U. Piarulli

发表

Diacetoneglucose Complexes of Manganese(II) and Iron(II) and Their Organometallic Derivatization

C. Floriani, N. Re, D. Viterbo, 1998 .

Supramolecular ligand-ligand and ligand-substrate interactions for highly selective transition metal catalysis.

S. Carboni, L. Pignataro, C. Gennari, 2011, Dalton transactions.

Optimization of New Chiral Ligands for the Copper-Catalysed Enantioselective Conjugate Addition of Et2Zn to Nitroolefins by High-Throughput Screening of a Parallel Library

R. F. Jackson, C. Gennari, U. Piarulli, 2001 .

Investigation of a New Family of Chiral Ligands for Enantioselective Catalysis via Parallel Synthesis and High-Throughput Screening

S. Ceccarelli, R. F. Jackson, C. Montalbetti, 1998 .

Oxo- and imido-molybdenum(VI) and -tungsten(VI) functionalities supported by diacetoneglucose

C. Floriani, D. Viterbo, G. Gervasio, 1995 .

Transition metal carbohydrate chemistry Part 4. Homoleptic diacetoneglucose complexes of molybdenum and tungsten: chiral ligands associated with an MM triple bond☆

C. Floriani, D. Viterbo, G. Gervasio, 1995 .

Carbohydrate metal complexes as ligands for alkali cations

C. Floriani, D. Viterbo, G. Gervasio, 1994 .

Resolution of Racemic N‐Benzyl α‐Amino Acids by Liquid‐Liquid Extraction: A Practical Method Using a Lipophilic Chiral Cobalt(III) Salen Complex and Mechanistic Studies

Toby B. Reeve, I. Tvaroška, C. Gennari, 2008 .

Efficient resolution of racemic N-benzyl beta3-amino acids by iterative liquid-liquid extraction with a chiral (salen)cobalt(III) complex as enantioselective selector.

C. Gennari, P. Dżygiel, U. Piarulli, 2007, Organic & biomolecular chemistry.

A practical approach to the resolution of racemic N-benzyl alpha-amino acids by liquid-liquid extraction with a lipophilic chiral salen-cobalt(III) complex.

Toby B. Reeve, J. D. de Vries, C. Gennari, 2006, Angewandte Chemie.

Combinatorial Libraries: Studies in Molecular Recognition and the Quest for New Catalysts

H. Nestler, C. Gennari, U. Piarulli, 1997 .

2-(2-Hydroxyaryl)cinnamic amides: a new class of axially chiral molecules

N. Masciocchi, S. Galli, U. Piarulli, 2006 .

Rational Design of Antiangiogenic Helical Oligopeptides Targeting the Vascular Endothelial Growth Factor Receptors

F. Formaggio, L. Belvisi, F. Marino, 2019, Front. Chem..

Effects of a novel cyclic RGD peptidomimetic on cell proliferation, migration and angiogenic activity in human endothelial cells

R. Fanelli, M. Cosentino, F. Marino, 2014, Vascular cell.

Combinatorial libraries of chiral ligands for enantioselective catalysis.

C. Gennari, U. Piarulli, 2003, Chemical reviews.

The Importance of Detail: How Differences in Ligand Structures Determine Distinct Functional Responses in Integrin αv β3.

G. Colombo, M. Civera, L. Belvisi, 2019, Chemistry.

Intramolecular Palladium-Catalyzed Aminocarboxylation of Olefins as a Direct Route to Bicyclic Oxazolidinones

S. Galli, G. Broggini, U. Piarulli, 2011 .

Synthesis and Biological Evaluation of RGD and isoDGR–Monomethyl Auristatin Conjugates Targeting Integrin αVβ3

L. Belvisi, C. Steinkühler, D. Arosio, 2019, ChemMedChem.

Conjugates of Cryptophycin and RGD or isoDGR Peptidomimetics for Targeted Drug Delivery

P. Gallinari, C. Steinkühler, M. Frese, 2019, ChemistryOpen.

Tumor Targeting with an isoDGR–Drug Conjugate

L. Belvisi, F. Gasparri, A. Marsiglio, 2017, Chemistry.

Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers.

L. Belvisi, F. Gasparri, F. Sola, 2015, Chemistry.

Cyclic RGD and isoDGR Integrin Ligands Containing cis-2-amino-1-cyclopentanecarboxylic (cis-β-ACPC) Scaffolds

M. Civera, F. Vasile, D. Potenza, 2020, Molecules.

Synthesis and biological evaluation (in vitro and in vivo) of cyclic arginine-glycine-aspartate (RGD) peptidomimetic-paclitaxel conjugates targeting integrin αVβ3.

