones: Umpolung of Michael Acceptors via Ene Reaction with Arynes.

Yun He, İ. Kıran, R. Santhosh Reddy, 2016, Organic letters.

Construction of Bridged-Ring-Fused Naphthalenone Derivatives Through an Unexpected Zn(OTf)2-Catalyzed Cascade Transformation.

Sreenivas Banne, Jian Guo, Yun He, 2019, Organic letters.

Thiyl radical promoted chemo- and regioselective oxidation of CC bonds using molecular oxygen via iron catalysis

Zhange Feng, Xiaoqing Zeng, Yun He, 2018 .

Asymmetric Total Syntheses of Aetheramides and Their Stereoisomers: Stereochemical Assignment of Aetheramides.

Srinivasarao Allu, Jian Guo, Yun He, 2016, Organic letters.

A reactive oxygen species (ROS) activated hydrogen sulfide (H2S) donor with self-reporting fluorescence.

Yun He, Zhanlong Wang, Ning Zhang, 2020, ACS sensors.

Hollow and Porous Fe3C-NC Nanoballoons Nanozymes for Cancer Cell H2O2 Detection

Jian Guo, Yun He, Xiaohong Yang, 2021 .

Microbial transformation of diosgenin to diosgenone by Wickerhamomyces anomalus JQ-1 obtained from Naxi traditional Jiu Qu.

Aizhong Liu, Yun He, Lixin Yang, 2019, Bioorganic chemistry.

A mitochondrial targeting two-channel responsive fluorescence probe for imaging the superoxide radical anion in vitro and in vivo.

Yun He, Ning Zhang, Ping Hu, 2019, Talanta.

Crystal structures of human HSP90α-complexed with dihydroxyphenylpyrazoles

J. Caldwell, S. Lesley, A. Kreusch, 2005 .

Label-Free Electrochemical Aptasensor Based on Stone-like Gold Nanoparticles for Ultrasensitive Detection of Tetracycline

Yun He, Chenhui Wang, Haibo Peng, 2021 .

Difuran-substituted quinoxalines as a novel class of PI3Kα H1047R mutant inhibitors: Synthesis, biological evaluation and structure-activity relationship.

Ming-Wei Wang, Jia Wang, Yun He, 2018, European journal of medicinal chemistry.

Inhalable functional mixed-polymer microspheres to enhance doxorubicin release behavior for lung cancer treatment.

Jian Guo, Yun He, Chenhui Wang, 2020, Colloids and surfaces. B, Biointerfaces.

Dual thermo/oxidation-responsive block copolymers with self-assembly behaviour and synergistic release

J. Gu, N. Tirelli, Yun He, 2017 .

Identification of novel potent bicyclic peptide deformylase inhibitors.

A. Kreusch, T. Shin, B. Bursulaya, 2004, Bioorganic & medicinal chemistry letters.

Catalytic asymmetric synthesis of pyrrolidine derivatives bearing heteroatom-substituted quaternary stereocenters

Pan‐Lin Shao, Zhi-Peng Wang, Yun He, 2018 .

Development of an Extended-Release Formulation for Apremilast and a Level A in Vitro-in Vivo Correlation Study in Beagle Dogs.

Hao-Hsin Yu, Yun He, Meiqiong Tang, 2016, Chemical & pharmaceutical bulletin.

Synthesis and biological evaluations of novel benzimidazoles as potential antibacterial agents.

E. Swayze, L. Risen, Yun He, 2004, Bioorganic & medicinal chemistry letters.

2-piperidin-4-yl-benzimidazoles with broad spectrum antibacterial activities.

L. Blyn, E. Swayze, R. Ranken, 2003, Bioorganic & medicinal chemistry letters.

A practical and efficient route to heteraphanes: synthesis of structurally simplified analogues of ansamycins

Yun He, Zheng Shaojun, R. Reddy, 2016 .

Discovery of pyrimidine benzimidazoles as Lck inhibitors: part I.

