R. Fan

发表

Direct assembly of 3,4-difunctionalized benzofurans and polycyclic benzofurans by phenol dearomatization and palladium-catalyzed domino reaction.

Liang Zhang, Zhaomeng Han, Zhiming Li, 2014, Angewandte Chemie.

Selective C3C3 Oxidative Cross‐Coupling between Unactivated Anilines and Indoles

Zhaomeng Han, R. Fan, Linfei Wang, 2010 .

Facile synthesis of 4-acetoxyindoles via PhI(OAc)2-mediated dearomatization of 2-alkynylanilines

Yue Wang, R. Fan, Qiuqin He, 2021 .

PhI(OAc)2 induced intramolecular oxidative bromocyclization of homoallylic sulfonamides with KBr as the bromine source

R. Fan, B. Wang, L. Qin, 2007 .

Metal-controlled cycloaddition of 2-alkynyl-1,4-benzoquinones and styrenyl systems: Lewis acid versus π acid.

Zhiming Li, R. Fan, Li Zhang, 2013, Organic letters.

Formal group insertion into aryl C‒N bonds through an aromaticity destruction-reconstruction process

Dandan Han, R. Fan, Qiuqin He, 2018, Nature Communications.

Self-assembly and proton conductance of organic nanotubes from pillar[5]arenes

Zhenxia Chen, L. Weng, Jun‐Li Hou, 2011 .

One-pot synthesis of diarylamines from two aromatic amines via oxidative dearomatization-imino exchange-reductive aromatization.

R. Fan, Li Zhang, Weibin Wang, 2013, Organic letters.

Accessing N-heteroarylated indoles and benzimidazoles from 2-alkynyl cyclohexadienimines and cyclohexadienones through metal-catalyzed tandem reactions.

Jie Tang, R. Fan, Min Yang, 2012, Chemical communications.

A general and efficient route to 3-amino-4-sulfanylcoumarins via substitution and palladium-catalyzed amination of 3-bromo-4-tosyloxycoumarins

Jie Wu, Q. Ding, R. Fan, 2007 .

1,2- and 1,4-additions of 2-alkynylcyclohexadienimines with aromatic amines to access 4-amino-N-arylindoles and -azepinoindoles.

Zhiming Li, R. Fan, Li Zhang, 2012, Organic letters.

Transition-metal-free intermolecular amination of sp3 C-H bonds with sulfonamides.

R. Fan, D. Pu, Li Zhang, 2009, Organic letters.

Construction of 3-oxyindoles via hypervalent iodine mediated tandem cyclization-acetoxylation of o-acyl anilines.

R. Fan, Yi Sun, 2010, Chemical communications.

FeCl3‐Catalyzed Aza‐Diels–Alder Reactions of Methylenecyclopropanes with Imines

Jie Wu, Huixia Sun, R. Fan, 2007 .

Synthesis of 15N-labeled heterocycles via the cleavage of C-N bonds of anilines and glycine-15N.

Jiwen He, R. Fan, Hao Guo, 2021, Chemical communications.

Recent Advances in Phenol Dearomatization and Its Application in Complex Syntheses

Q. Ding, R. Fan, Y. Ye, 2012, Synthesis.

Chapter 4.3 - Five-Membered Ring Systems: Furans and Benzofurans

Jie Wu, K. Yeung, X. Hou, 2013 .

Synthesis of N-indolated amino acids or peptides from 2-alkynylanilines via a dearomatization process

R. Fan, Yin Liu, W. Qiu, 2021, Organic Chemistry Frontiers.

Design and synthesis of novel desfluoroquinolone-aminopyrimidine hybrids as potent anti-MRSA agents with low hERG activity.

Cai-Guang Yang, Song Yang, Jianfeng Cai, 2020, Bioorganic chemistry.

One-pot synthesis of highly substituted 4-acetonylindoles via sequential dearomatization and silver-catalyzed domino reaction.

Xinhui Feng, Bo Yang, R. Fan, 2014, Organic letters.

Dearomatization strategy and palladium-catalyzed domino reaction: construction of azepino[5,4,3-cd]indoles from 2-alkynylanilines.

C. Zheng, R. Fan, J. Chen, 2014, Organic letters.

Dearomatization strategy of β-enamino ester: construction of indenoazepines via tandem Michael addition/polycyclization.