L. Belvisi, N. Zaffaroni, P. Perego, 2012, Journal of medicinal chemistry.

Kiss and Run: Promoting Effective and Targeted Cellular Uptake of a Drug Delivery Vehicle Composed of an Integrin-Targeting Diketopiperazine Peptidomimetic and a Cell-Penetrating Peptide.

S. Parente, D. Arosio, I. Neundorf, 2019, Bioconjugate chemistry.

Highly enantioselective Rh-catalyzed hydrogenations with heterocombinations of pentafluorobenzyl- and methoxybenzyl-derived binaphthyl phosphites

J. Cvengroš, C. Gennari, U. Piarulli, 2008 .

Solid‐Phase Synthesis of Peptides Containing Reverse‐Turn Mimetic Bicyclic Lactams

D. Potenza, L. Manzoni, C. Gennari, 1999 .

Synthesis and Biological Evaluation of an iso DGR‐Paclitaxel Conjugate Containing a Cell‐Penetrating Peptide to Promote Cellular Uptake

S. Parente, I. Neundorf, Annika Klimpel, 2021 .

Combination of a binaphthol-derived phosphite and a C1-symmetric phosphinamine generates heteroleptic catalysts in Rh- and Pd-mediated reactions.

S. Carboni, L. Pignataro, R. Colombo, 2009, Chemical communications.

Asymmetric Transfer Hydrogenation of Ketones with Modified Grubbs Metathesis Catalysts: On the Way to a Tandem Process

J. G. Vries, L. Pignataro, L. Lefort, 2016 .

SupraBox: Chiral Supramolecular Oxazoline Ligands†

O. Reiser, L. Pignataro, U. Piarulli, 2012 .

A combined fragment-based virtual screening and STD-NMR approach for the identification of E-cadherin ligands

M. Civera, F. Vasile, Chiara Vettraino, 2022, Frontiers in Chemistry.

Asymmetric Hydrogenation of 3-Substituted Pyridinium Salts.

J. D. de Vries, L. Pignataro, L. Lefort, 2016, Chemistry.

Assisted Tandem Catalysis: Metathesis Followed by Asymmetric Hydrogenation from a Single Ruthenium Source

J. G. Vries, L. Pignataro, L. Lefort, 2015 .

A library approach to the development of BenzaPhos: highly efficient chiral supramolecular ligands for asymmetric hydrogenation.

M. Civera, L. Pignataro, C. Gennari, 2012, Chemistry.

Rhodium-catalyzed asymmetric hydrogenation of olefins with PhthalaPhos, a new class of chiral supramolecular ligands.

M. Civera, S. Carboni, L. Pignataro, 2012, Chemistry.

Efficient Synthesis of Amines by Iron‐Catalyzed C=N Transfer Hydrogenation and C=O Reductive Amination

M. Cettolin, L. Pignataro, C. Gennari, 2018 .

Assembling Sugars and Metals: Novel Architectures and Reactivities in Transition Metal Chemistry

C. Floriani, U. Piarulli, 2007 .

A trifunctional steroid-based scaffold for combinatorial chemistry

A. P. Davis, C. Gennari, U. Piarulli, 1999 .

Enantioselective cyanosilylation of aldehydes catalysed by a diastereomeric mixture of atropisomeric thioureas

Federico Andreoli, N. Vanthuyne, C. Roussel, 2006 .

Copper catalysed 1,4-addition of organozinc reagents to α,β-unsaturated carbonyl compounds: a mechanistic investigation

E. Gallo, C. Gennari, U. Piarulli, 2004 .

Microwave-assisted solvent-free synthesis of a quinoline-3,4-dicarboximide library on inorganic solid supports

Nickolas Regalia, S. Gagliardi, U. Piarulli, 2004 .

Bifunctional 2,5‐Diketopiperazines as Efficient Organocatalysts for the Enantioselective Conjugate Addition of Aldehydes to Nitroolefins

M. Civera, C. Gennari, U. Piarulli, 2011 .

Rh-catalyzed enantioselective conjugate addition of arylboronic acids with a dynamic library of chiral tropos phosphorus ligands.

C. Gennari, U. Piarulli, Chiara Monti, 2007, Chemistry.

Enantioselective conjugate addition of phenylboronic acid to enones catalysed by a chiral tropos/atropos rhodium complex at the coalescence temperature.

