C. Hoarau

发表

A new synthetic approach to biaryls of the rhazinilam type. Application to synthesis of three novel phenylpyridine-carbamate analogues.

Anne-Laure Bonneau, N. Robert, C. Hoarau, 2007, Organic & biomolecular chemistry.

Mechanism selection for regiocontrol in base-assisted, palladium-catalysed direct C-H coupling with halides: first approach for oxazole- and thiazole-4-carboxylates.

L. van Hijfte, C. Hoarau, F. Marsais, 2011, Chemistry.

Direct palladium-catalyzed alkenylation, benzylation and alkylation of ethyl oxazole-4-carboxylate with alkenyl-, benzyl- and alkyl halides.

C. Hoarau, F. Marsais, Cécile Verrier, 2009, Organic & biomolecular chemistry.

A New Approach to Isoindolobenzazepines. A Simple Synthesis of Lennoxamine

A. Couture, E. Deniau, P. Grandclaudon, 2000 .

Ligand controlled orthogonal base-assisted direct C–H bond arylation in oxa(thia)zole-4-carboxylate series. New insights in nCMD mechanism

C. Hoarau, O. Querolle, G. Dupas, 2013 .

Direct Stereoselective β-Arylation of Enol Ethers by a Decarboxylative Heck-Type Reaction

C. Hoarau, C. Schneider, Mahmoud Hachem, 2020 .

Copper-catalyzed direct C-H fluoroalkenylation of heteroarenes.

X. Pannecoucke, C. Hoarau, C. Schneider, 2016, Organic & biomolecular chemistry.

Pd- and Cu-catalyzed stereo- and regiocontrolled decarboxylative/C-H fluoroalkenylation of heteroarenes.

X. Pannecoucke, C. Hoarau, C. Schneider, 2014, Chemistry.

Palladium- and copper-catalyzed stereocontrolled direct C-H fluoroalkenylation of heteroarenes using gem-bromofluoroalkenes.

X. Pannecoucke, C. Hoarau, C. Schneider, 2013, Angewandte Chemie.

Palladium-Catalyzed Domino Allenamide Carbopalladation/Direct C-H Allylation of Heteroarenes: Synthesis of Primprinine and Papaverine Analogues.

C. Hoarau, I. Gillaizeau, C. Schneider, 2018, Organic letters.

On study of sterically controlled regioselective lithiation of meta-halopyridocarboxamides derivatives

N. Robert, C. Hoarau, F. Marsais, 2009 .

Deprotonation of pyridine carboxamides using lithium magnesiates bases

C. Hoarau, F. Marsais, G. Quéguiner, 2008 .

Efficient and fast Heck vinylation of 2-bromo-6-methyl pyridines with methylacrylate. Application to the synthesis of 6-methyl cyclopenta[b]pyridinone

Sylvain Celanire, N. Robert, C. Hoarau, 2005 .

Regioselective Pd-Catalyzed Carbopalladation / Decarboxylative Allylic Alkynylation of ortho-Iodoallenamides with alkynyl carboxylic acids.

C. Hoarau, I. Gillaizeau, C. Schneider, 2019, The Journal of organic chemistry.

Synthesis of the heterocyclic core of the D-series GE2270

C. Hoarau, F. Marsais, C. Berini, 2017, Beilstein journal of organic chemistry.

Carbonates: eco-friendly solvents for palladium-catalysed direct arylation of heteroaromatics

C. Hoarau, H. Doucet, J. Dong, 2010 .

Carbonates: ecofriendly solvents for palladium-catalyzed direct 2-arylation of oxazole derivatives.

Ronan Le Goff, C. Hoarau, H. Doucet, 2009, ChemSusChem.

Chemoenzymatic synthesis of highly enantiomerically enriched secondary alcohols with a thiazolic core

M. Toșa, F. Irimie, L. Bencze, 2012 .

Unusual sterically controlled regioselective lithiation of 3-bromo-5-(4,4'-dimethyl)oxazolinylpyridine. Straightforward access to highly substituted nicotinic acid derivatives.

