C Ceccarelli

Nonpeptidic inhibitors of human leukocyte elastase. 5. Design, synthesis, and X-ray crystallography of a series of orally active 5-aminopyrimidin-6-one-containing trifluoromethyl ketones.

P. Bernstein, J. R. Damewood, P R Bernstein, 1995, Journal of medicinal chemistry.

Nonpeptidic inhibitors of human leukocyte elastase. 3. Design, synthesis, X-ray crystallographic analysis, and structure-activity relationships for a series of orally active 3-amino-6-phenylpyridin-2-one trifluoromethyl ketones.

P. Bernstein, J. R. Damewood, P. Edwards, 1994, Journal of medicinal chemistry.