C. Gennari, U. Piarulli, Chiara Monti, 2005, Chemical communications.

Chiral (cyclopentadienone)iron complexes with a stereogenic plane as pre-catalysts for the asymmetric hydrogenation of polar double bonds

V. Colombo, M. Cettolin, L. Pignataro, 2019, Tetrahedron.

Improving C=N Bond Reductions with (Cyclopentadienone)iron Complexes: Scope and Limitations

M. Cettolin, L. Pignataro, C. Gennari, 2018, European Journal of Organic Chemistry.

Chiral (Cyclopentadienone)iron Complexes for the Catalytic Asymmetric Hydrogenation of Ketones

A. Forni, J. G. Vries, L. Pignataro, 2015 .

Rh-catalyzed asymmetric hydrogenation of prochiral olefins with a dynamic library of chiral TROPOS phosphorus ligands.

J. D. de Vries, L. Lefort, C. Gennari, 2005, Chemistry.

Rh-catalysed asymmetric hydrogenations with a dynamic library of chiral tropos phosphorus-ligands

C. Gennari, U. Piarulli, Chiara Monti, 2004 .

Bifunctional 2,5‐Diketopiperazines as Rigid Three‐Dimensional Scaffolds in Receptors and Peptidomimetics

Ana S Ressurreição, C. Gennari, U. Piarulli, 2011 .

Expanding the Catalytic Scope of (Cyclopentadienone)iron Complexes to the Hydrogenation of Activated Esters to Alcohols

L. Pignataro, L. Lefort, C. Gennari, 2016 .

Synthesis of (R)-BINOL-Derived (Cyclopentadienone)iron Complexes and Their Application in the Catalytic Asymmetric Hydrogenation of Ketones

J. G. Vries, L. Pignataro, L. Lefort, 2015 .

Ureas: New efficient Lewis base catalysts for the allylation of aldehydes

I. Chataigner, C. Gennari, U. Piarulli, 1999 .

Transition metal–carbohydrate chemistry. Part 2. Homoleptic diacetoneglucose complexes of aluminium and Group 4 metals

C. Rizzoli, C. Floriani, A. Chiesi-Villa, 1994 .

Synthetic studies on the sarcodictyins: synthesis of fully functionalized cyclization precursors

S. Ceccarelli, C. Gennari, U. Piarulli, 2001 .

Enantioselective Reductions Promoted by (Cyclopentadienone)iron Complexes.

L. Pignataro, U. Piarulli, Sofia Vailati Fachini, 2017, Chimia.

Stereocontrolled synthesis of polyketide libraries: Boron-mediated aldol reactions with aldehydes on solid support

S. Ceccarelli, M. Donghi, I. Paterson, 1998 .

Synthesis and screening of new chiral ligands for the copper-catalysed enantioselective allylic substitution

C. Gennari, U. Piarulli, S. Ongeri, 2002 .

A catalytic and enantioselective desymmetrization of meso cyclic allylic bisdiethylphosphates with organozinc reagents.

C. Claverie, C. Gennari, U. Piarulli, 2003, Angewandte Chemie.

Copper-catalysed, enantioselective desymmetrisation of meso cyclic allylic bis(diethyl phosphates) with organozinc reagents

C. Claverie, C. Gennari, U. Piarulli, 2005 .

Chiral (salen)Co(III)(N-benzyl-l-serine)-derived phosphites: monodentate P-ligands for enantioselective catalytic applications

S. Carboni, L. Pignataro, C. Gennari, 2009 .

PhthalaPhos: chiral supramolecular ligands for enantioselective rhodium-catalyzed hydrogenation reactions.

M. Civera, S. Carboni, L. Pignataro, 2010, Angewandte Chemie.

Combinations of Acidic and Basic Monodentate Binaphtholic Phosphites as Supramolecular Bidentate Ligands for Enantioselective Rh-Catalyzed Hydrogenations

J. Cvengroš, L. Pignataro, C. Gennari, 2009 .

Discovery of a new efficient chiral ligand for copper-catalyzed enantioselective Michael additions by high-throughput screening of a parallel library

S. Ceccarelli, I. Chataigner, C. Gennari, 2001 .

A carbonylative cross-coupling strategy to the total synthesis of the sarcodictyins: preliminary studies and synthesis of a cyclization precursor

S. Ceccarelli, C. Gennari, J. Telser, 2001 .

A Mixed Ligand Approach for the Asymmetric Hydrogenation of 2-Substituted Pyridinium Salts