Anne-Laure Bonneau, N. Robert, C. Hoarau, 2006, Organic letters.

Diastereoselective dearomatization of resorcinols directed by a lactic acid tether: unprecedented enantioselective access to p-quinols.

T. Pettus, C. Hoarau, Lupe H. Mejorado, 2004, Organic Letters.

Neat total synthesis of six monoterpenic alkaloids of the actinidine series

N. Robert, C. Hoarau, F. Marsais, 2007 .

Recent advances in direct C–H arylation: Methodology, selectivity and mechanism in oxazole series

C. Hoarau, F. Marsais, G. Quéguiner, 2011, Beilstein journal of organic chemistry.

Deprotonation of benzoxazole and oxazole using lithium magnesates.

F. Mongin, C. Hoarau, F. Marsais, 2005, The Journal of organic chemistry.

Metal-Catalyzed Direct C-H Fluoroalkenylation of Pyridine N-Oxides and Related Derivatives

X. Pannecoucke, C. Hoarau, C. Schneider, 2017 .

Pd-catalyzed decarboxylative cross-coupling of 2-carboxyazine N-oxides with various (hetero)aryl halides.

Corinne Fruit, C. Hoarau, C. Schneider, 2014, Chemistry.

Direct C-2 arylation of alkyl 4-thiazolecarboxylates: new insights in synthesis of heterocyclic core of thiopeptide antibiotics.

C. Hoarau, F. Marsais, Cécile Verrier, 2008, Organic letters.

Ortho-directed functionalization of arenes using magnesate bases.

C. Hoarau, F. Marsais, G. Quéguiner, 2010, Chemical communications.

iso-PsE, a new pseudopterosin

R. Little, Guang Wu, R. Jacobs, 2008 .

Regioselective decarboxylative cross-coupling of carboxy isoquinoline N-oxides.

Corinne Fruit, C. Hoarau, C. Schneider, 2015, The Journal of organic chemistry.

Palladium-catalyzed direct (hetero)arylation of ethyl oxazole-4-carboxylate: an efficient access to (hetero)aryloxazoles.

C. Hoarau, F. Marsais, Cécile Verrier, 2008, The Journal of organic chemistry.

Oxidative dearomatization of resorcinol derivatives: useful conditions leading to valuable cyclohexa-2,5-dienones

T. Pettus, C. Hoarau, R. Water, 2003 .

Regioselective palladium-catalyzed phenylation of ethyl 4-oxazolecarboxylate

A. Couture, P. Grandclaudon, C. Hoarau, 2005 .

A Convenient Synthesis of Alkyl- and Dialkylphenanthren-9-ylamines

A. Couture, E. Deniau, P. Grandclaudon, 2004 .

A New Synthetic Approach to Dioxoaporphines − Application to the Synthesis of N-Methylouregidione

A. Couture, E. Deniau, P. Grandclaudon, 2001 .

Ortho-Directed Palladium-Catalyzed Direct C–H Functionalization of 3-Picolinyl- and 3-(2-Cyanoethyl)pyrimidin-4(3H)-ones with Aryl Halides

C. Hoarau, V. Levacher, L. Bischoff, 2020, Synlett.

Ligand-free Pd-catalyzed and copper-assisted C-H arylation of quinazolin-4-ones with aryl iodides under microwave heating.

Corinne Fruit, Sylvain Laclef, T. Besson, 2015, Organic letters.

A concise total synthesis of the azaphenanthrene alkaloid eupolauramine.

