Huan He

发表

Diversified Synthesis of 2-(4-Oxo[1,2,3]triazolo[1,5-a]quinoxalin-5(4H)-yl)acetamide Derivatives through Ugi-4-CR and Copper-Catalyzed Tandem Reactions

Xiaoyun Lu, Yong Zhang, Q. Cai, 2017, Synthesis.

Stereoselective synthesis of α-d-fructofuranosides using a 4,6-O-siloxane-protected donor

Xiao‐Yu Liu, Rui Wang, Yong Qin, 2021 .

Copper-catalyzed coupling of (S)-1-(3-bromophenyl)-ethylamine and N–H containing heteroarenes using microwave heating

Yong-Jin Wu, Huan He, A. L’Heureux, 2003 .

Lanthanide Germanate Cluster Organic Frameworks Based on {Ln8Ge12} Clusters: From One-Dimensional Chains to Two-Dimensional Layers and Three-Dimensional Frameworks.

Junwei Zhao, G. Cao, Huan He, 2016, Inorganic chemistry.

Na₂B₁₀O₁₇·H₂en: a three-dimensional open-framework layered borate co-templated by inorganic cations and organic amines.

Jun-hua Wang, Huan He, Bai-Feng Yang, 2015, Chemical communications.

NaB3O5·0.5H2O and NH4NaB6O10: Two Cluster Open Frameworks with Chiral Quartz and Achiral Primitive Cubic Nets Constructed from Oxo Boron Cluster Building Units

Jun-hua Wang, Huan He, Bai-Feng Yang, 2014 .

Optimization and biological evaluation of nicotinamide derivatives as Aurora kinase inhibitors.

Xingwei Xu, Huan He, Ying Yang, 2019, Bioorganic & medicinal chemistry.

The first 2-D organic–inorganic hybrid containing two types of hexa-CuII sandwiched polyoxotungstate units and mixed amines

Junwei Zhao, Huan He, Bai-Feng Yang, 2014 .

Temperature-Dependent Organic Functionalization of {Ni6PW9} Species: from Isolated Clusters to 1D Chain

Junwei Zhao, B. Cai, Huan He, 2014, Journal of Cluster Science.

Syntheses, structures and properties of two multi-iron–samarium/multi-iron substituted germanotungstates

Junwei Zhao, Huan He, Bai-Feng Yang, 2014 .

Discovery of thiazolidin-4-one urea analogues as novel multikinase inhibitors that potently inhibit FLT3 and VEGFR2.

Yuting Zhou, Tao Chen, Xingwei Xu, 2019, Bioorganic & medicinal chemistry.

Novel organic–inorganic hybrid one-dimensional chain assembled by oxalate-bridging terbium-substituted phosphotungstate dimers and dinuclear copper(II)–oxalate clusters

Junwei Zhao, Huan He, Bai-Feng Yang, 2013 .

Asymmetric synthesis of chiral P-stereogenic triaryl phosphine oxides via Pd-catalyzed kinetic arylation of diaryl phosphine oxides

Yong Zhang, Qiu-Ying Wang, Q. Cai, 2016 .

Synthesis of diaryl ethers through the copper-catalyzed arylation of phenols with aryl halides using microwave heating

Yong-Jin Wu, Huan He, 2003 .

Palladium-catalyzed amination of 3-bromo-4-fluoro-acetophenone

Yong-Jin Wu, Huan He, Jie Chen, 2002 .

A Desulfurative Strategy for the Generation of Alkyl Radicals Enabled by Visible-Light Photoredox Catalysis.

Xiao‐Yu Liu, Yong Qin, F. Xue, 2018, Angewandte Chemie.

Chiral Aryliodine-Catalyzed Asymmetric Oxidative C-N Bond Formation via Desymmetrization Strategy.

Q. Ding, Q. Cai, Huan He, 2018, Organic letters.

A 3D aluminoborate open framework interpenetrated by 2D zinc-amine coordination-polymer networks in its 11-ring channels.

Zhien Lin, Huan He, Bai-Feng Yang, 2014, Angewandte Chemie.

Two organic-inorganic hybrid 3D {P(5)W(30)}-based heteropolyoxotungstates with transition-metal/Ln-carboxylate-Ln connectors.

Junwei Zhao, Huan He, Bai-Feng Yang, 2014, Chemistry, an Asian journal.

A series of organic–inorganic hybrids based on lanthanide-substituted Dawson-type phosphotungstate dimers and copper–en linkers

Junwei Zhao, Huan He, Bai-Feng Yang, 2014 .