J. G. Vries, L. Pignataro, L. Lefort, 2016 .

SYNTHESIS OF COMBINATORIAL LIBRARIES OF VINYLOGOUS SULFONAMIDOPEPTIDES (VS-PEPTIDES)

S. Ceccarelli, C. Gennari, U. Piarulli, 1998 .

A new method for the solution and solid phase synthesis of chiral β-sulfonopeptides under mild conditions

D. Potenza, C. Gennari, U. Piarulli, 1996 .

Synthesis of [Bis(hexamethylene)cyclopentadienone]iron Tricarbonyl and its Application to the Catalytic Reduction of C=O Bonds

M. Cettolin, J. Neudörfl, A. Berkessel, 2017 .

A Long Journey through Organic Chemistry – Celebrating Cesare Gennari's 70th Birthday

L. Pignataro, U. Piarulli, 2022, European Journal of Organic Chemistry.

Cyclic RGD peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands.

Laura Belvisi, Francesca Vasile, Donatella Potenza, 2009, Chemistry.

Rhodium-catalyzed asymmetric reactions with a dynamic library of chiral tropos phosphorus ligands

C. Gennari, U. Piarulli, Chiara Monti, 2006 .

Rhodium‐Catalyzed Asymmetric Reactions with a Dynamic Library of Chiral Tropos Phosphorus Ligands

C. Gennari, U. Piarulli, Chiara Monti, 2006 .

Toward the First Nonpeptidic Molecular Tong Inhibitor of Wild‐Type and Mutated HIV‐1 Protease Dimerization

L. Bannwarth, J. Soulier, S. Sicsic, 2010, ChemMedChem.

Synthesis and Conformational Studies of Peptidomimetics Containing a New Bifunctional Diketopiperazine Scaffold Acting as a β-Hairpin Inducer

M. Civera, L. Belvisi, Ana S Ressurreição, 2008 .

Synthesis and conformational studies of a stable peptidomimetic β-hairpin based on a bifunctional diketopiperazine turn inducer

R. Fanelli, O. Lequin, Isabelle Correia, 2015 .

REDOX CHEMISTRY ASSOCIATED WITH THE COMPLEXATION OF VANADIUM(V) AND TUNGSTEN(VI) BY MESO-OCTAETHYLPOPHYRINOGEN : FORMATION AND CLEAVAGE OF CYCLOPROPAN E UNITS FUNCTIONING AS SHUTTLES OF TWO ELECTRONS

C. Rizzoli, C. Floriani, E. Solari, 1996 .

Hydrogen‐Bonding Donor/Acceptor Scales in β‐Sulfonamidopeptides

D. Potenza, C. Gennari, U. Piarulli, 1998 .

The four-electron oxidation of meso-octaethylporphyrinogen via a metal-mediated dealkylation process: formation of [RuL(PhCN)2][H2L = 5,15-dihydro-5,5,10,15,15,20-hexaethylporphyrin]

C. Rizzoli, C. Floriani, A. Chiesi-Villa, 1994 .

Peptide bond formation using an enzyme mimicking approach

F. Molinari, C. Gennari, U. Piarulli, 1990 .

Enantioselective binding of dipeptides using acyclic receptors

D. Potenza, J. Frey, J. Kilburn, 2001 .

Synthesis, conformational studies and binding properties of acyclic receptors for N-protected amino acids and dipeptides

D. Potenza, J. Frey, J. Kilburn, 2001 .

Cell-penetrating peptides containing 2,5-diketopiperazine (DKP) scaffolds as shuttles for anti-cancer drugs: conformational studies and biological activity.

S. Parente, I. Neundorf, Lucia Feni, 2020, Chemical communications.

Copper phosphoramidite-catalyzed enantioselective desymmetrization of meso-cyclic allylic bisdiethyl phosphates.

B. Feringa, A. Minnaard, C. Claverie, 2003, Organic letters.

A catalytic and enantioselective desymmetrization of meso cyclic allylic bisdiethylphosphates with organozinc reagents.

C. Claverie, C. Gennari, U. Piarulli, 2003, Angewandte Chemie.

Molecular association of normal alkanoic acids with their thallium(I) salts: a new homologous series of fatty acid metal soaps.