N. Gray, Jianwei Che, P. Ren, 2008, Bioorganic & medicinal chemistry letters.

Exosome-encapsulated antibiotic against intracellular infections of methicillin-resistant Staphylococcus aureus

Jian Guo, Yun He, Chenhui Wang, 2018, International journal of nanomedicine.

Synthesis of linked carbohydrates and evaluation of their binding for 16S RNA by mass spectrometry.

R. Griffey, E. Swayze, S. Hofstadler, 2003, Bioorganic & medicinal chemistry letters.

Discovery of pyrimidine benzimidazoles as Src-family selective Lck inhibitors. Part II.

N. Gray, Jianwei Che, P. Ren, 2009, Bioorganic & medicinal chemistry letters.

Discovery of 2-amino-6-carboxamidobenzothiazoles as potent Lck inhibitors.

Shenlin Huang, R. Romeo, M. Sandberg, 2008, Bioorganic & medicinal chemistry letters.

Synthesis and biological evaluation of unique stereodimers of sinomenine analogues as potential inhibitors of NO production.

Qiang Xu, Jian-Xin Li, Liping Feng, 2011, Bioorganic & medicinal chemistry.

Controlled coassembly of dumbbell-like Au nanoparticles with a porous nitrogen doped carbon aerogel for cancer cell H2O2 detection.

Yun He, Chenhui Wang, Haibo Peng, 2020, Analytica chimica acta.

Palladium-catalyzed oxidative arylacetoxylation of alkenes: synthesis of indole and indoline derivatives.

Pan‐Lin Shao, Yun He, Ping Hu, 2017, Chemical communications.

Asymmetric Total Synthesis of Nannocystin A.

Yun He, Qiang Liu, Ping Hu, 2017, The Journal of organic chemistry.

Eradicating intracellular MRSA via targeted delivery of lysostaphin and vancomycin with mannose-modified exosomes.

Jian Guo, Yun He, Chenhui Wang, 2020, Journal of controlled release : official journal of the Controlled Release Society.

Synthesis of novel ring-contracted artemisinin dimers with potent anticancer activities.

Yun He, Xiaohong Yang, Ning Zhang, 2018, European journal of medicinal chemistry.

4-Aminopyrimidines as novel HIV-1 inhibitors.

J. Caldwell, K. Kuhen, Yun He, 2007, Bioorganic & Medicinal Chemistry Letters.

Catalytic Asymmetric [3 + 2] Cycloaddition Reaction between Aurones and Isocyanoacetates: Access to Spiropyrrolines via Silver Catalysis.

Pan‐Lin Shao, Zhi-Peng Wang, Yun He, 2018, The Journal of organic chemistry.

Design, synthesis, and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part 2.

J. Caldwell, K. Kuhen, B. Bursulaya, 2006, Bioorganic & medicinal chemistry letters.

Thiyl radical promoted iron-catalyzed-selective oxidation of benzylic sp3 C-H bonds with molecular oxygen.

Zhange Feng, Yun He, Juan Zhang, 2019, Chemical communications.

A Unified Synthetic Approach to Optically Pure Curvularin-Type Metabolites.

Srinivasarao Allu, Sreenivas Banne, Jian Guo, 2019, The Journal of organic chemistry.

Optimization of small molecule agonists of the thrombopoietin (Tpo) receptor derived from a benzo[a]carbazole hit scaffold.

J. Lao, D. Chow, T. Marsilje, 2008, Bioorganic & medicinal chemistry letters.

Synthesis of Dihydrophenanthridines and Oxoimidazolidines from Anilines and Ethylglyoxylate via Aza Diels-Alder Reaction of Arynes and KF-Induced Annulation.

Yun He, İ. Kıran, R. Reddy, 2016, Organic letters.

Discovery and biological evaluation of benzo[a]carbazole-based small molecule agonists of the thrombopoietin (Tpo) receptor.

J. Lao, A. Chatterjee, T. Tuntland, 2008, Bioorganic & medicinal chemistry letters.

An asymmetric Mannich reaction of α-diazocarbonyl compounds and N-sulfonyl cyclic ketimines catalyzed by complexes generated from chiral and achiral phosphines with gold(i).

