Anas Al-Khawaja

发表

Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements.

G. Ecker, B. Frølund, R. Clausen, 2017, Advances in neurobiology.

Glial GABA Transporters as Modulators of Inhibitory Signalling in Epilepsy and Stroke.

A. Schousboe, A. Clarkson, P. Wellendorph, 2017, Advances in neurobiology.

Monastrol, a 3,4-dihydropyrimidin-2(1H)-thione, as structural scaffold for the development of modulators for GHB high-affinity binding sites and α1β2δ GABAA receptors.

P. Wellendorph, B. Frølund, M. Damgaard, 2017, European journal of medicinal chemistry.

Structure-Activity Relationship, Pharmacological Characterization, and Molecular Modeling of Noncompetitive Inhibitors of the Betaine/γ-Aminobutyric Acid Transporter 1 (BGT1).

G. Ecker, A. Schousboe, P. Wellendorph, 2017, Journal of medicinal chemistry.

Pharmacological Characterization of [3H]ATPCA as a Substrate for Studying the Functional Role of the Betaine/GABA Transporter 1 and the Creatine Transporter.

C. Bundgaard, P. Wellendorph, B. Frølund, 2017, ACS chemical neuroscience.

Demonstration of the dynamic mass redistribution label-free technology as a useful cell-based pharmacological assay for endogenously expressed GABAA receptors

P. Wellendorph, Anas Al-Khawaja, A. Klein, 2016 .

Molecular Determinants and Pharmacological Analysis for a Class of Competitive Non-transported Bicyclic Inhibitors of the Betaine/GABA Transporter BGT1

S. Shuto, G. Ecker, P. Wellendorph, 2021, Frontiers in Chemistry.

Identification of the First Highly Subtype-Selective Inhibitor of Human GABA Transporter GAT3.

G. Ecker, P. Wellendorph, B. Frølund, 2015, ACS chemical neuroscience.

Exploring the molecular determinants for subtype-selectivity of 2-amino-1,4,5,6-tetrahydropyrimidine-5-carboxylic acid analogs as betaine/GABA transporter 1 (BGT1) substrate-inhibitors

G. Ecker, P. Wellendorph, B. Frølund, 2020, Scientific Reports.

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

P. Wellendorph, B. Frølund, R. Clausen, 2014, Neurochemical Research.

Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements.

G. Ecker, B. Frølund, R. Clausen, 2017, Advances in neurobiology.

Pharmacological Characterization of [3H]ATPCA as a Substrate for Studying the Functional Role of the Betaine/GABA Transporter 1 and the Creatine Transporter.

C. Bundgaard, P. Wellendorph, B. Frølund, 2017, ACS chemical neuroscience.

Pharmacological Identification of a Guanidine-Containing β-Alanine Analogue with Low Micromolar Potency and Selectivity for the Betaine/GABA Transporter 1 (BGT1)

P. Wellendorph, B. Frølund, R. Clausen, 2014, Neurochemical Research.