Y. Hsiao

发表

Preparation of the HIV Attachment Inhibitor BMS-663068. Part 7. Development of a Regioselective Ullmann–Goldberg–Buchwald Reaction

Martin D. Eastgate, D. Blackmond, R. J. Fox, 2017 .

Catalytic Production of Dimethylformamide from Supercritical Carbon Dioxide

P. Jessop, T. Ikariya, R. Noyori, 1994 .

Synthesis of Sitagliptin

Feng Xu, Edward J. J. Grabowski, Shane W. Krska, 2009 .

Highly efficient asymmetric synthesis of sitagliptin.

Feng Xu, Andrew Clausen, Shane W. Krska, 2009, Journal of the American Chemical Society.

Highly efficient synthesis of beta-amino acid derivatives via asymmetric hydrogenation of unprotected enamines.

Shane W. Krska, E. Njolito, F. Wang, 2004, Journal of the American Chemical Society.

Identification of Ammonium Chloride as an Effective Promoter of the Asymmetric Hydrogenation of a β-Enamine Amide

C. Starbuck, Mahmoud S. Kaba, Y. Hsiao, 2006 .

Methyl formate synthesis by hydrogenation of supercritical carbon dioxide in the presence of methanol

P. Jessop, T. Ikariya, R. Noyori, 1995 .

C-H Arylation in the Formation of a Complex Pyrrolopyridine, the Commercial Synthesis of the Potent JAK2 Inhibitor, BMS-911543.

Martin D. Eastgate, Paul C. Lobben, R. J. Fox, 2018, The Journal of organic chemistry.

Effects of Multiple Catalyst Deactivation Pathways and Continuous Ligand Recycling on the Kinetics of Pd-Catalyzed C-N Coupling Reactions.

Martin D. Eastgate, Maxime C Soumeillant, Y. Hsiao, 2018, The Journal of organic chemistry.

Stereoselective synthesis of an anti-HIV drug candidate.

M. Palucki, D. Conlon, D. Hughes, 2005, Chirality.

Mechanistic Studies of a Pd-Catalyzed Direct Arylation En Route to Beclabuvir: Dual Role of a Tetramethylammonium Cation and an Unusual Turnover-Limiting Step

Antonio Ramirez, C. Hang, E. Simmons, 2021 .

Highly diastereoselective heterogeneously catalyzed hydrogenation of enamines for the synthesis of chiral beta-amino acid derivatives.

E. Njolito, D. Tellers, J. Armstrong, 2004, Journal of the American Chemical Society.

Synthesis of Optically Active Imidazolines, Azapenams, Dioxocyclams, and Bis-dioxocyclams

L. Hegedus, Y. Hsiao, 1997 .

The First Kilogram Synthesis of Beclabuvir, an HCV NS5B Polymerase Inhibitor

Richard L. Schild, C. Hang, Zhinong Gao, 2018, Organic Process Research & Development.

Ligand-Enabled β-C-H Arylation of α-Amino Acids Without Installing Exogenous Directing Groups.

jin-quan yu, Y. Hsiao, Zhe Zhuang, 2017, Angewandte Chemie.

An efficient synthesis of an alphavbeta3 antagonist.

L. Tan, M. Palucki, R. Volante, 2004, The Journal of organic chemistry.

Synthesis of an anti-methicillin-resistant Staphylococcus aureus (MRSA) carbapenem via stannatrane-mediated Stille coupling.

P. Reider, D. Hughes, Y. Hsiao, 2000, Organic letters.

Synthesis Optimization, Scale-Up, and Catalyst Screening Efforts toward the MGAT2 Clinical Candidate, BMS-963272

Lidet K. Negash, A. Mathur, R. Lawrence, 2022, Organic Process Research & Development.

Adventures in Atropisomerism: Total Synthesis of a Complex Active Pharmaceutical Ingredient with Two Chirality Axes.

Jason M. Stevens, Thomas M. Razler, Antonio Ramirez, 2018, Organic letters.

Nickel complexes incorporating an amido phosphine chelate with a pendant amine arm: synthesis, structure, and catalytic Kumada coupling.

Lan‐Chang Liang, Y. Hsiao, Wei-Ying Lee, 2012, Dalton transactions.

Synthesis of Fmoc-Protected Arylphenylalanines (Bip Derivatives) via Nonaqueous Suzuki-Miyaura Cross-Coupling Reactions.

M. Poss, Jennifer X. Qiao, Y. Hsiao, 2016, The Journal of organic chemistry.

First Generation Process for the Preparation of the DPP-IV Inhibitor Sitagliptin

Edward J. J. Grabowski, Spencer D. Dreher, J. Armstrong, 2005 .

Preparation of the HIV Attachment Inhibitor BMS-663068. Part 2. Strategic Selections in the Transition from an Enabling Route to a Commercial Synthesis

Bin Zheng, Ke Chen, Martin D. Eastgate, 2017 .