Total Synthesis of Liangshanone.

Xiao‐Yu Liu, Feng-peng Wang, Yong Qin, 2020, Angewandte Chemie.

Two novel 2D organic–inorganic hybrid silicotungstates assembled by {Cu2Ln2(ox)(SiW11)2} dimers and [Cu(en)(ox)]/[Cu(en)2] linkers

Zhihui Zhang, Zhong Zhang, Huan He, 2016 .

Novel Three-Dimensional Organic–Inorganic Heterometallic Hybrid Built by Sandwich-Type Tetra-Mn-Substituted Germanotungstates through Mixed 3d and 4f Metal Linkers

Junwei Zhao, Huan He, Bai-Feng Yang, 2013 .

(S,E)-N-[1-(3-heteroarylphenyl)ethyl]-3-(2-fluorophenyl)acrylamides: synthesis and KCNQ2 potassium channel opener activity.

S. Dworetzky, Ronald J. Knox, Joanne Natale, 2005, Bioorganic & medicinal chemistry letters.

Enantioselective Synthesis of Chiral Oxygen-Containing Heterocycles Using Copper-Catalyzed Aryl C-O Coupling Reactions via Asymmetric Desymmetrization.

Xinhao Zhang, Yong Zhang, Qiu-Ying Wang, 2017, The Journal of organic chemistry.

Discovery of a cyclopentylamine as an orally active dual NK1 receptor antagonist-serotonin reuptake transporter inhibitor.

J. Macor, R. Westphal, R. Bertekap, 2014, Bioorganic & medicinal chemistry letters.

Discovery of disubstituted piperidines and homopiperidines as potent dual NK1 receptor antagonists-serotonin reuptake transporter inhibitors for the treatment of depression.

J. Macor, R. Westphal, R. Bertekap, 2013, Bioorganic & medicinal chemistry.

Aluminum Effects in the Syndiospecific Copolymerization of Styrene with Ethylene by Cationic Fluorenyl Scandium Alkyl Catalysts

Xiaoying Wang, Z. Hou, Y. Liu, 2013 .

Bis(imino)diphenylamido rare-earth metal dialkyl complexes: synthesis, structure, and catalytic activity in living ring-opening ε-caprolactone polymerization and copolymerization with γ-butyrolactone.

Gaixia Du, Zhengguo Lin, Yuping Dong, 2013, Dalton transactions.

Copper-catalyzed cross-coupling of aryl iodides and aryl acetylenes using microwave heating

Yong-Jin Wu, Huan He, 2004 .

Identification of a potent and selective 5-HT(6) antagonist: one-step synthesis of (E)-3-(benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin-4-ylidenamine from 2-(benzenesulfonyl)-3,3-bis(methylsulfanyl)acrylonitrile.

R. Westphal, P. Scola, R. Bertekap, 2003, Journal of medicinal chemistry.

Copper-catalyzed N-arylation of sulfonamides with aryl bromides and iodides using microwave heating

Yong-Jin Wu, Huan He, 2003 .

Regiospecific alkyl addition of (hetero)arene-fused thiophenes enabled by a visible-light-mediated photocatalytic desulfuration approach.

Xiao‐Yu Liu, Yong Qin, F. Xue, 2018, Chemical communications.

Identification of novel N1-(2-aryl-1, 3-thiazolidin-4-one)-N3-aryl ureas showing potent multi-tyrosine kinase inhibitory activities.

Yuting Zhou, Min Liu, Anmian Zhang, 2018, European journal of medicinal chemistry.

Copper‐Catalyzed Cross‐Coupling of Aryl Halides and Thiols Using Microwave Heating.

Yong-Jin Wu, Huan He, 2004 .

Synthesis and Characterization of a 3-D Framework Constructed from [V12B18O54(OH)6(H2O)]10− Clusters and K+ Cations

Junwei Zhao, Huan He, Bai-Feng Yang, 2014, Journal of Cluster Science.

A Series of Aluminoborates Templated or Supported by Zinc-Amine Complexes.

Qiang Zhang, Huan He, Bai-Feng Yang, 2015, Chemistry.

Copper-Catalyzed Cross-Coupling of Aryl Halides and Thiols Using Microwave Heating

Yong-Jin Wu, Huan He, 2003 .

Two New Borates Made of [B5O6(OH)4]− and [B5O10(OH)]6− Clusters, Accompanying a Novel In Situ Organic Reaction

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2015, Journal of Cluster Science.