O. Reiser, S. Carboni, K. Guitot, 2009 .

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

A. Pahl, D. Arosio, L. Pignataro, 2018, Beilstein journal of organic chemistry.

Cyclative cleavage via solid-phase supported stabilized sulfur ylides: synthesis of macrocyclic lactones

P. Seneci, S. Provera, C. Gennari, 2002 .

Synthetic studies on sarcodictyins and eleutherobin: Synthesis of fully functionalized cyclization precursors

S. Ceccarelli, C. Gennari, U. Piarulli, 1999 .

Computational design of novel peptidomimetic inhibitors of cadherin homophilic interactions.

M. Civera, C. Colombo, E. Parisini, 2015, Organic & biomolecular chemistry.

Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists.

Laura Belvisi, Cesare Gennari, L. Belvisi, 2015, Chemistry.

Cyclic isoDGR peptidomimetics as low-nanomolar αvβ3 integrin ligands.

M. Civera, D. Potenza, L. Belvisi, 2013, Chemistry.

Cyclic isoDGR Peptidomimetics as Low-Nanomolar alphaVbeta3 Integrin Ligands

M. Civera, D. Potenza, L. Belvisi, 2013 .

Conformational switch and multiple supramolecular structures of a newly identified self-assembling protein-mimetic peptide from Pseudomonas aeruginosa YeaZ protein

M. Marelli, S. Pieraccini, G. Bertoni, 2022, Frontiers in Chemistry.

Stereoselective aldol reactions of γ-thiobutyrolactone: The benzaldehyde anomaly.

F. Molinari, C. Gennari, U. Piarulli, 1991 .

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors**

F. Formaggio, L. Belvisi, R. Fanelli, 2015, ChemistryOpen.

Cyclic RGD-peptidomimetics containing bifunctional diketopiperazine scaffolds as new potent integrin ligands.

M. Civera, D. Potenza, L. Belvisi, 2009, Chemistry.

Selective O-acylation of unprotected N-benzylserine methyl ester and O,N-acyl transfer in the formation of cyclo[Asp-Ser] diketopiperazines

R. Colombo, C. Gennari, U. Piarulli, 2010 .

Investigating the Interaction of Cyclic RGD Peptidomimetics with αVβ6 Integrin by Biochemical and Molecular Docking Studies

M. Civera, L. Belvisi, S. Zanella, 2017, Cancers.

Determination of the binding epitope of RGD-peptidomimetics to αvβ3 and α(IIb)β3 integrin-rich intact cells by NMR and computational studies.

Laura Belvisi, Monica Civera, Francesca Vasile, 2013, Organic & biomolecular chemistry.

Insights into the Binding of Cyclic RGD Peptidomimetics to α5β1 Integrin by using Live‐Cell NMR And Computational Studies

M. Civera, F. Vasile, D. Potenza, 2016, ChemistryOpen.

Hydrogen-Borrowing Amination of Secondary Alcohols Promoted by a (Cyclopentadienone)iron Complex

M. Cettolin, L. Pignataro, A. Dal Corso, 2019, Synthesis.

Chiral Iron Complexes in Asymmetric Organic Transformations

G. Fusi, S. Gazzola, U. Piarulli, 2021, Advanced Synthesis & Catalysis.

Discovery of a new efficient chiral ligand for copper-catalyzed enantioselective Michael additions by high-throughput screening of a parallel library.

S. Ceccarelli, I. Chataigner, C. Gennari, 2000, Chemistry.

Acceleration of hemiacetal cleavage through hydrogen bonding: a new synthetic catalyst with balanced conformational flexibility and preorganization

D. Potenza, F. Molinari, C. Gennari, 1991 .

Optimizing the enzymatic release of MMAE from isoDGR-based small molecule drug conjugate by incorporation of a GPLG-PABC enzymatically cleavable linker

G. Mező, Adina Borbély, S. Gazzola, 2023, Frontiers in pharmacology.

Synthesis and Characterization of Hairpin Mimics that Modulate the Early Oligomerization and Fibrillization of Amyloid β‐Peptide

R. Fanelli, O. Lequin, M. Taverna, 2017 .

Foldamers of bifunctional diketopiperazines displaying a β-bend ribbon structure

M. Civera, L. Belvisi, U. Piarulli, 2010 .

Enantioselective Rh-Catalyzed Addition of Arylboronic Acids to N-Tosylarylimines

C. Gennari, U. Piarulli, Chiara Monti, 2007 .

Synthesis and biological evaluation of RGD and isoDGR peptidomimetic-α-amanitin conjugates for tumor-targeting

D. Arosio, L. Pignataro, C. Gennari, 2018, Beilstein journal of organic chemistry.

Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers.

L. Belvisi, F. Gasparri, F. Sola, 2015, Chemistry.