A. Couture, H. Cornet, E. Deniau, 2001, The Journal of organic chemistry.

Diastereoselective addition of metalated isoindolin-1-ones to aldehydes. Stereoselective preparation of (E)-3-arylideneisoindolin-1-ones

A. Couture, E. Deniau, P. Grandclaudon, 2002 .

TOTAL SYNTHESES OF TALISCANINE, VELUTINAM, AND ENTEROCARPAM II

A. Couture, E. Deniau, P. Grandclaudon, 1998 .

A Versatile Synthesis of Poly- and Diversely Substituted Isoindolin-1-ones

A. Couture, E. Deniau, P. Grandclaudon, 2000 .

Orthopalladation of GFP-Like Fluorophores Through C-H Bond Activation: Scope and Photophysical Properties

C. Cativiela, A. Jiménez, E. Urriolabeitia, 2018, European Journal of Organic Chemistry.

Organometallic Fluorophores of d8 Metals (Pd, Pt, Au)

E. Urriolabeitia, C. Hoarau, L. Bischoff, 2018 .

Palladium catalyzed one-pot sequential Suzuki cross-coupling-direct C-H functionalization of imidazo[1,2-a]pyrazines.

P. Jubault, J. Bonfanti, C. Hoarau, 2012, Organic letters.

Stereoselective synthesis of the lituarine tricyclic spiroacetal.

J. Robertson, C. Hoarau, Paul Meo, 2004, Organic letters.

DMAP-Catalyzed Regel-Type Direct C-2 (Hetero)Aroylation of Oxazoles and Thiazoles Derivatives with Acid Chlorides

C. Hoarau, F. Marsais, P. Lassalas, 2013 .

Orthogonal Palladium‐Catalyzed Direct C−H Bond Arylation of Heteroaromatics with Aryl Halides

Corinne Fruit, C. Hoarau, C. Schneider, 2016 .

Synthesis and orthogonal functionalization of oxazolo[5',4':4,5]pyrano[2,3-b]pyridine by intra- and intermolecular Pd-catalyzed direct C-H bond heteroarylation.

L. Meerpoel, C. Hoarau, O. Querolle, 2016, Organic & biomolecular chemistry.

Metalation of 4-oxazolinyloxazole derivatives. A convenient route to 2,4-bifunctionalized oxazoles.

R. Houssin, J. Hénichart, A. Couture, 2002, The Journal of organic chemistry.

Strategies for the Preparation of Differentially Protected ortho-Prenylated Phenols.

T. Pettus, C. Hoarau, 2003, Synlett : accounts and rapid communications in synthetic organic chemistry.

Miyaura borylation/Suzuki-Miyaura coupling (MBSC) sequence of 4-bromo-2,4'-bithiazoles with halides: straightforward access to a heterocylic cluster of d-series of thiopeptide GE2270.

C. Hoarau, F. Marsais, C. Berini, 2018, Organic & biomolecular chemistry.

Pd-Catalyzed Regioselective Decarboxylative/C–H α-Alkoxyalkenylation of Heterocycles Using α-Carboxyvinylethers

C. Hoarau, C. Schneider, Jean-Baptiste E. Y. Rouchet, 2017 .

Direct Synthesis of Benzo[c]carbazoles by Pd-Catalyzed C-H [4 + 2] Annulation of 3-Arylindoles with External 1,3-Dienes.

C. Hoarau, S. Pal, Y. Ramondenc, 2022, Organic letters.

A mild anionic method for generating o-quinone methides: facile preparations of ortho-functionalized phenols.

T. Pettus, C. Hoarau, T. Ung, 2001, The Journal of organic chemistry.

A New Synthetic Approach to Dioxoaporphines — Application to the Synthesis of N‐Methylouregidione (Xb).

A. Couture, E. Deniau, P. Grandclaudon, 2002 .

Deprotonation of thiophenes using lithium magnesates

F. Mongin, C. Hoarau, F. Marsais, 2005 .

Dearomatization applications of I(III) reagents and some unusual reactivity amongst resorcinol derived cyclohexadienones.

T. Pettus, C. Hoarau, Todd A. Wenderski, 2010, Tetrahedron.

General synthesis for chiral 4-alkyl-4-hydroxycyclohexenones.

