Z. Bouaziz

发表

Carbazolequinone induction of caspase-dependent cell death in Src-overexpressing cells.

G. Gillet, A. Aouacheria, B. Néel, 2002, Biochemical pharmacology.

Screening of indeno[1,2-b]indoloquinones by MALDI-MS: a new set of potential CDC25 phosphatase inhibitors brought to light

P. Chaimbault, J. Jose, D. Bagrel, 2016, Journal of enzyme inhibition and medicinal chemistry.

Phenolic indeno[1,2-b]indoles as ABCG2-selective potent and non-toxic inhibitors stimulating basal ATPase activity

Mathieu Marchivie, Joachim Jose, Jean Guillon, 2015, Drug design, development and therapy.

Uncompetitive nanomolar dimeric indenoindole inhibitors of the human breast cancer resistance pump ABCG2.

A. di Pietro, B. Sarkadi, P. Falson, 2020, European journal of medicinal chemistry.

QSAR Model of Indeno[1,2-b]indole Derivatives and Identification of N-isopentyl-2-methyl-4,9-dioxo-4,9-Dihydronaphtho[2,3-b]furan-3-carboxamide as a Potent CK2 Inhibitor

S. Haidar, J. Jose, M. Le Borgne, 2019, Molecules.

Self-Assembled Supramolecular Nanoparticles Improve the Cytotoxic Efficacy of CK2 Inhibitor THN7

F. Perret, J. Jose, M. Le Borgne, 2018, Pharmaceuticals.

Development of Pharmacophore Model for Indeno[1,2-b]indoles as Human Protein Kinase CK2 Inhibitors and Database Mining

A. Poso, T. Laitinen, S. Haidar, 2017, Pharmaceuticals.

Inhibition of Shiga toxin-converting bacteriophage development by novel antioxidant compounds

Karolina Pierzynowska, G. Węgrzyn, L. Saso, 2018, Journal of enzyme inhibition and medicinal chemistry.

Microwave-accelerated multicomponent synthesis and X-ray characterization of novel benzothiadiazinone dioxide derivatives, analogues of Monastrol

S. Bouacida, M. Le Borgne, Z. Bouaziz, 2021, Research on Chemical Intermediates.

Broad-Spectrum Anticancer Activity and Pharmacokinetic Properties of a Prenyloxy-Substituted Indeno[1,2-b]indole Derivative, Discovered as CK2 Inhibitor

J. Jose, M. Le Borgne, Ehab El-Awaad, 2021, Pharmaceuticals.

Synthesis, Spectroscopic Characterization, and In Vitro Antibacterial Evaluation of Novel Functionalized Sulfamidocarbonyloxyphosphonates

M. Le Borgne, Z. Bouaziz, J. Lebreton, 2018, Molecules.

Synthesis and Diels-Alder reactivity of ortho-carbazolequinones.

Z. Bouaziz, N. Walchshofer, Muriel Compain-Batissou, 2004, Chemical & pharmaceutical bulletin.

Crystal structure of 13-phenyl-2,3,4,13-tetrahydro-1H-indazolo[1,2-b]phthalazine-1,6,11-trione

A. Bouraiou, S. Bouacida, M. Le Borgne, 2015, Acta crystallographica. Section E, Crystallographic communications.

Crystal structure of 13-(2-methoxyphenyl)-3,4-dihydro-2H-indazolo[1,2-b]phthalazine-1,6,11(13H)-trione

A. Bouraiou, S. Bouacida, Z. Bouaziz, 2015, Acta crystallographica. Section E, Crystallographic communications.

Indenoindoles and cyclopentacarbazoles as bioactive compounds: synthesis and biological applications.

G. Kirsch, J. Jose, M. Le Borgne, 2013, European journal of medicinal chemistry.

Synthesis and antiproliferative activity of oxazinocarbazole and N,N-bis(carbazolylmethyl)amine derivatives.

I. Kassab, Z. Bouaziz, N. Walchshofer, 2010, European journal of medicinal chemistry.

Candidate Molecule Selection Based on In Silico Predicted ADMET Properties of 12 Indenoindole Derivatives

R. Terreux, A. Pietro, M. Gustin, 2016 .

Ninhydrins inhibit carbonic anhydrases directly binding to the metal ion.