Yun He, Zhen Wang, Minghui Zhou, 2018, Organic & biomolecular chemistry.

Insertion of Arynes into P-O Bonds: One-Step Simultaneous Construction of C-P and C-O Bonds.

Srinivasarao Allu, Jian Guo, Yun He, 2016, Organic letters.

Development and Mechanistic Studies of Iron-Catalyzed Construction of Csp2-B Bonds via C-O Bond Activation.

Zhange Feng, Xiaoqing Zeng, Yun He, 2020, Organic letters.

C-O Bond Silylation Catalyzed by Iron: A General Method for the Construction of Csp2-Si Bonds.

Zhange Feng, Xiaoqing Zeng, Yun He, 2020, Organic letters.

A Short, Efficient Synthesis of the Novel Cholinergic Channel Activator, ABT 418, from L-Proline

D. Garvey, N. Lin, Yun He, 1995 .

Synthesis and anticancer activity evaluation of novel azacalix[2]arene[2]pyrimidines.

Yun He, Xiaohong Yang, Shao-Lin Zhang, 2018, European journal of medicinal chemistry.

Formal [3 + 2] cycloaddition of α-unsubstituted isocyanoacetates and methyleneindolinones: enantioselective synthesis of spirooxindoles

Pan‐Lin Shao, Zhi-Peng Wang, Yu Zhao, 2017 .

Enantioselective Synthesis of Tetrahydropyridines/Piperidines via Stepwise [4 + 2]/[2 + 2] Cyclizations.

Pan‐Lin Shao, Yixin Lu, Yun He, 2017, Organic letters.

Transition-metal-free synthesis of polysubstituted pyrrole derivatives via cyclization of methyl isocyanoacetate with aurone analogues.

Pan‐Lin Shao, Zhi-Peng Wang, Yun He, 2018, Organic & biomolecular chemistry.

Studies On Isoxazole Formation from Alkyl Carboxylic Esters

N. Lin, Yun He, 1994 .

2‐Piperidin‐4‐yl‐benzimidazoles with Broad Spectrum Antibacterial Activities.

L. Blyn, E. Swayze, R. Ranken, 2003 .

Design, synthesis and biological evaluations of novel oxindoles as HIV-1 non-nucleoside reverse transcriptase inhibitors. Part I.

J. Caldwell, K. Kuhen, B. Bursulaya, 2006, Bioorganic & medicinal chemistry letters.

Design, synthesis, and biological evaluations of novel quinolones as HIV-1 non-nucleoside reverse transcriptase inhibitors.

J. Caldwell, K. Kuhen, B. Bursulaya, 2006, Bioorganic & medicinal chemistry letters.

Boron-Promoted Umpolung Reaction of Sulfonyl Chlorides for the Stereospecific Synthesis of Thioglycosides via Reductive Deoxygenation Coupling Reactions.

Siyu Li, Yun He, Yuanwei Dai, 2022, Organic letters.

A Unified Modular Synthetic Strategy for Dictyodendrins F, H, I, and G.

Sreenivas Banne, Jian Guo, Yun He, 2017, Organic letters.

Synthesis of 1,4,5,6-tetrahydropyridazines and pyridazines via transition-metal-free (4 + 2) cycloaddition of alkoxyallenes with 1,2-diaza-1,3-dienes

Pan‐Lin Shao, Yun He, Qi Wu, 2019, RSC advances.

Selective Aza Diels-Alder and Domino [4+2]/[2+2] Cycloaddition Reactions of Arynes with N-Sulfonyl Ketimines.

Yun He, İ. Kıran, R. Reddy, 2017, The Journal of organic chemistry.

Iron-Catalyzed Borylation of Aryl Ethers via Cleavage of C-O Bonds.

Zhange Feng, Xiaoqing Zeng, Yun He, 2020, Organic letters.

Tandem Diels-Alder/oxidation-aromatization reactions involving 2-styrylchromones and arynes.

Yun He, Zhimei Yu, Cheng Zou, 2018, Organic & biomolecular chemistry.

Catalytic Multisite-Selective Acetoxylation Reactions at sp2 vs sp3 C-H Bonds in Cyclic Olefins.

