N. Walchshofer

发表

Carbazolequinone induction of caspase-dependent cell death in Src-overexpressing cells.

G. Gillet, A. Aouacheria, B. Néel, 2002, Biochemical pharmacology.

Isoflavonoids in non-leguminous families: an update.

R. Terreux, N. Walchshofer, J. Reynaud, 2005, Natural product reports.

Critical residue combinations dictate peptide presentation by MHC class II molecules

C. Rabourdin-Combe, D. Gerlier, Jean‐François Hernandez, 1994, Peptides.

Deoxycholic acid derivatives as inhibitors of P-glycoprotein-mediated multidrug efflux

L. Rocheblave, E. Matera, C. Dumontet, 2016, Steroids.

Unsymmetrical α,ω-end-functionalized oligo(cyclohexylidenes): efficient synthesis and conformational analysis

R. Terreux, S. Radix, N. Walchshofer, 2016 .

Synthesis and Diels-Alder reactivity of ortho-carbazolequinones.

Z. Bouaziz, N. Walchshofer, Muriel Compain-Batissou, 2004, Chemical & pharmaceutical bulletin.

Progesterone–adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux: Design, synthesis, characterization and biological evaluation

L. Rocheblave, E. Matera, C. Dumontet, 2012, Steroids.

Design, synthesis and evaluation of progesterone-adenine hybrids as bivalent inhibitors of P-glycoprotein-mediated multidrug efflux.

C. Dumontet, S. Radix, N. Walchshofer, 2010, Bioorganic & medicinal chemistry letters.

Design of peptide competitors for the MHC class II molecule I-Ak

C. Rabourdin-Combe, D. Gerlier, Jean‐François Hernandez, 1993 .

Synthesis of new steroidal inhibitors of P-glycoprotein-mediated multidrug resistance and biological evaluation on K562/R7 erythroleukemia cells.

L. Rocheblave, E. Matera, C. Dumontet, 2015, Journal of medicinal chemistry.

Synthesis and antiproliferative activity of oxazinocarbazole and N,N-bis(carbazolylmethyl)amine derivatives.

I. Kassab, Z. Bouaziz, N. Walchshofer, 2010, European journal of medicinal chemistry.

A Diels–Alder Strategy for the Building of Imidazo[4,5‐g]quinoline‐4,9‐dione Derivatives

R. Terreux, N. Walchshofer, H. Fillion, 2005 .

Synthesis and antiprotozoal activity of naphthofuranquinones and naphthothiophenequinones containing a fused thiazole ring.

R. Tapia, J. Valderrama, N. Walchshofer, 2003, Bioorganic & medicinal chemistry.

Overexpression, purification and characterization of a hexahistidine-tagged recombinant extended nucleotide-binding domain 1 (NBD1) of the Cryptosporidium parvum CpABC3 for rational drug design.

M. Pélandakis, N. Walchshofer, A. Pétavy, 2007, Molecular and biochemical parasitology.

Synthesis and modulation properties of imidazo[4,5-b]pyridin-7-one and indazole-4,7-dione derivatives towards the Cryptosporidium parvum CpABC3 transporter.

S. Radix, N. Walchshofer, P. Lawton, 2010, European journal of medicinal chemistry.

Formation of bis (Fmoc-amino ethyl)-N-glycine derivatives by reductive amination of Fmoc-amino aldehydes with NaBH3CN

N. Walchshofer, J. Paris, J. Salvi, 1994 .

N,N'-disubstituted cinnamamide derivatives potentiate ciprofloxacin activity against overexpressing NorA efflux pump Staphylococcus aureus 1199B strains.

L. Rocheblave, S. Radix, S. Michalet, 2018, European journal of medicinal chemistry.

Synthesis and Antileishmanial Activity of Indoloquinones Containing a Fused Benzothiazole Ring

R. Tapia, N. Walchshofer, H. Fillion, 2002 .

AN IMPROVED METHODOLOGY FOR THE PREPARATION OF 4,7-DIMETHOXY-1H-BENZIMIDAZOLE, A KEY INTERMEDIATE IN THE SYNTHESIS OF 1-ALKYL-1H-BENZIMIDAZOLE-4,7-DIONES

N. Walchshofer, P. Nebois, Abbass Taleb, 2006 .

Antileishmanial activity of polycyclic derivatives.

R. Terreux, R. Tapia, M. Cuellar, 2005, Parasite.

Study on the hydatid cyst membrane: permeation of model molecules and interactions with drug-loaded nanoparticles.