C. Supuran, J. Jose, Silvia Bua, 2020, European journal of medicinal chemistry.

Solubility enhancement of mefenamic acid by inclusion complex with β-cyclodextrin: in silico modelling, formulation, characterisation, and in vitro studies

M. Boutahala, M. Le Borgne, M. Baitiche, 2021, Journal of enzyme inhibition and medicinal chemistry.

Microwave-assisted oxidation of indan-1-ones into ninhydrins

J. Jose, Z. Bouaziz, Christelle Marminon, 2015 .

Cycloadditions of α,β-Unsaturated N,N-Dimethylhydrazones. A Diels-Alder Strategy for the Building of Aza-Hetero Rings

Z. Bouaziz, H. Fillion, F. Pautet, 2001 .

Regiospecific hetero diels-alder synthesis of pyrido[2,3-b]- and pyrido[3,2-b]carbazole-5,11-diones

Z. Bouaziz, H. Fillion, M. Domard, 1997 .

DMAP as a new efficient catalyst for the one-pot synthesis of condensed phthalazines

A. Bouraiou, S. Bouacida, M. Le Borgne, 2017 .

Sequential MCR/Fisher indolization strategy for the construction of polycyclic carbazole derivatives

A. Bouraiou, S. Bouacida, Z. Bouaziz, 2017 .

A one-pot three-component synthesis of novel α-sulfamidophosphonates under ultrasound irradiation and catalyst-free conditions

Z. Bouaziz, J. Lebreton, M. Berredjem, 2015 .

Synthesis, in silico study (DFT, ADMET) and crystal structure of novel sulfamoyloxy-oxazolidinones: Interaction with SARS-CoV-2

K. Bacharı, S. Bouacida, Z. Bouaziz, 2022, Journal of Molecular Structure.

Synthesis, Biological Evaluation and Molecular Modeling of Substituted Indeno[1,2-b]indoles as Inhibitors of Human Protein Kinase CK2

H. Gohlke, J. Delcros, C. Gertzen, 2015, Pharmaceuticals.

Carbazole scaffolds in cancer therapy: a review from 2012 to 2018

S. Yous, Anthony Prandina, M. Le Borgne, 2019, Journal of enzyme inhibition and medicinal chemistry.

Converting potent indeno[1,2-b]indole inhibitors of protein kinase CK2 into selective inhibitors of the breast cancer resistance protein ABCG2.

Joachim Jose, Jean Guillon, A. di Pietro, 2015, Journal of medicinal chemistry.

A One-Pot Three-Component Synthesis of Novel α-Sulfamidophosphonates under Ultrasound Irradiation and Catalyst-Free Conditions.

Z. Bouaziz, J. Lebreton, M. Berredjem, 2015 .

Synthesis of Furnaphth[1, 3]oxazine and Furo[1, 3]oxazinoquinoline Derivatives as Precursors for an o-Quinonemethide Structure and Potential Antitumor Agents

Z. Bouaziz, H. Fillion, M. Bartoli, 1996 .

Synthesis of some naphthoxazine carbolactone derivatives with in vitro cytotoxic and antifungal activities

J. Villard, Z. Bouaziz, H. Fillion, 1991 .

Additions of crotonaldehyde N,N-dimethylhydrazone to p-quinones under ultrasonic and thermal conditions

J. Luche, Z. Bouaziz, H. Fillion, 1995 .

Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α′

J. Jose, K. Niefind, D. Lindenblatt, 2017, Pharmaceuticals.

Carbazole-1,4-diones:Syntheses and Properties

Z. Bouaziz, H. Fillion, P. Nebois, 2000 .

Regiospecific synthesis of pyrido[3,4-b]- and pyrido[4,3-b]carbazole-5,11-dione derivatives. Evaluation of their in vitro antifungal or antiprotozoological activities.

