M. Kraus

发表

Crystal structure of human dipeptidyl peptidase IV in complex with a decapeptide reveals details on substrate specificity and tetrahedral intermediate formation

Biching Sang, K. Aertgeerts, S. Ye, 2004, Protein science : a publication of the Protein Society.

Small molecule inhibitors reveal PTK6 kinase is not an oncogenic driver in breast cancers

Timothy L. Foley, K. Gajiwala, R. Kania, 2018, PloS one.

Modulation of cellular S1P levels with a novel, potent and specific inhibitor of sphingosine kinase-1.

T. Kasten, J. Chrencik, A. Wittwer, 2012, The Biochemical journal.

Structural and Kinetic Analysis of the Substrate Specificity of Human Fibroblast Activation Protein α*

K. Aertgeerts, Lihong Shi, A. Jennings, 2005, Journal of Biological Chemistry.

Structural Basis for the Autoinhibition and STI-571 Inhibition of c-Kit Tyrosine Kinase*

K. Wilson, Biching Sang, C. Mol, 2004, Journal of Biological Chemistry.

Discovery of novel, potent, and selective inhibitors of 3-phosphoinositide-dependent kinase (PDK1).

S. Kazmirski, M. Hickey, G. Alton, 2011, Journal of medicinal chemistry.

Structural and Biophysical Characterization of the EphB4·EphrinB2 Protein-Protein Interaction and Receptor Specificity*

Manfred Auer, Peter Kuhn, Gye Won Han, 2006, Journal of Biological Chemistry.

Structure and thermodynamic characterization of the EphB4/Ephrin-B2 antagonist peptide complex reveals the determinants for receptor specificity.

P. Kuhn, G. Martiny-Baron, J. Chrencik, 2006, Structure.

Discovery of Potent, Selective, and Peripherally Restricted Pan-Trk Kinase Inhibitors for the Treatment of Pain.

Gareth J Waldron, R. Grimley, M. Andrews, 2018, Journal of medicinal chemistry.

Study of the PDK1/AKT signaling pathway using selective PDK1 inhibitors, HCS, and enhanced biochemical assays.

S. Gridley, G. Alton, M. Gehring, 2011, Analytical biochemistry.

Discovery of Allosteric, Potent, Subtype Selective, and Peripherally Restricted TrkA Kinase Inhibitors.

R. Grimley, J. Bilsland, J. Cui, 2019, Journal of medicinal chemistry.

Drug information specialists.

M. Kraus, K. Brand, 2006, American Journal of Health-System Pharmacy.