F. Pirot, Tien-Thanh Nguyen, F. Falson, 2008, International journal of pharmaceutics.

Synthesis and antiprotozoal evaluation of benzothiazolopyrroloquinoxalinones, analogues of kuanoniamine A.

B. Fenet, R. Tapia, N. Walchshofer, 2003, Bioorganic & medicinal chemistry.

Pharmacokinetics of an anthelmintic potential prodrug of a new benzimidazole in gerbil, mouse and sheep

N. Walchshofer, J. Paris, P. Delatour, 1991 .

Anthelmintic activity of 3,6-dibenzyl-2,5-dioxopiperazine, cyclo(L-Phe-L-Phe)

F. Garnier, N. Walchshofer, J. Paris, 1997, Amino Acids.

Biological effects of a dipeptide methyl ester on Echinococcus multilocularis metacestodes in vivo

N. Walchshofer, J. Paris, A. Pétavy, 1993 .

Synthesis of Carbazolequinone Derivatives as Inhibitors ofToxoplasma gondii Purine Nucleoside Phosphorylase

B. Fenet, Z. Bouaziz, N. Walchshofer, 2002 .

In vitro effects of isoprinosine and a dipeptide methyl ester on Echinococcus multilocularis protoscoleces

N. Walchshofer, P. Lawton, M. Sarciron, 2001, Journal of Helminthology.

In vivo morphological damage induced by a new benzimidazole prodrug in Echinococcus multilocularis metacestodes.

N. Walchshofer, J. Paris, A. Pétavy, 1990, Journal of pharmaceutical sciences.

Regioselective N-alkylation of imidazo[4,5-b]pyridine-4-oxide derivatives: an experimental and DFT study

J. Pilmé, S. Radix, N. Walchshofer, 2009 .

Mannich Reaction of 5‐Hydroxy‐β‐carboline. Application to the Synthesis of Novel Oxazinopyrimidocarboline Derivatives.

I. Kassab, Z. Bouaziz, N. Walchshofer, 2009 .

Mannich Reaction of 5-Hydroxy-b-carboline. Application to the Synthesis of Novel Oxazinopyrimidocarboline Derivatives

I. Kassab, Z. Bouaziz, N. Walchshofer, 2008 .

Regioselectivity in the 1,3‐Dipolar Cycloaddition Reactions of Nitrile Oxides and Organic Azides with Bromocarbazole‐1,4‐diones.

B. Fenet, Z. Bouaziz, N. Walchshofer, 2007 .

Regioselectivity in the 1,3-Dipolar Cycloaddition Reactions of Nitrile Oxides and Organic Azides with Bromocarbazole-1,4-diones

B. Fenet, Z. Bouaziz, N. Walchshofer, 2007 .

Synthesis and Diels—Alder Reactivity of ortho-Carbazolequinones.

Z. Bouaziz, N. Walchshofer, Muriel Compain-Batissou, 2005 .

Quinonic derivatives active against Toxoplasma gondii

N. Walchshofer, H. Fillion, A. Pétavy, 2002, Parasitology Research.

Quinonic derivatives active against a virulent strain of Toxoplasma gondii. Synthesis of 2-methylfuro[2,3-g]- and [3,2-g]isoquinolinetriones.

O. Cherkaoui, B. Bibal, N. Walchshofer, 2000, Bioorganic & medicinal chemistry letters.

Benzimidazole-4,7-diones as inhibitors of protozoal (Toxoplasma gondii) purine nucleoside phosphorylase.

N. Walchshofer, A. Pétavy, P. Nebois, 2002, Bioorganic & Medicinal Chemistry Letters.

Solvent- and metal-free hydroboration of alkynes under microwave irradiation

L. Rocheblave, S. Radix, N. Walchshofer, 2020 .

Synthesis and antiproliferative activity of [2-(phthaloylamino)alkyl]triphenyl phosphonium derivatives against K562 cell line

C. Trentesaux, N. Walchshofer, J. Paris, 2001, Anti-cancer drugs.

A STRAIGHTFORWARD SYNTHESIS OF O-PROTECTED 3-HYDROXYPROPANAL DERIVATIVES

N. Walchshofer, J. Paris, J. Salvi, 1994 .

A convenient method for the stereoselective preparation of 3-hydroxy-2-substituted propionaldehyde derivatives, C-terminal precursors for the synthesis of trans-alkene dipeptide isosteres

N. Walchshofer, J. Paris, Philippe Roure, 1995, Letters in Peptide Science.

A Straightforward Synthesis of O-Protected 3-Hydroxypropanal Derivatives.

N. Walchshofer, J. Paris, J. Salvi, 1994 .