Jie Tang, R. Fan, Min Yang, 2013, Organic letters.

syn Additions to 4α-Epoxypyranosides: Synthesis of l-Idopyranosides

A. Wei, Gang Cheng, R. Fan, 2007 .

Orthogonal sulfation strategy for synthetic heparan sulfate ligands.

A. Wei, R. Fan, Jihane Achkar, 2005, Organic letters.

PhI(OAc)2/I2 induced aziridination of alkenes with TsNH2 under mild conditions

B. Wang, R. Fan, D. Pu, 2008 .

Amine-Mediated Transimination and Aromatization-Triggered Domino Reaction in the Synthesis of Polyfunctionalized 4-Aminoquinolines.

Zhaomeng Han, R. Fan, Qiuqin He, 2016, Organic letters.

One‐Pot Oxidative Heteroannulations of N‐Sulfonylanilines with Styrenes for the Construction of 5‐Aminocoumaran Derivatives

R. Fan, Linfei Wang, Weixun Li, 2008 .

Dearomatization-Induced Cycloaddition and Aromatization-Triggered Rearrangement: Synthesis of Vertically Expanded Five-Ring Fused Benzofurans.

Dandan Han, R. Fan, Qiuqin He, 2016, Organic letters.

Iodine(III)-induced regioselective carbocyclization of terminal alkynes: a facile approach to prepare 1,1-diiodomethylene substituted cyclic compounds

C. Zheng, R. Fan, Zeyu Wang, 2017 .

Iodine(III)-mediated oxidative cross-coupling of enamines and propargylamines under metal-free conditions: an alternative way to prepare highly substituted 3-pyrrolines.

C. Zheng, R. Fan, Yu Wang, 2015, Organic letters.

Hypervalent iodine-mediated regioselective cyclization of acetylenic malonates: facile synthesis of 1-diiodomethylene indane and cyclopentane derivatives.

C. Zheng, R. Fan, 2011, Chemical communications.

Facile Construction of Oxa‐Aza Spirobicycles via a Tandem Carbon‐Hydrogen Bond Oxidation

R. Fan, Yi Sun, Jianhong Gan, 2011 .

Base-promoted selective β-fragmentation of homoallylamines

R. Fan, Weixun Li, Jianhong Gan, 2010 .

PhIO/Bu4NI mediated oxidative cyclization of amidoalkylation adducts for the synthesis of N-benzoyl aziridines and oxazolines

Hua Wang, R. Fan, Y. Ye, 2010 .

Facile iodine(III)-induced oxidative cycloaddition of N-sulfonyl imines with methylene compounds under neutral conditions

R. Fan, Linfei Wang, Jin Zhang, 2009 .

A one-pot oxidative decarboxylation-Friedel-Crafts reaction of acyclic alpha-amino acid derivatives activated by the combination of iodobenzene diacetate/iodine and iron dust.

R. Fan, B. Wang, Weixun Li, 2008, Organic & biomolecular chemistry.

Efficient Stereoselective Synthesis of Nitrocyclopropanes by the Oxidative Cyclization of Michael Adducts of Nitroolefins with Activated Methylene Compounds

R. Fan, Lingfei Wang, Weixun Li, 2008 .

Iodobenzene Diacetate/Tetrabutylammonium Iodide-Induced Aziridination of N-Tosylimines with Activated Methylene Compounds under Mild Conditions

R. Fan, Y. Ye, 2008 .

Conversion of anilines to chiral benzylic amines via formal one-carbon insertion into aromatic C–N bonds

Lei Li, R. Fan, Qiuqin He, 2020, Nature Communications.

Metal- and solvent-free conditions for the acylation reaction catalyzed by carbon tetrabromide (CBr4)

Jie Wu, Liang Zhang, R. Fan, 2007 .

Tributylphosphine-catalyzed ring-opening reaction of epoxides and aziridines with acetic anhydride

X. Hou, R. Fan, 2003 .

AgOTf-catalyzed three-component reactions of 2-alkynylbenzaldehydes, amines, and diethylphosphite. An efficient route to 2,3-disubstituted-1,2-dihydroisoquinolin-1-ylphosphonates.

Jie Wu, Wei Sun, Q. Ding, 2007, Journal of combinatorial chemistry.

Gold(III) Chloride/Silver Triflate: A Highly Efficient Catalyst for Ring-Opening Reaction of Aziridines with Electron-Rich Arenes

Jie Wu, Wei Sun, R. Fan, 2007 .

Efficient ring-opening reaction of epoxides and aziridines promoted by tributylphosphine in water.