Cheng-Lin Liu, Pan‐Lin Shao, Yun He, 2016, Organic letters.

Synthesis of Spiro-dihydroquinoline and Octahydrophenanthrene Derivatives via Palladium-Catalyzed Intramolecular Oxidative Arylation.

Pan‐Lin Shao, Yun He, Ping Hu, 2017, Organic letters.

Design, Synthesis and Biological Evaluations of Novel Oxindoles as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors. Part 1.

J. Caldwell, K. Kuhen, B. Bursulaya, 2006 .

Total synthesis and antimicrobial evaluation of natural albomycins against clinical pathogens

Jian Guo, Yun He, Xiaohong Yang, 2018, Nature Communications.

Enantioselective Synthesis of Alkylthioetherpyrrolidine Derivatives via [3+2] Cycloaddition of α-Thioacrylates with Isocyanoacetates.

Pan‐Lin Shao, Zhi-Peng Wang, Yun He, 2017, The Journal of organic chemistry.

Synthesis of Carbazolequinones by Formal [3 + 2] Cycloaddition of Arynes and 2-Aminoquinones.

Yuyin Liu, Jian Guo, Yun He, 2016, Organic letters.

Reexamination of neomycin B degradation: efficient preparation of its CD and D rings as protected glycosyl donors.

E. Swayze, Yun He, Baogen Wu, 2002, Organic letters.

Novel nannocystin A analogues as anticancer therapeutics: Synthesis, biological evaluations and structure-activity relationship studies.

Yun He, Xiaohong Yang, Shao-Lin Zhang, 2019, European journal of medicinal chemistry.

Iron-Catalyzed Borylation and Silylation of Unactivated Tertiary, Secondary, and Primary Alkyl Chlorides

Ming‐Hui Sun, Zhange Feng, Yun He, 2020 .

Synthesis and evaluation of N-aryl pyrrolidinones as novel anti-HIV-1 agents. Part 1.

J. Caldwell, K. Kuhen, H. Yin, 2006, Bioorganic & medicinal chemistry letters.

Targeting cancer metabolism to develop human lactate dehydrogenase (hLDH)5 inhibitors.

K. Tam, Yun He, Shao-Lin Zhang, 2018, Drug discovery today.

Total Synthesis of Kanamienamide.

Yun He, Ning Zhang, Zhimei Yu, 2017, The Journal of organic chemistry.

Synthesis, biological evaluation and structure-activity relationship of a novel class of PI3Kα H1047R mutant inhibitors.

Ming-Wei Wang, Jia Wang, Yun He, 2018, European journal of medicinal chemistry.

Bench-stable imine surrogates for the one-pot and catalytic asymmetric synthesis of α-amino esters/ketones.

Zhi-Peng Wang, Yun He, Adila Nazli, 2020, Chemical communications.

Design and synthesis of TPP+-Mitomycin C conjugate with reduced toxicity.

Yun He, Shao-Lin Zhang, Dong-Mei Luo, 2022, Bioorganic & medicinal chemistry letters.

Iridium-Catalyzed Cycloisomerization of N-Tethered 1,7-Enynes: Construction of Azabicyclo [5.1.0] octene System.

Siyu Li, Jian Guo, Yun He, 2020, The Journal of organic chemistry.

Pd-Catalyzed remote site- and stereo-selective C(alkenyl)-H alkenylation of unactivated cycloalkenes.

Cheng‐He Zhou, Yun He, Gui-Xin Cai, 2019, The Journal of organic chemistry.

Design and synthesis of 7H-pyrrolo[2,3-d]pyrimidines as focal adhesion kinase inhibitors. Part 2.

J. Caldwell, N. Gray, T. Honda, 2006, Bioorganic & medicinal chemistry letters.

Polymeric micelles with dual thermal and reactive oxygen species (ROS)-responsiveness for inflammatory cancer cell delivery

N. Tirelli, Yun He, Xiaohong Yang, 2017, Journal of Nanobiotechnology.

Synthesis and structure-activity relationships of 2′-(R) and (S) pyrrolidine-modified analogs of the cholinergic channel activator, ABT-418

S. Arneric, J. Sullivan, N. Lin, 1995 .

Design and synthesis of 7H-pyrrolo[2,3-d]pyrimidines as focal adhesion kinase inhibitors. Part 1.