Z. Bouaziz, H. Fillion, A. Pétavy, 1999, Chemical & pharmaceutical bulletin.

The Diels-Alder cycloaddition, an intriguing problem in organic sonochemistry

A. Riera, J. Luche, A. Moyano, 1996 .

Methyl 3-(Quinolin-2-yl)indolizine-1-carboxylate

A. Bouraiou, Z. Bouaziz, Esma Lamera, 2015 .

Synthesis of Carbazolequinone Derivatives as Inhibitors ofToxoplasma gondii Purine Nucleoside Phosphorylase

B. Fenet, Z. Bouaziz, N. Walchshofer, 2002 .

Biologically active carbazole derivatives: focus on oxazinocarbazoles and related compounds

A. di Pietro, S. Døskeland, L. Herfindal, 2015, Journal of Enzyme Inhibition and Medicinal Chemistry.

Diacritic Binding of an Indenoindole Inhibitor by CK2α Paralogs Explored by a Reliable Path to Atomic Resolution CK2α′ Structures

J. Jose, K. Niefind, D. Lindenblatt, 2019, ACS omega.

Ebisilc ® Organosilicate Particles for Innovative Galenic Formulation

Samar, Z. Bouaziz, A. Pensé-Lhéritier, 2017 .

Mannich Reaction of 5‐Hydroxy‐β‐carboline. Application to the Synthesis of Novel Oxazinopyrimidocarboline Derivatives.

I. Kassab, Z. Bouaziz, N. Walchshofer, 2009 .

Mannich Reaction of 5-Hydroxy-b-carboline. Application to the Synthesis of Novel Oxazinopyrimidocarboline Derivatives

I. Kassab, Z. Bouaziz, N. Walchshofer, 2008 .

Regioselectivity in the 1,3‐Dipolar Cycloaddition Reactions of Nitrile Oxides and Organic Azides with Bromocarbazole‐1,4‐diones.

B. Fenet, Z. Bouaziz, N. Walchshofer, 2007 .

Regioselectivity in the 1,3-Dipolar Cycloaddition Reactions of Nitrile Oxides and Organic Azides with Bromocarbazole-1,4-diones

B. Fenet, Z. Bouaziz, N. Walchshofer, 2007 .

Synthesis and Diels—Alder Reactivity of ortho-Carbazolequinones.

Z. Bouaziz, N. Walchshofer, Muriel Compain-Batissou, 2005 .

Regiospecific Hetero Diels‐Alder Synthesis of Pyrido(2,3‐b)‐ and Pyrido(3,2‐b)carbazole‐5,11‐diones.

Z. Bouaziz, H. Fillion, M. Domard, 1997 .

Mechanistic basis of breast cancer resistance protein inhibition by new indeno[1,2-b]indoles

S. Ambudkar, J. Jose, F. Rego, 2021, Scientific Reports.

Synthesis of Mannich bases of 5-hydroxynapthalene-1,8-carbolactone as potential antifungal or antitumor agents.

J. Villard, M. Porte, Z. Bouaziz, 1991, Chemical & pharmaceutical bulletin.

Synthesis, X-ray structure, in silico calculation, and carbonic anhydrase inhibitory properties of benzylimidazole metal complexes

C. Supuran, Silvia Bua, A. Bouraiou, 2018, Journal of enzyme inhibition and medicinal chemistry.

Synthesis, proton NMR stereochemical study and diels-alder reaction of (E)-7-arylidene-2H,6H-naphtho[1,8-bc]furan-2,6-diones

Z. Bouaziz, H. Fillion, H. Pinatel, 1993 .

Synthesis, Proton NMR Stereochemical Study and Diels-Alder Reaction of (E)-7-Arylidene-2H,6H-naphtho(1,8-bc)furan-2,6-diones.

Z. Bouaziz, H. Fillion, H. Pinatel, 1993 .

Unexpected Binding Mode of a Potent Indeno[1,2-b]indole-Type Inhibitor of Protein Kinase CK2 Revealed by Complex Structures with the Catalytic Subunit CK2α and Its Paralog CK2α′

J. Jose, K. Niefind, D. Lindenblatt, 2017, Pharmaceuticals.