I. Biancofiore

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An ultra-high-affinity small organic ligand of fibroblast activation protein for tumor-targeting applications

D. Neri, Florent Samain, S. Cazzamalli, 2021, Proceedings of the National Academy of Sciences.

Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs.

S. Harper, S. Altamura, N. Gennari, 2016, ACS medicinal chemistry letters.

Sulphide as a leaving group: highly stereoselective bromination of alkyl phenyl sulphides† †Electronic supplementary information (ESI) available: Experimental procedures and spectroscopic characterization for all new compounds, including details of NMR experiments and racemisation study. See DOI: 10

Mauro F. A. Adamo, M. Ruether, H. Ibrahim, 2019, Chemical science.

Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides.

S. Harper, V. Summa, P. Pace, 2018, ACS medicinal chemistry letters.

A deep learning approach for the discovery of tumor-targeting small organic ligands from DNA-Encoded Chemical Libraries

Ian A. Watson, Jianwen A. Feng, S. Cazzamalli, 2023, bioRxiv.

Discovery of 2-(1H-imidazo-2-yl)piperazines as a new class of potent and non-cytotoxic inhibitors of Trypanosoma brucei growth in vitro.

S. Harper, N. Gennari, V. Summa, 2018, Bioorganic & medicinal chemistry letters.

Optimization of 2-(1H-imidazo-2-yl)piperazines series of Trypanosoma brucei growth inhibitors as potential treatment for the second stage of HAT.

S. Harper, N. Gennari, V. Summa, 2020, Bioorganic & medicinal chemistry letters.

Combined Peptide and Small-Molecule Approach toward Nonacidic THIQ Inhibitors of the KEAP1/NRF2 Interaction.

S. Steinbacher, M. Augustin, S. Harper, 2020, ACS medicinal chemistry letters.

Deep Learning Approach for the Discovery of Tumor-Targeting Small Organic Ligands from DNA-Encoded Chemical Libraries

Ian A. Watson, Jianwen A. Feng, S. Cazzamalli, 2023, ACS omega.

Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs.

S. Harper, S. Altamura, N. Gennari, 2016, ACS medicinal chemistry letters.