T. Pettus, C. Hoarau, 2006, Organic letters.

An Expeditious Synthesis of Goniothalactam

A. Couture, E. Deniau, P. Grandclaudon, 1999 .

Pd(0)-Catalyzed Direct Inter- and Intramolecular C–H Functionalization of 4-Carboxyimidazoles

L. Meerpoel, P. Angibaud, C. Hoarau, 2020, Synlett.

Chemoselective Palladium‐Catalyzed Direct C–H Arylation of 5‐Carboxyimidazoles: Unparalleled Access to Fused Imidazole‐Based Tricycles Containing Six‐, Seven‐ or Eight‐Membered Rings

L. Meerpoel, P. Angibaud, C. Hoarau, 2017 .

Lead optimization of purine based orally bioavailable Mps1 (TTK) inhibitors.

P. Slattum, M. Bursavich, Bruce L. Roth, 2012, Bioorganic & medicinal chemistry letters.

Concerted vs Nonconcerted Metalation-Deprotonation in Orthogonal Direct C-H Arylation of Heterocycles with Halides: A Computational Study.

V. Gandon, C. Hoarau, 2021, Journal of Organic Chemistry.

Highly efficient borylation Suzuki coupling process for 4-bromo-2-ketothiazoles: straightforward access to micrococcinate and saramycetate esters.

C. Hoarau, F. Marsais, Thibaut Martin, 2009, Organic letters.

Cyclocondensation of amidines with dimethyl acetylenedicarboxylate: A convenient entry into tetramic acids

W. Cao, I. Erden, C. Hoarau, 2006 .

Amine Directed Palladium Catalyzed C-H Halogenation of Phenylalanine Derivatives.

Sébastien Coufourier, G. Journot, C. Hoarau, 2021, Chemistry.

Cyclocondensation of Amidines with Dimethyl Acetylenedicarboxylate: A Convenient Entry into Tetramic Acids.

W. Cao, I. Erden, C. Hoarau, 2006 .

Highly Efficient Borylation Suzuki Coupling Process for 4‐Bromo‐2‐ketothiazoles: Straightforward Access to Micrococcinate and Saramycetate Esters.

C. Hoarau, F. Marsais, Thibaut Martin, 2010 .

Insights in the Synthesis of Imidazolones from Aldehydes, Isocyanides, or Oxazolines.

C. Hoarau, L. Bischoff, Christine Baudequin, 2022, The Journal of organic chemistry.

DPO and POPOP carboxylate-analog sensors by sequential palladium-catalysed direct arylation of oxazole-4-carboxylates.

C. Hoarau, F. Marsais, Cécile Verrier, 2011, Organic & biomolecular chemistry.

Total Syntheses of Taliscanine, Velutinam, and Enterocarpam II.

A. Couture, E. Deniau, P. Grandclaudon, 2010 .

Pd-Catalyzed direct C-H functionalization of imidazolones with aryl- and alkenyl halides.

C. Hoarau, L. Bischoff, Christine Baudequin, 2015, Chemical Communications.

Formation of Imidazolones by Ring Closure of α-Isocyanoamides: Exploring New Reactivities

C. Hoarau, L. Bischoff, Christine Baudequin, 2020, Synlett.

Pd(0)-Catalyzed Direct C-H Functionalization of 2-H-4-Benzylidene Imidazolones: Friendly and Large-Scale Access to GFP and Kaede Protein Fluorophores.

C. Hoarau, C. Perrio, L. Bischoff, 2016, Chemistry.

Pd-Catalyzed Direct C—H Functionalization of Imidazolones with Aryl- and Alkenyl Halides.

C. Hoarau, L. Bischoff, Christine Baudequin, 2015 .

Mild, Efficient, One-Pot Synthesis of Imidazolones Promoted by N,O-Bistrimethylsilylacetamide (BSA)

L. Colombeau, C. Hoarau, L. Bischoff, 2016, Synlett.