W. Tueckmantel

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Synthesis and biology of a 7-nitro-2,1,3-benzoxadiazol-4-yl derivative of 2-phenylindole-3-acetamide: a fluorescent probe for the peripheral-type benzodiazepine receptor.

A. Kozikowski, N. Boujrad, M. Kotoula, 1997, Journal of medicinal chemistry.

Identification of novel α4β2-nicotinic acetylcholine receptor (nAChR) agonists based on an isoxazole ether scaffold that demonstrate antidepressant-like activity.

D. Brunner, R. Lukas, A. Kozikowski, 2012, Journal of medicinal chemistry.

Studies in polyphenol chemistry and bioactivity. 4.(1) Synthesis of trimeric, tetrameric, pentameric, and higher oligomeric epicatechin-derived procyanidins having all-4beta,8-interflavan connectivity and their inhibition of cancer cell growth through cell cycle arrest.

A. Kozikowski, W. Tueckmantel, L. Romanczyk, 2003, The Journal of organic chemistry.

Studies in Polyphenol Chemistry and Bioactivity. 1. Preparation of Building Blocks from (+)-Catechin. Procyanidin Formation. Synthesis of the Cancer Cell Growth Inhibitor, 3- O -Galloyl-(2 R ,3 R )-epicatechin-4β,8-[3- O -galloyl-(2 R ,3 R )-epicatechin]

A. Kozikowski, W. Tueckmantel, L. Romanczyk, 1999 .

Synthesis of 1D-3-deoxy- and -2,3-dideoxyphosphatidylinositol

G. Powis, L. Qiao, A. Kozikowski, 1997 .

Huperzine A--a potent acetylcholinesterase inhibitor of use in the treatment of Alzheimer's disease.

A. Kozikowski, S. Geib, W. Tueckmantel, 1991, Acta crystallographica. Section C, Crystal structure communications.

Inositol Analogs as Potential Anticancer Therapeutics

G. Powis, A. Kozikowski, M. Malaska, 1994, Current Medicinal Chemistry.

3,8‐Methanoaza[10]annulene (Homoisoquinoline)

D. Cremer, E. Kraka, E. Vogel, 1985 .

Copper(I) Oxide

W. Tueckmantel, R. Dembinski, Nicholas Bewick, 2009 .

Transition-metal catalyzed silylzincation and silylalumination of acetylenic compounds

K. Oshima, W. Tueckmantel, H. Nozaki, 1986 .

Synthesis of D-3-deoxy-3-phosphonomethyl-myo-inositol and its dimethyl ester - compounds of use in studying the ptdins-3′-kinase signalling pathway

G. Powis, A. Gallegos, A. Kozikowski, 1993 .

Chemistry and behavioral studies identify chiral cyclopropanes as selective α4β2-nicotinic acetylcholine receptor partial agonists exhibiting an antidepressant profile.

D. Brunner, R. Lukas, A. Kozikowski, 2012, Journal of medicinal chemistry.

1,4‐Addition of triorganozincates and silyldiorganozincates to α,β‐unsaturated ketones

K. Oshima, W. Tueckmantel, H. Nozaki, 1986 .

The synthesis of 2,3,3a,4,5,7a-hexahydro-1H-inden-1-ols by intramolecular Diels-Alder reactions of 1,3,8-nonatrien-5-ols. Dependence of product stereochemistry on the substitution pattern

A. Kozikowski, W. Tueckmantel, 1991 .

Studies in polyphenol chemistry and bioactivity. 2. Establishment of interflavan linkage regio- and stereochemistry by oxidative degradation of an O-alkylated derivative of procyanidin B2 to (R)-(-)-2,4-diphenylbutyric acid.

C. George, A. Kozikowski, C. George, 2000, The Journal of organic chemistry.

Synthesis and reactions of oligomethylene‐clamped 1 H‐azepines and benzene imines. Their valence tautomeric equilibrium and nitrogen stereochemistry

W. Tueckmantel, W. Lange, W. Tückmantel, 1989 .

Synthesis, molecular modeling, and biology of the 1-benzyl derivative of APDC-AN apparent mGluR6 selective ligand

J. Wroblewski, Shaomeng Wang, A. Kozikowski, 1997 .

Methods for Synthesizing the Cocoa‐Derived Oligomeric Epi‐Catechins – Observations on the Anticancer Activity of the Cocoa Polyphenols

A. Kozikowski, W. Tueckmantel, 2009 .

An Approach to Open Chain and Modified Heterocyclic Analogues of the Acetylcholine-sterase Inhibitor, Huperzine A, through a Bicyclo[3.3.1]nonane Intermediate

G. Campiani, A. Kozikowski, W. Tueckmantel, 1994 .

Synthesis of the thiazolone analogue of the acetylcholinesterase inhibitor, huperzine A

B. P. Doctor, A. Kozikowski, W. Tueckmantel, 1994 .

Synthesis and biology of the rigidified glutamate analogue, trans-2-carboxyazetidine-3-acetic acid (t-CAA)

J. Wroblewski, Shaomeng Wang, A. Kozikowski, 1996 .

Synthesis, nicotinic acetylcholine receptor binding affinities, and molecular modeling of constrained epibatidine analogues.

C. George, A. Kozikowski, K. Kellar, 2003, Journal of medicinal chemistry.

Synthesis and biology of the conformationally restricted ACPD analogue, 2-aminobicyclo[2.1.1]hexane-2,5-dicarboxylic acid-I, a potent mGluR agonist.

J. Wroblewski, A. Kozikowski, S. Wang, 1998, Journal of medicinal chemistry.

1-amino-APDC, a partial agonist of group II metabotropic glutamate receptors with neuroprotective properties.

J. Wroblewski, A. Kozikowski, S. Pshenichkin, 1999, Bioorganic & medicinal chemistry letters.

Synthesis of Pyrano[4,3‐b]Azepines by [4 + 2] Cycloaddition of Photochemically Generated 3‐Alkoxycarbonyl‐1,2‐Didehydroazepines with Enol Ethers

W. Tueckmantel, 1994 .

Studies in polyphenol chemistry and bioactivity. 3.(1,2) stereocontrolled synthesis of epicatechin-4alpha,8-epicatechin, an unnatural isomer of the B-type procyanidins.

A. Kozikowski, Y. Hu, W. Tueckmantel, 2001, The Journal of organic chemistry.

Synthesis of a biotin conjugate of the PCP analogue “metaphit” for potential use in NMDA/PCP receptor isolation

A. Kozikowski, K. Krueger, W. Tueckmantel, 1989 .