X. Hou, R. Fan, 2003, The Journal of organic chemistry.

Selective synthesis of 2,3-disubstituted-2H-isoindol-1-ylphosphonate and 2,3-disubstituted-1,2-dihydroiso-quinolin-1-ylphosphonate via metal-tuned reaction of alpha-amino (2-alkynylphenyl)methylphosphonate.

Jie Wu, Q. Ding, R. Fan, 2007, The Journal of organic chemistry.

Palladium-catalyzed regioselective cross-coupling reactions of 3 -bromo -4 -tosyloxyquinolin -2 (1H) -one with arylboronic acids. a facile and convenient route to 3,4-disubstituted quinolin-2(1H)-ones

Jie Wu, Zhiyong Wang, R. Fan, 2007 .

Tandem Palladium Catalysis for Rapid Construction of 3,4‐Fused Tricyclic Indoles

Dandan Han, R. Fan, Qiuqin He, 2020 .

Aniline Dearomatization and Silver-Catalyzed [3+3] Dipolar Cycloaddition: Efficient Construction of Oxocino[4,3,2-cd]indoles from 2-Alkynylanilines and 2-Alkynylbenzaldoximes.

Dandan Han, R. Fan, Qiuqin He, 2015, Angewandte Chemie.

Divergent synthesis of 4-amino indoles with free amine groups via tandem reaction of 2-alkynylanilines

R. Fan, Qiuqin He, Xiaohua Li, 2022, Organic Chemistry Frontiers.

Oxidative nucleophilic cyclization of 2-alkynylanilines with thiophenols under metal-free conditions.

Dandan Han, Zhiming Li, R. Fan, 2014, Organic letters.

Accessing bridged bicyclic compounds or meta carbon-functionalized anilines from the dearomatization of anilines

R. Fan, Linfei Wang, Weibin Wang, 2013 .

Tributylphosphine: a remarkable promoting reagent for the ring-opening reaction of aziridines.

R. Fan, L. Dai, X. Hou, 2002, The Journal of organic chemistry.

Metal- and Solvent-Free Conditions for the Acylation Reaction Catalyzed by Carbon Tetrabromide (CBr4).

Jie Wu, Liang Zhang, R. Fan, 2008 .

Aqueous iodine(III)-mediated stereoselective oxidative cyclization for the synthesis of functionalized fused dihydrofuran derivatives.

R. Fan, Linfei Wang, Y. Ye, 2010, The Journal of organic chemistry.

General and efficient route for the synthesis of 3,4-disubstituted coumarins via Pd-catalyzed site-selective cross-coupling reactions.

Jie Wu, Liang Zhang, R. Fan, 2007, The Journal of organic chemistry.

Divergent construction of nitrogen-containing polycyclic compounds with a dearomatization strategy.

R. Fan, Linfei Wang, 2012, Organic letters.

Destruction and Construction: Application of Dearomatization Strategy in Aromatic Carbon-Nitrogen Bond Functionalization.

R. Fan, Linfei Wang, Qiuqin He, 2015, Angewandte Chemie.

Solvent-controlled oxidative cyclization for divergent synthesis of highly functionalized oxetanes and cyclopropanes.

C. Zheng, R. Fan, Y. Ye, 2009, Organic letters.

Recent advances in dearomatization of heteroaromatic compounds.

Q. Ding, R. Fan, Xiaoli Zhou, 2014, Organic & biomolecular chemistry.

δ and α SP3 C-H bond oxidation of sulfonamides with Phi(OAc)2/I2 under metal-free conditions

Jie Wu, R. Fan, F. Wen, 2007 .

Stereoselective construction of highly functionalized azetidines via a [2 + 2]-cycloaddition.

Hua Wang, R. Fan, Y. Ye, 2010, Organic letters.

Stereoselective Synthesis of Acyclic Tetrasubstituted Alkenes from Anilines by Dearomatization and Trimethylenemethane Cycloaddition.

Lei Li, R. Fan, Qiuqin He, 2021, Organic letters.

Application of dearomatization strategy on the synthesis of furoquinolinone and angelicin derivatives.

R. Fan, Li Zhang, Y. Ye, 2012, Organic letters.

Synthesis and Reactivity of 4′-Deoxypentenosyl Disaccharides

M. D. Casselman, A. Wei, Gang Cheng, 2014, The Journal of organic chemistry.

A facile synthesis of N-sulfonyl and N-sulfinyl aldimines under Barbier-type conditions.

