Waleed A. Zalloum

发表

Discovery of phenylalanine derivatives as potent HIV-1 capsid inhibitors from click chemistry-based compound library.

Fangfang Zhang, Peng Zhan, Ye Tian, 2018, European journal of medicinal chemistry.

Comparative anti-proliferative effects of potential HER2 inhibitors on a panel of breast cancer cell lines

Mohammad S. Mubarak, Hiba M Zalloum, Waleed A Zalloum, 2019, Breast Cancer.

Comparative QM/MM Molecular Dynamics and Umbrella Sampling Simulations: Interaction of the Zinc-Bound Intermediate Gem-Diolate Trapoxin A Inhibitor and Acetyl-l-lysine Substrate with Histone Deacetylase 8.

Waleed A Zalloum, Waleed A. Zalloum, Needa Zalloum, 2021, The journal of physical chemistry. B.

Discovery and optimizing polycyclic pyridone compounds as anti-HBV agents

Dongwei Kang, P. Zhan, Xinyong Liu, 2020, Expert opinion on therapeutic patents.

Homology modeling of MCH1 receptor and validation by docking/scoring and protein-aligned CoMFA.

M. Taha, Hiba M Zalloum, Waleed A Zalloum, 2009, European journal of medicinal chemistry.

Discovery of new potent human protein tyrosine phosphatase inhibitors via pharmacophore and QSAR analysis followed by in silico screening.

M. Taha, Y. Bustanji, A. Al-Bakri, 2007, Journal of molecular graphics & modelling.

Exploring the Active Center of the LSD1/CoREST Complex by Molecular Dynamics Simulation Utilizing Its Co-crystallized Co-factor Tetrahydrofolate as a Probe

Hiba M Zalloum, Waleed A Zalloum, Waleed A. Zalloum, 2017, J. Chem. Inf. Model..

Novel in vitro and in vivo anti-Helicobacter pylori effects of pomegranate peel ethanol extract

Waleed A Zalloum, T. Aburjai, I. Hamad, 2021, Veterinary world.

Design, synthesis, and mechanism study of dimerized phenylalanine derivatives as novel HIV-1 capsid inhibitors.

E. De Clercq, Dongwei Kang, C. Pannecouque, 2021, European journal of medicinal chemistry.

From design to biological mechanism evaluation of phenylalanine-bearing HIV-1 capsid inhibitors targeting a vital assembly interface

E. De Clercq, Dongwei Kang, C. Pannecouque, 2022, Chinese Chemical Letters.

Discovery of novel "Dual-site" binding oseltamivir derivatives as potent influenza virus neuraminidase inhibitors.

P. Zhan, Xinyong Liu, Waleed A Zalloum, 2020, European journal of medicinal chemistry.

Perception, knowledge and attitude towards influenza vaccine during COVID-19 pandemic in Jordanian population

Waleed A. Zalloum, Eman R Elayeh, Needa Zalloum, 2022, European Journal of Integrative Medicine.

The effect of ferrous ions, calcium ions and citric acid on absorption of ciprofloxacin across caco-2 cells: practical and structural approach

I. Hamdan, Waleed A Zalloum, Dina El-Sabawi, 2018, Drug development and industrial pharmacy.

Novel urate transporter 1 (URAT1) inhibitors: a review of recent patent literature (2016–2019)

Dongwei Kang, P. Zhan, Xinyong Liu, 2019, Expert opinion on therapeutic patents.

Design, Synthesis, and Mechanism Study of Benzenesulfonamide-containing Phenylalanine Derivatives as Novel HIV-1 Capsid Inhibitors with Improved Antiviral Activities.

E. De Clercq, Dongwei Kang, C. Pannecouque, 2020, Journal of medicinal chemistry.

Discovery of novel 1,4-disubstituted 1,2,3-triazole phenylalanine derivatives as HIV-1 capsid inhibitors

Dongwei Kang, P. Zhan, Xinyong Liu, 2019, RSC advances.

Chemical and bacterial reduction of azo-probes: monitoring a conformational change using fluorescence spectroscopy

N. Rattray, M. Jaffar, D. Mansell, 2013 .

RNA knockdown by synthetic peptidyl-oligonucleotide ribonucleases: behavior of recognition and cleavage elements under physiological conditions

M. Zenkova, E. Bichenkova, S. Miles, 2020, Journal of biomolecular structure & dynamics.

Design, synthesis, and antiviral evaluation of novel piperidine-substituted arylpyrimidines as HIV-1 NNRTIs by exploring the hydrophobic channel of NNIBP.

E. De Clercq, Dongwei Kang, C. Pannecouque, 2021, Bioorganic chemistry.

Design, synthesis, and mechanistic investigations of phenylalanine derivatives containing a benzothiazole moiety as HIV-1 capsid inhibitors with improved metabolic stability.

E. De Clercq, Dongwei Kang, C. Pannecouque, 2021, European journal of medicinal chemistry.

Discovery of potent inhibitors of pseudomonal quorum sensing via pharmacophore modeling and in silico screening.

M. Taha, A. Al-Bakri, Waleed A. Zalloum, 2006, Bioorganic & medicinal chemistry letters.

Design, synthesis and structure-activity relationships of 4-phenyl-1H-1,2,3-triazole phenylalanine derivatives as novel HIV-1 capsid inhibitors with promising antiviral activities.

P. Zhan, Xinyong Liu, Chin-Ho Chen, 2020, European journal of medicinal chemistry.

The current progress in the use of boron as a platform for novel antiviral drug design

Shuo Wang, P. Zhan, Xinyong Liu, 2022, Expert opinion on drug discovery.

Discovery of diarylpyrimidine derivatives bearing piperazine sulfonyl as potent HIV-1 nonnucleoside reverse transcriptase inhibitors

E. De Clercq, Dongwei Kang, Boshi Huang, 2023, Communications chemistry.

Discovery and Mechanistic Investigation of Piperazinone Phenylalanine Derivatives with Terminal Indole or Benzene Ring as Novel HIV-1 Capsid Modulators

E. De Clercq, C. Pannecouque, P. Zhan, 2022, Molecules.

Discovery of Novel Dihydrothiopyrano[4,3-d]pyrimidine Derivatives as Potent HIV-1 NNRTIs with Significantly Reduced hERG Inhibitory Activity and Improved Resistance Profiles.

E. De Clercq, Dongwei Kang, C. Pannecouque, 2021, Journal of medicinal chemistry.

Anti-Proliferative Effect of Potential LSD1/CoREST Inhibitors Based on Molecular Dynamics Model for Treatment of SH-SY5Y Neuroblastoma Cancer Cell Line

Hiba M Zalloum, Waleed A Zalloum, M. Zihlif, 2022, bioRxiv.

The effect of Ginkgo biloba and psycho-education on stress, anxiety and fatigue among refugees

L. Tawalbeh, H. Attarian, Waleed A Zalloum, 2018 .

Discovery of novel diarypyrimidine derivatives bearing six-membered non-aromatic heterocycles as potent HIV-1 NNRTIs with improved anti-resistance and drug-like profiles.

E. De Clercq, Dongwei Kang, Boshi Huang, 2023, European journal of medicinal chemistry.