J. Caldwell, N. Gray, O. Ohmori, 2006, Bioorganic & medicinal chemistry letters.

Construction of Polycyclic Indole Derivatives via Multiple Aryne Reactions with Azaheptafulvenes.

Yun He, Zhen Wang, Yesu Addepalli, 2018, Organic letters.

Synthesis and properties of gem-dinitro energetic salts based on 1,2,4-oxadiazole with low impact sensitivity

Jia Song, T. Lu, Yun He, 2021 .

Total Syntheses of Anti-HIV Cyclodepsipeptides Aetheramides A and B.

Srinivasarao Allu, Jian Guo, Yun He, 2016, The Journal of organic chemistry.

pH-dependent, stereoselective dimerization of sinomenine.

Jian-Xin Li, Yu Zhao, Yun He, 2008, Organic letters.

A short, efficient chiral synthesis of a novel cholinergic channel activator, ABT-418 [(S)-3-methyl-5-(1-methyl-2-pyrrolidinyl)isoxazole], from (S)-pyroglutamic acid

N. Lin, Yun He, H. Kopecká, 1995 .

Development of dual inhibitors targeting pyruvate dehydrogenase kinases and human lactate dehydrogenase A: High-throughput virtual screening, synthesis and biological validation.

K. Tam, Yun He, Shao-Lin Zhang, 2020, European journal of medicinal chemistry.

Crystal structures of human HSP90alpha-complexed with dihydroxyphenylpyrazoles.

Scott A Lesley, Andreas Kreusch, Yun He, 2005, Bioorganic & medicinal chemistry letters.

Synthesis of Vitamin B12-Antibiotic Conjugates with Greatly Improved Activity against Gram-Negative Bacteria.

Siyu Li, Zhi-Peng Wang, Jian Guo, 2020, Organic letters.

Near-Infrared Laser-Triggered, Self-Immolative Smart Polymersomes for in vivo Cancer Therapy

Yun He, Haibo Peng, Ning Zhang, 2020, International journal of nanomedicine.

Total synthesis and antimicrobial evaluation of natural albomycins against clinical pathogens

Jian Guo, Yun He, Xiaohong Yang, 2018, Nature Communications.

Stevens rearrangement of thioethers with arynes: a facile access to multi-substituted β-keto thioethers.

Yuyin Liu, Jian Guo, Yun He, 2017, Organic & biomolecular chemistry.

Synthesis and evaluation of novel bacterial rRNA-binding benzimidazoles by mass spectrometry.

R. Griffey, P. Kung, V. Mohan, 2004, Bioorganic & medicinal chemistry letters.

Synthesis and structure–activity relationships of 5-substituted pyridine analogues of 3-[2-((S)-pyrrolidinyl)methoxy]pyridine, A-84543: A potent nicotinic receptor ligand

S. Arneric, T. Kuntzweiler, N. Lin, 2001 .

Synthesis and biological evaluation of unique stereodimers of sinomenine analogues as potential inhibitors of NO production.

Qiang Xu, Jian-Xin Li, Liping Feng, 2011, Bioorganic & medicinal chemistry.

[3 + 2] Cycloaddition of Azaoxyallyl Cations with Cyclic Ketones: Access to Spiro-4-oxazolidinones.

Pan‐Lin Shao, Zhi-Peng Wang, Yun He, 2017, The Journal of organic chemistry.

Design, synthesis and biological evaluation of artemisinin derivatives containing fluorine atoms as anticancer agents.

Yun He, Xiaohong Yang, Qian Meng, 2018, Bioorganic & medicinal chemistry letters.

Discovery of 2-amino-6-carboxamidobenzothiazoles as potent Lck inhibitors.

Shenlin Huang, R. Romeo, T. Spalding, 2008, Bioorganic & medicinal chemistry letters.