G. Caltabiano

发表

The role of Cysteine 6.47 in class A GPCRs

Gianluigi Caltabiano, Arnau Cordomí, Mireia Olivella, 2013, BMC Structural Biology.

Structure-based rationalization of antitumor drugs mechanism of action by a MIF approach.

D. Condorelli, G. Cruciani, G. Musumarra, 2004, European journal of medicinal chemistry.

Analysis of Human Dopamine D3 Receptor Quaternary Structure*

G. Milligan, Sara Marsango, C. Pou, 2015, The Journal of Biological Chemistry.

The Parkinson's disease‐associated GPR37 receptor‐mediated cytotoxicity is controlled by its intracellular cysteine‐rich domain

L. Pardo, F. Ciruela, I. Stagljar, 2013, Journal of neurochemistry.

Design, synthesis, and biological evaluation of 4-alkyliden-beta lactams: new products with promising antibiotic activity against resistant bacteria.

G. Musumarra, C. Fortuna, R. Musumeci, 2006, Journal of medicinal chemistry.

The role of residue stability in transient protein–protein interactions involved in enzymatic phosphate hydrolysis. A computational study

Michael A. Johnston, J. Teyra, J. Bonet, 2005, Proteins: Structure, Function, and Bioinformatics.

Modulation of the Interaction between a Peptide Ligand and a G Protein-Coupled Receptor by Halogen Atoms.

J. C. Gómez-Tamayo, L. Pardo, A. Ardá, 2015, ACS medicinal chemistry letters.

New potent antibacterials against Gram-positive multiresistant pathogens: effects of side chain modification and chirality in linezolid-like 1,2,4-oxadiazoles.

L. Goracci, G. Musumarra, C. Fortuna, 2014, Bioorganic & medicinal chemistry.

New linezolid-like 1,2,4-oxadiazoles active against Gram-positive multiresistant pathogens.

L. Goracci, G. Musumarra, C. Fortuna, 2013, European journal of medicinal chemistry.

Structural Determinants for the Interaction of Formyl Peptide Receptor 2 with Peptide Ligands*

L. Pardo, R. Ye, G. Caltabiano, 2013, The Journal of Biological Chemistry.

Identification of the first germline mutation in the extracellular domain of the follitropin receptor responsible for spontaneous ovarian hyperstimulation syndrome

L. Pardo, S. Costagliola, G. Vassart, 2008, Human mutation.

Tracking G-protein-coupled receptor activation using genetically encoded infrared probes

T. Sakmar, X. Deupí, G. Schertler, 2010, Nature.

Design, synthesis and in vitro antitumor activity of new trans 2-[2-(heteroaryl)vinyl]-1,3-dimethylimidazolium iodides.

G. Musumarra, C. Fortuna, Paolo Benedetti, 2004, Bioorganic & medicinal chemistry.

GPCRtm: An amino acid substitution matrix for the transmembrane region of class A G Protein-Coupled Receptors

Gianluigi Caltabiano, Leonardo Pardo, Angel Gonzalez, 2015, BMC Bioinformatics.

Membrane Protein Simulations Using AMBER Force Field and Berger Lipid Parameters.

Gianluigi Caltabiano, Arnau Cordomí, Leonardo Pardo, 2012, Journal of chemical theory and computation.

A Molecular Basis for Selective Antagonist Destabilization of Dopamine D3 Receptor Quaternary Organization

M. Millan, R. Ward, J. Pediani, 2017, Scientific Reports.

The Antiallergic Mast Cell Stabilizers Lodoxamide and Bufrolin as the First High and Equipotent Agonists of Human and Rat GPR35

B. Hudson, G. Milligan, S. Nicklin, 2014, Molecular Pharmacology.

Microsoft Word-23820973-file00

B. Hudson, G. Milligan, Jennifer, 2013 .

The cloned equine thyrotropin receptor is hypersensitive to human chorionic gonadotropin; identification of three residues in the extracellular domain involved in ligand specificity.

L. Pardo, F. Savagner, Y. Malthiéry, 2008, Endocrinology.

The extracellular entrance provides selectivity to serotonin 5-HT7 receptor antagonists with antidepressant-like behavior in vivo.

Gianluigi Caltabiano, Leonardo Pardo, Bellinda Benhamú, 2014, Journal of medicinal chemistry.

Halogenated triazinediones behave as antagonists of PKR1: in vitro and in vivo pharmacological characterization

S. Salvadori, G. Balboni, A. Francioso, 2014 .

Impact of Helix Irregularities on Sequence Alignment and Homology Modeling of G Protein‐Coupled Receptors

Gianluigi Caltabiano, Arnau Cordomí, Leonardo Pardo, 2012, Chembiochem : a European journal of chemical biology.

A Molecular Basis for Selective Antagonist Destabilization of Dopamine D3 Receptor Quaternary Organization

M. Millan, G. Milligan, R. Ward, 2017, Scientific Reports.

Identification of transmembrane domains that regulate spatial arrangements and activity of prokineticin receptor 2 dimers

A. Hanyaloglu, S. Sposini, R. Miele, 2015, Molecular and Cellular Endocrinology.

GPCRtm: An amino acid substitution matrix for the transmembrane region of class A G Protein-Coupled Receptors

L. Pardo, M. Fernandez, M. Campillo, 2015, BMC Bioinformatics.

The role of hydrophobic amino acids in the structure and function of the rhodopsin family of G protein-coupled receptors.

L. Pardo, M. Campillo, Ángel González, 2013, Methods in enzymology.

Structural determinants for the interaction of formyl peptide receptor 2 with peptide ligands.

L. Pardo, R. Ye, G. Caltabiano, 2014, The Journal of Biological Chemistry.

The coexistence of a novel inactivating mutant thyrotropin receptor allele with two thyroid peroxidase mutations: a genotype-phenotype correlation.

L. Pardo, S. Refetoff, Chutintorn Sriphrapradang, 2011, The Journal of clinical endocrinology and metabolism.

The extracellular entrance provides selectivity to serotonin 5-HT7 receptor antagonists with antidepressant-like behavior in vivo.

J. C. Gómez-Tamayo, L. Pardo, M. López-Rodríguez, 2014, Journal of medicinal chemistry.

Defining the organizational structure of dopamine and muscarninic acetylcholine receptors

G. Milligan, Sara Marsango, G. Caltabiano, 2015, SpringerPlus.

The Molecular Basis of Oligomeric Organization of the Human M3 Muscarinic Acetylcholine Receptor

G. Milligan, R. Ward, Sara Marsango, 2015, Molecular Pharmacology.

Microsoft Word-73148042-file00.docx

G. Milligan, R. Ward, G. Caltabiano, 2015 .

The specificity of binding of glycoprotein hormones to their receptors

L. Pardo, S. Costagliola, A. D. Leener, 2008, Cellular and Molecular Life Sciences.