Two New Borates Containing [B5O6(OH)4] Clusters, Accompanying a Novel In Situ Organic Reaction Between Ethylenediamine and CH3COO− Group

Qiang Zhang, Huan He, Bai-Feng Yang, 2015, Journal of Cluster Science.

Two new organic borates with the large [B14O20(OH)6]4− oxoboron clusters

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2014, Journal of Cluster Science.

Syntheses and Crystal Structures of Two New Pentaborates Templated by Transition-Metal Complexes

Huan He, Bai-Feng Yang, Guoming Wang, 2014, Journal of Cluster Science.

Two Borate Supramolecular Frameworks Based on B4O5(OH)4 Cluster Units

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2015, Journal of Cluster Science.

Fluorine substitution can block CYP3A4 metabolism-dependent inhibition: identification of (S)-N-[1-(4-fluoro-3- morpholin-4-ylphenyl)ethyl]-3- (4-fluorophenyl)acrylamide as an orally bioavailable KCNQ2 opener devoid of CYP3A4 metabolism-dependent inhibition.

S. Dworetzky, Ronald J. Knox, C. Polson, 2003, Journal of medicinal chemistry.

Separation and purification of five alkaloids from Aconitum duclouxii by counter-current chromatography.

Weili Huang, Yang Chen, Canhui Xiang, 2015, Journal of separation science.

Three new mixed-alkali- and alkaline-earth-metal borates: from 1D chain to 2D layer to 3D framework.

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2013, Inorganic chemistry.

Two Hexa-Ni-Substituted AsW9O34 Clusters Functionalized by Organic Ligands

Junwei Zhao, B. Cai, Huan He, 2014, Journal of Cluster Science.

Series of open-framework aluminoborates containing [B5O10] clusters.

Huan He, Bai-Feng Yang, Guoming Wang, 2015, Dalton transactions.

Synthesis, structure and properties of a new noncentrosymmetric aluminoborate

Huan He, Bai-Feng Yang, Guoming Wang, 2014 .

Novel organic–inorganic hybrid monomeric Keggin-type phosphotungstate containing heterometallic {Ni6WNi} clusters

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2015 .

Solvothermal Synthesis and Structure of Two New Borates Containing [B7O9(OH)5]2− and [B12O18(OH)6]6− Clusters

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2016, Journal of Cluster Science.

A novel lead borate of NaPb4(H2O)(B5O9)2·BO3 with nonlinear optical property

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2015 .

[Pb(en)0.5][B5O8(OH)]: A New Bilayered Organic–Inorganic Hybrid Lead Borate Built by B5O8(OH) Cluster Units

Qiang Zhang, Huan He, Bai-Feng Yang, 2015, Journal of Cluster Science.

A new mixed metal borate of BaPb[B5O9(OH)]·H2O with acentric structure

Huan He, Guo‐Yu Yang, Han‐Qing Wu, 2013 .

Synthesis, Structure and Properties of a New Noncentrosymmetric Aluminoborate.

Huan He, Bai-Feng Yang, Guoming Wang, 2014 .

Asymmetric Synthesis of (-)-Pterocarine and (-)-Galeon via Chiral Phase Transfer-Catalyzed Atropselective Formation of Diarylether Cyclophane Skeleton.

Q. Ding, Qiu-Ying Wang, Q. Cai, 2017, Organic letters.

Two New Mixed Metal Borates Made of Mg(B6O7(OH)6)2 and B8O14(OH)4 Cluster Units

Huan He, Bai-Feng Yang, Guo‐Yu Yang, 2015, Journal of Cluster Science.

Synthesis of fluorinated 1-(3-morpholin-4-yl-phenyl)-ethylamines.

Yong-Jin Wu, Qi Gao, Huan He, 2003, Bioorganic & medicinal chemistry letters.

Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT₆ antagonists.

D. Langley, R. Westphal, P. Sivaprakasam, 2014, Bioorganic & medicinal chemistry.

Identification of novel quinoline analogues bearing thiazolidinones as potent kinase inhibitors for the treatment of colorectal cancer.

Yuting Zhou, Xingwei Xu, Guowei Gong, 2020, European journal of medicinal chemistry.

Discovery of N1-(4-((7-(3-(4-ethylpiperazin-1-yl)propoxy)-6-methoxyquinolin-4-yl)oxy)-3,5-difluorophenyl)-N3-(2-(2,6-difluorophenyl)-4-oxothiazolidin-3-yl)urea as a multi-tyrosine kinase inhibitor for drug-sensitive and drug-resistant cancers treatment.