R. Fan, F. Wen, D. Pu, 2008, The Journal of organic chemistry.

Tandem Knoevenagel-Michael addition of aryl sulfonimines with diethyl malonate for synthesis of arylidene dimalonates.

Jie Wu, R. Fan, D. Pu, 2007, The Journal of organic chemistry.

Unexpected Ring-opening Reaction of Aziridine with Acetic Anhydride in DMF

Jie Wu, T. Diao, R. Fan, 2007 .

Tributylphosphine-Catalyzed Ring-Opening Reaction of Epoxides and Aziridines with Acetic Anhydride.

X. Hou, R. Fan, 2003 .

Tetrabutylammonium bisulfate: a new effective catalyst for the hydrolysis of aziridines or epoxides.

X. Hou, R. Fan, 2003, Organic & biomolecular chemistry.

Formation of P-ylide under neutral and metal-free conditions: transformation of aziridines and epoxides to conjugated dienes in the presence of phosphine.

X. Hou, R. Fan, L. Dai, 2004, The Journal of organic chemistry.

Selective Synthesis of 2,3-Disubstituted-2H-isoindol-1-ylphosphonate and 2,3-Disubstituted-1,2-dihydroisoquinolin-1-ylphosphonate via Metal-Tuned Reaction of α-Amino (2-Alkynylphenyl)methylphosphonate.

Jie Wu, Q. Ding, R. Fan, 2007 .

Dy(OTf)3-mediated selective substitution of N-(α-benzotriazolyl-alkyl)amides with active methylene compounds for synthesis of benzotriazole derivatives

R. Fan, Jin Zhang, Weixun Li, 2009 .

Iodobenzene-Catalyzed Ortho-Dearomatization and Aromatization-Triggered Rearrangement of 2-Allylanilines: Construction of Indolin-3-ylmethanols with High Diastereoselectivities.

R. Fan, Qiuqin He, Shuo-En Wang, 2017, Organic letters.

Silver-catalyzed synthesis of 4-substituted benzofurans via a cascade oxidative coupling-annulation protocol.

R. Fan, Y. Ye, 2011, Chemical communications.

PhI(OAc)2/I2 Induced Aziridination of Alkenes with TsNH2 under Mild Conditions.

B. Wang, R. Fan, D. Pu, 2008 .

Efficient three-component one-pot benzylation and allylation of aldehydes and amines for synthesis of homobenzylamines and homoallylamines.

Jie Wu, R. Fan, L. Qin, 2007, The Journal of organic chemistry.

Towards Reaction Selectivities of Imines and Aziridines

Jie Wu, X. Hou, Chang-Hua Ding, 2006 .

Facile preparation of beta-fluoro amines by the reaction of aziridines with potassium fluoride dihydrate in the presence of Bu4NHSO4.

Yong‐Gui Zhou, X. Hou, R. Fan, 2004, The Journal of organic chemistry.

PhI(OAc)2-mediated dialkoxylation of 4-aminostyrenes through a dearomatization process under metal-free conditions

R. Fan, Qiuqin He, Weiyi Wang, 2017 .

Synthesis of C7-Functionalized Indoles through an Aromaticity Destruction-Reconstruction Process.

R. Fan, Qiuqin He, Ting Xu, 2022, Organic Letters.

Synthesis of 4-Alkylindoles from 2-Alkynylanilines via Dearomatization- and Aromatization-Triggered Alkyl Migration.

Lei Li, Xiaohua Li, R. Fan, 2021, Organic letters.

Synthesis of 4,7-Difunctionalized Indoles via Imino Exchange and Sulfinyl Migration.

Lei Li, Xiaohua Li, R. Fan, 2020, Organic letters.

Formal group insertion into aryl C‒N bonds through an aromaticity destruction-reconstruction process

Dandan Han, R. Fan, Qiuqin He, 2018, Nature Communications.

Synthesis of chiral N-alkylated indoles through replacement of aniline nitrogen by natural amino acids

Xiaohua Li, R. Fan, Qiuqin He, 2022, Green Synthesis and Catalysis.

Recent Advances in Dearomatization of Heteroaromatic Compounds

Q. Ding, R. Fan, Xiaoli Zhou, 2014 .

Efficient Stereoselective Synthesis of Nitrocyclopropanes by the Oxidative Cyclization of Michael Adducts of Nitroolefins with Activated Methylene Compounds

R. Fan, Lingfei Wang, Weixun Li, 2008 .