Geoffrey A Holdgate

Measurements of binding thermodynamics in drug discovery.

G. Holdgate, W. Ward, Geoffrey A Holdgate, 2005, Drug discovery today.

Kinetic efficiency: the missing metric for enhancing compound quality?

A. Gill, G. Holdgate, Adrian L Gill, 2011, Drug discovery today.

Design and synthesis of novel lactate dehydrogenase A inhibitors by fragment-based lead generation.

Jon Winter, David Whittaker, Gareth Davies, 2012, Journal of medicinal chemistry.

Prevention of MKK6-dependent activation by binding to p38alpha MAP kinase.

Jon Read, Alexander L Breeze, Richard A Norman, 2005, Biochemistry.