Míriam Andrés

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Application of a phenotypic drug discovery strategy to identify biological and chemical starting points for inhibition of TSLP production in lung epithelial cells

Rosa López, Estrella Lozoya, Stephane Paris, 2018, PloS one.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists I.

M. Calbet, M. Zanuy, P. Eichhorn, 2014, Bioorganic & medicinal chemistry letters.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists III: the role of a hydrogen-bond acceptor in long receptor residence times.

M. Calbet, E. Gómez, R. S. Roberts, 2014, Bioorganic & medicinal chemistry letters.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of bicyclic heteroaromatic acetic acids as potent CRTh2 antagonists II: lead optimization.

M. Calbet, M. Zanuy, P. Eichhorn, 2014, Bioorganic & medicinal chemistry letters.

Synthesis and biological activity of pyrido[3',2':4,5]furo[3,2-d]pyrimidine derivatives as novel and potent phosphodiesterase type 4 inhibitors.

J. Montero, A. Gavaldá, J. Beleta, 2011, European journal of medicinal chemistry.

Pharmacological characterization of CRTh2 antagonist LAS191859: Long receptor residence time translates into long-lasting in vivo efficacy.

M. Calbet, P. Eichhorn, V. García-González, 2016, Pharmacological research.

2-(1H-Pyrazol-1-yl)acetic acids as chemoattractant receptor-homologous molecule expressed on Th2 lymphocytes (CRTh2) antagonists.

M. Lehner, M. Calbet, P. Eichhorn, 2014, European journal of medicinal chemistry.

2-(1H-Pyrazol-4-yl)acetic acids as CRTh2 antagonists.

M. Lehner, M. Calbet, P. Eichhorn, 2013, Bioorganic & medicinal chemistry letters.

4-Amino-7,8-dihydro-1,6-naphthyridin-5(6 H)-ones as Inhaled Phosphodiesterase Type 4 (PDE4) Inhibitors: Structural Biology and Structure-Activity Relationships.

M. Lehner, V. Segarra, P. Eichhorn, 2018, Journal of medicinal chemistry.

Biphenyl Pyridazinone Derivatives as Inhaled PDE4 Inhibitors: Structural Biology and Structure-Activity Relationships.

M. Lehner, V. Segarra, P. Eichhorn, 2016, Journal of medicinal chemistry.

Biaryl analogues of teriflunomide as potent DHODH inhibitors.

P. Pizcueta, N. Godessart, R. F. Reinoso, 2011, Bioorganic & medicinal chemistry letters.

Structure-activity relationships (SAR) and structure-kinetic relationships (SKR) of pyrrolopiperidinone acetic acids as CRTh2 antagonists.

M. Calbet, P. Eichhorn, R. S. Roberts, 2014, Bioorganic & medicinal chemistry letters.

Identification of novel small molecule-based strategies of COL7A1 upregulation and readthrough activity for the treatment of recessive dystrophic epidermolysis bullosa

F. Larcher, O. Genilloud, J. Tormo, 2024, Scientific reports.