A. Sadeque

发表

Discovery of a novel trans-1,4-dioxycyclohexane GPR119 agonist series.

S. H. Kim, Michael E. Morgan, Robert M. Jones, 2015, Bioorganic & medicinal chemistry letters.

Discovery and optimization of 5-fluoro-4,6-dialkoxypyrimidine GPR119 agonists.

S. H. Kim, Michael E. Morgan, K. Whelan, 2014, Bioorganic & medicinal chemistry letters.

Pharmaceutical Excipients in Drug–Drug Interaction

Chuan Chen, A. Sadeque, 2010 .

Identification of Human Sulfotransferases Involved in Lorcaserin N-Sulfamate Formation

Chuan Chen, K. Usmani, A. Sadeque, 2016, Drug Metabolism and Disposition.

Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists.

I. Gaidarov, Michael E. Morgan, K. Whelan, 2015, Bioorganic & medicinal chemistry letters.

Multiscale Design of Nanostructured Thermoelectric Coolers: Effects of Contact Resistances

S. Ahmed, Vamsi Gaddipati, M. Z. Rashid, 2015, Journal of Electronic Materials.

Discovery of 2-(((1r,4r)-4-(((4-Chlorophenyl)(phenyl)carbamoyl)oxy)methyl)cyclohexyl)methoxy)acetate (Ralinepag): An Orally Active Prostacyclin Receptor Agonist for the Treatment of Pulmonary Arterial Hypertension.

John W. Adams, A. Blackburn, I. Gaidarov, 2017, Journal of medicinal chemistry.

Kinetics of 5-HT2B Receptor Signaling: Profound Agonist-Dependent Effects on Signaling Onset and Duration

I. Gaidarov, John M Frazer, D. Unett, 2013, The Journal of Pharmacology and Experimental Therapeutics.

Identification of Human UDP-Glucuronosyltransferases Involved in N -Carbamoyl Glucuronidation of Lorcaserin

K. Usmani, A. Sadeque, Weichao G. Chen, 2012 .

(7-Benzyloxy-2,3-dihydro-1H-pyrrolo[1,2-a]indol-1-yl)acetic Acids as S1P1 Functional Antagonists.

A. Blackburn, I. Gaidarov, S. H. Kim, 2014, ACS medicinal chemistry letters.

Fused tricyclic indoles as S1P₁ agonists with robust efficacy in animal models of autoimmune disease.

D. Sengupta, Michael E. Morgan, K. Whelan, 2012, Bioorganic & medicinal chemistry letters.

Discovery of APD371: Identification of a Highly Potent and Selective CB2 Agonist for the Treatment of Chronic Pain.

I. Gaidarov, A. Grottick, Robert M. Jones, 2017, ACS medicinal chemistry letters.

morpholinoethoxy ) phenyl ) benzamide ( APD 791 ) : AHighly Selective 5-Hydroxytryptamine 2 A Receptor Inverse Agonist for the Treatment of Arterial Thrombosis

John W. Adams, D. Connolly, P. Dosa, 2010 .

Interactions of fluoroaniline with a heme-octapeptide of cytochrome c: a 19F NMR study

Toru Shimizu, M. Hatano, A. Sadeque, 1987 .

Identification of Human Cytochrome P450 and Flavin-Containing Monooxygenase Enzymes Involved in the Metabolism of Lorcaserin, a Novel Selective Human 5-Hydroxytryptamine 2C Agonist

K. Usmani, A. Sadeque, Weichao G. Chen, 2012, Drug Metabolism and Disposition.

Interaction of fluoroaniline with cytochrome P-450scc and myoglobin: temperature and pH dependence studies

Toru Shimizu, M. Hatano, A. Sadeque, 1988 .

Identification of Human UDP-Glucuronosyltransferases Involved in N-Carbamoyl Glucuronidation of Lorcaserin

K. Usmani, A. Sadeque, Weichao G. Chen, 2012, Drug Metabolism and Disposition.

Discovery of APD334: Design of a Clinical Stage Functional Antagonist of the Sphingosine-1-phosphate-1 Receptor.

A. Blackburn, David Mills, I. Gaidarov, 2014, ACS medicinal chemistry letters.

Biopharmaceutics permeability classification of lorcaserin, a selective 5-hydroxytryptamine 2C agonist: method suitability and permeability class membership.

Chuan Chen, A. Sadeque, Weichao G. Chen, 2013, Molecular pharmaceutics.

Interaction of fluoroaniline with cytochrome P-450d mutants: Difference absorption spectral studies

Y. Fujii‐Kuriyama, Toru Shimizu, K. Hirano, 1988 .

Fused tricyclic indoles as S1P₁ agonists with robust efficacy in animal models of autoimmune disease.

D. Sengupta, Michael E. Morgan, K. Whelan, 2012, Bioorganic & medicinal chemistry letters.

Identification of Human Cytochrome P450 and Flavin-Containing Monooxygenase Enzymes Involved in the Metabolism of Lorcaserin, a Novel Selective Human 5-Hydroxytryptamine 2C Agonist

K. Usmani, A. Sadeque, Weichao G. Chen, 2012, Drug Metabolism and Disposition.

Discovery of 1a,2,5,5a-tetrahydro-1H-2,3-diaza-cyclopropa[a]pentalen-4-carboxamides as potent and selective CB2 receptor agonists.

I. Gaidarov, Michael E. Morgan, K. Whelan, 2015, Bioorganic & medicinal chemistry letters.