Dipesh S. Harmalkar

发表

Methyl 3-(3-(4-(2,4,4-Trimethylpentan-2-yl)phenoxy)-propanamido)benzoate as a Novel and Dual Malate Dehydrogenase (MDH) 1/2 Inhibitor Targeting Cancer Metabolism.

M. Won, Bo-Kyung Kim, B. Ku, 2017, Journal of medicinal chemistry.

AIMP2-DX2 provides therapeutic interface to control KRAS-driven tumorigenesis

Dae Kim, Yuno Lee, Doyeun Kim, 2022, Nature Communications.

Bioactive benzofuran derivatives: moracins A-Z in medicinal chemistry.

Kyeong Lee, R. Naik, Kyusic Jang, 2015, European journal of medicinal chemistry.

Schweinfurthins A–Q: isolation, synthesis, and biochemical properties

Yongseok Choi, Kyeong Lee, Jyotirling R. Mali, 2018, RSC advances.

Fructose-1,6-bisphosphatase Inhibitors: A review of Recent (2000-2017) Advances and Structure-Activity Relationship Studies.

Yongseok Choi, Kyeong Lee, Dipesh S. Harmalkar, 2018, Current medicinal chemistry.

A protecting group-free divergent synthesis of natural benzofurans via one-pot synthesis of 2-bromo-6-hydroxybenzofurans.

Yongseok Choi, Kyeong Lee, Dipesh S. Harmalkar, 2019, Organic & biomolecular chemistry.

An Overview of Saturated Cyclic Ethers: Biological Profiles and Synthetic Strategies

Yongseok Choi, Kyeong Lee, Dipesh S. Harmalkar, 2019, Molecules.

DK-1108 exerts anti-inflammatory activity against phorbol 12-myristate 13-acetate-induced inflammation and protective effect against OVA-induced allergic asthma.

H. Jeong, Ji-won Park, Jung-hee Kim, 2020, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.

Synthesis and Cytotoxicity Studies of Bioactive Benzofurans from Lavandula agustifolia and Modified Synthesis of Ailanthoidol, Homoegonol, and Egonol.

Joong-Won Park, Yongseok Choi, Kyungtae Kim, 2020, Journal of Natural Products.

Novel benzofuran derivative DK-1014 attenuates lung inflammation via blocking of MAPK/AP-1 and AKT/mTOR signaling in vitro and in vivo

H. Jeong, I. Shin, K. Ahn, 2019, Scientific Reports.

Total Synthesis of Gramistilbenoids A, B, and C.

Kyeong Lee, Dipesh S. Harmalkar, Qili Lu, 2018, Journal of natural products.

The novel hypoxia-inducible factor-1α inhibitor IDF-11774 regulates cancer metabolism, thereby suppressing tumor growth

M. Won, Bo-Kyung Kim, G. Hwang, 2017, Cell Death & Disease.

Identification of novel non-nucleoside vinyl-stilbene analogs as potent norovirus replication inhibitors with a potential host-targeting mechanism.

Choongho Lee, Sungjin Lee, Kyeong Lee, 2019, European journal of medicinal chemistry.

Elucidation of Mechanism for Ligand Efficacy at Leukotriene B4 Receptor 2 (BLT2).

Jae-Hong Kim, Minsup Kim, A. Cho, 2020, ACS medicinal chemistry letters.

Total Synthesis of the Neuroprotective Agent Cudraisoflavone J.

Dongho Lee, Yongseok Choi, Kyeong Lee, 2021, Journal of natural products.

Discovery of a novel BLT2 antagonist for the treatment of inflammatory airway diseases.

J. Song, Dipesh S. Harmalkar, Jun-Dong Wei, 2023, European journal of medicinal chemistry.

Chemical induction of the interaction between AIMP2-DX2 and Siah1 to enhance ubiquitination.

Jiwon Kong, Ja-Il Goo, Hossam Nada, 2024, Cell chemical biology.

Natural products as IL‐6 inhibitors for inflammatory diseases: Synthetic and SAR perspective

Hossam Nada, Dipesh S. Harmalkar, Aneesh Sivaraman, 2024, Medicinal research reviews.