Methods for the Synthesis of 5,6,7,8-Tetrahydro-1,8-naphthyridine Fragments for αVβ3 Integrin Antagonists

L. Tan, D. Zewge, M. Palucki, 2004 .

Asymmetric synthesis of isoquinoline alkaloids by homogeneous catalysis

R. Noyori, M. Kitamura, Y. Hsiao, 1986 .

Synthetic approaches to a chiral 4-amino-3-hydroxy piperidine with pharmaceutical relevance.

M. Sugiyama, D. Conlon, I. S. Young, 2012, Organic & biomolecular chemistry.

General asymmetric synthesis of isoquinoline alkaloids. Enantioselective hydrogenation of enamides catalyzed by BINAP-Ruthenium(II) complexes

R. Noyori, M. Kitamura, Y. Hsiao, 1994 .

Stereoselective synhtesis of a precursor of 1β-methylcarbapenems

R. Noyori, M. Kitamura, Y. Hsiao, 1990 .

Stereoselective Synthesis of a Precursor of 1β-Methylcarbapenems.

R. Noyori, M. Kitamura, Y. Hsiao, 1990 .

Zirconium complexes containing a diarylamido diphosphine ligand: Structural preferences controlled by ligand electronics and sterics

Lan‐Chang Liang, Y. Hsiao, Chunbang Li, 2011 .

Ligand-Enabled β-C(sp3)-H Olefination of Free Carboxylic Acids.

M. Poss, jin-quan yu, Jennifer X. Qiao, 2018, Journal of the American Chemical Society.

Ligand-Enabled β-C-H Arylation of α-Amino Acids Without Installing Exogenous Directing Groups.

jin-quan yu, Y. Hsiao, Zhe Zhuang, 2017, Angewandte Chemie.

Proline-catalyzed, asymmetric mannich reactions in the synthesis of a DPP-IV inhibitor.

J. Armstrong, J. Janey, Y. Hsiao, 2006, The Journal of organic chemistry.

Highly regioselective Friedländer reaction.

P. Reider, D. Hughes, Y. Hsiao, 2001, Organic letters.

The impact of palladium(II) reduction pathways on the structure and activity of palladium(0) catalysts.

Qi Gao, Jacob Albrecht, Srinivas Tummala, 2013, Angewandte Chemie.

Nickel-Catalyzed Synthesis of Quinazolinediones.

Thomas M. Razler, E. Simmons, G. Beutner, 2017, Organic letters.

Development of a Kilogram-Scale Process for the Enantioselective Synthesis of 3-Isopropenyl-cyclohexan-1-one via Rh/DTBM-SEGPHOS-Catalyzed Asymmetric Hayashi Addition Enabled by 1,3-Diol Additives

Thomas M. Razler, Y. Qiu, E. Simmons, 2017 .

Development of a new and practical route to chiral 3,4-disubstituted cyclopentanones: asymmetric alkylation and intramolecular cyclopropanation as key C-C bond-forming steps.

M. Palucki, P. Reider, D. Conlon, 2002, The Journal of organic chemistry.

General asymmetric synthesis of benzomorphans and morphinans via enantioselective hydrogenation

R. Noyori, M. Kitamura, Y. Hsiao, 1987 .

Preparation of crystalline p-nitrobenzyl 2-formyl carbapenems by oxidative cleavage.

D. Hughes, Y. Hsiao, N. Yasuda, 1999, Bioorganic & medicinal chemistry letters.

A practical one-pot process for α-amino aryl ketone synthesis

Ross A. Miller, K. Conrad, Y. Hsiao, 2005 .

Mono-Oxidation of Bidentate Bis-phosphines in Catalyst Activation: Kinetic and Mechanistic Studies of a Pd/Xantphos-Catalyzed C-H Functionalization.

Michael Schmidt, Martin D. Eastgate, Yining Ji, 2015, Journal of the American Chemical Society.

Development of a scalable palladium-catalyzed α-arylation process for the synthesis of a CGRP antagonist

David K. Leahy, M. Hay, Y. Hsiao, 2013 .

A preparatively convenient ligand-free catalytic PEG 2000 Suzuki-Miyaura coupling.

Thomas M. Razler, Ruiling Fu, R. Khan, 2009, The Journal of organic chemistry.

Gas chromatographic analysis of the thermally unstable dimethyl methylphosphonate carbanion via trimethylsilyl derivatization.

Y. Hsiao, N. Yasuda, V. Antonucci, 2002, Journal of chromatography. A.

HOMOGENEOUS CATALYSIS IN SUPERCRITICAL FLUIDS : HYDROGENATION OF SUPERCRITICAL CARBON DIOXIDE TO FORMIC ACID, ALKYL FORMATES, AND FORMAMIDES

P. Jessop, R. Noyori, Y. Hsiao, 1996 .

Efficient and scalable enantioselective synthesis of a CGRP antagonist.

David K. Leahy, R. Hanson, M. Sugiyama, 2012, Organic letters.

The impact of palladium(II) reduction pathways on the structure and activity of palladium(0) catalysts.

Martin D. Eastgate, S. Tummala, O. Soltani, 2013, Angewandte Chemie.

Ligand-Enabled β-C(sp3)-H Olefination of Free Carboxylic Acids.

M. Poss, jin-quan yu, Jennifer X. Qiao, 2018, Journal of the American Chemical Society.