Jun Yu Li, Tao Chen, Xingwei Xu, 2019, European journal of medicinal chemistry.

(S)-N-[1-(3-morpholin-4-ylphenyl)ethyl]- 3-phenylacrylamide: an orally bioavailable KCNQ2 opener with significant activity in a cortical spreading depression model of migraine.

V. Gribkoff, S. Dworetzky, Ronald J. Knox, 2003, Journal of medicinal chemistry.

A new acentric metal borate Mg[B6O9(OH)2]·4H2O: Synthesis, structure and optical property

Qiang Zhang, Huan He, Bai-Feng Yang, 2014 .

Discovery of (S,E)-3-(2-fluorophenyl)-N-(1-(3-(pyridin-3-yloxy)phenyl)ethyl)-acrylamide as a potent and efficacious KCNQ2 (Kv7.2) opener for the treatment of neuropathic pain.

V. Gribkoff, Ping Chen, S. Dworetzky, 2013, Bioorganic & medicinal chemistry letters.

Synthesis and KCNQ2 opener activity of N-(1-benzo[1,3]dioxol-5-yl-ethyl, N-[1-(2,3-dihydro-benzofuran-5-yl)-ethyl, and N-[1-(2,3-dihydro-1H-indol-5-yl)-ethyl acrylamides.

Qi Gao, Jie Chen, Huan He, 2004, Bioorganic & medicinal chemistry letters.

(S)-N-[1-(4-cyclopropylmethyl-3,4-dihydro-2H-benzo[1,4]oxazin-6-yl)-ethyl]-3-(2-fluoro-phenyl)-acrylamide is a potent and efficacious KCNQ2 opener which inhibits induced hyperexcitability of rat hippocampal neurons.

Qi Gao, Jie Chen, Huan He, 2004, Bioorganic & medicinal chemistry letters.

Hydrothermal Syntheses and Structural Characterization of Two 3-D Supramolecular Networks Constructed from Tetra-CoII Sandwiched Polyoxometalates

Junwei Zhao, Huan He, Bai-Feng Yang, 2014, Journal of Cluster Science.

Synthesis, Structural Characterization and Properties of Two Strontium Borates Constructed from Oxo Boron Clusters

Jing Xue, Huan He, Bai-Feng Yang, 2014, Journal of Cluster Science.

LiBa1.5[B5O8(OH)3]: A new 1-D metal borate chain constructed from B5O9(OH)36 − cluster units

Huan He, Guo‐Yu Yang, Han‐Qing Wu, 2014 .

Amino Acid Functionalization of {Ni6PW9}-Based Clusters Under Hydrothermal Conditions

Junwei Zhao, B. Cai, Huan He, 2014, Journal of Cluster Science.

Concise syntheses of eburnane indole alkaloids.

Xiao‐Yu Liu, Yong Qin, Huan He, 2018, Chemical communications.

Synthesis and Structure−Activity Relationship of Acrylamides as KCNQ2 Potassium Channel Openers

V. Gribkoff, S. Dworetzky, Joanne Natale, 2004 .

Discovery of 4-((4-(4-(3-(2-(2,6-difluorophenyl)-4-oxothiazolidin-3-yl)ureido)-2-fluorophenoxy)-6-methoxyquinolin-7-yl)oxy)-N,N-diethylpiperidine-1-carboxamide as kinase inhibitor for the treatment of colorectal cancer.

Yuting Zhou, Xingwei Xu, Huan He, 2020, Bioorganic chemistry.

An improved glycal diazidation protocol with copper catalysis

Xiao‐Yu Liu, Yong Qin, Huan He, 2021 .

A Desulfurative Strategy for the Generation of Alkyl Radicals Enabled by Visible-Light Photoredox Catalysis.

Xiao‐Yu Liu, Yong Qin, F. Xue, 2018, Angewandte Chemie.

A 3D aluminoborate open framework interpenetrated by 2D zinc-amine coordination-polymer networks in its 11-ring channels.

Zhien Lin, Huan He, Bai-Feng Yang, 2014, Angewandte Chemie.

Na₂B₁₀O₁₇·H₂en: a three-dimensional open-framework layered borate co-templated by inorganic cations and organic amines.

Jun-hua Wang, Huan He, Bai-Feng Yang, 2015, Chemical communications.