G. Stavrakov

发表

Novel camphane-based anti-tuberculosis agents with nanomolar activity.

I. Doytchinova, V. Valcheva, G. Stavrakov, 2013, European journal of medicinal chemistry.

Cytisine as a scaffold for ortho-diphenylphosphinobenzenecarboxamide ligands for Pd-catalyzed asymmetric allylic alkylation

N. Vassilev, R. Nikolova, B. Shivachev, 2015 .

Galantamine Derivatives as Acetylcholinesterase Inhibitors: Docking, Design, Synthesis, and Inhibitory Activity

I. Doytchinova, M. Atanasova, G. Stavrakov, 2018 .

Docking‐based Design of Galantamine Derivatives with Dual‐site Binding to Acetylcholinesterase

I. Doytchinova, S. Konstantinov, M. Atanasova, 2016, Molecular informatics.

Discovery of a Novel Acetylcholinesterase Inhibitor by Fragment-Based Design and Virtual Screening

I. Doytchinova, S. Konstantinov, M. Atanasova, 2021, Molecules.

A Novel Galantamine-Curcumin Hybrid as a Potential Multi-Target Agent against Neurodegenerative Disorders

I. Doytchinova, I. Valkova, M. Atanasova, 2021, Molecules.

Antioxidant Activity of a Novel Acetylcholinesterase Inhibitor: In Vivo and Ex vivo Studies

I. Doytchinova, M. Atanasova, G. Stavrakov, 2020 .

A Galantamine–Curcumin Hybrid Decreases the Cytotoxicity of Amyloid-Beta Peptide on SH-SY5Y Cells

I. Doytchinova, K. Mladenova, J. Doumanov, 2021, International journal of molecular sciences.

From Central to Axial to Central Chirality: Enantioselective Construction of the trans‐4,5,9,10‐Tetrahydroxy‐9,10‐dihydrophenanthrene System

B. Breit, G. Stavrakov, M. Keller, 2007 .

Highly diastereoselective ortho-lithiation of chiral ferrocenecarboxamides

B. Ivanova, G. Stavrakov, I. Philipova, 2010 .

Synthesis of ferrocene-based amido-phosphine ligands via highly diastereoselective ortho-lithiation and their application in Pd-catalyzed asymmetric allylic alkylations

R. Nikolova, B. Shivachev, G. Stavrakov, 2011 .

SYNTHESIS AND ANTIMYCOBACTERIAL ACTIVITY OF NOVEL MANDELIC ACID DERIVED DIAMIDE

V. Valcheva, G. Stavrakov, I. Philipova, 2014 .

Synthetic piperine amide analogs with antimycobacterial activity

I. Doytchinova, V. Valcheva, G. Stavrakov, 2018, Chemical biology & drug design.

Galantamine derivatives: Synthesis, NMR study, DFT calculations and application in asymmetric catalysis

N. Vassilev, G. Stavrakov, I. Philipova, 2020 .

Theophylline-7-acetic acid derivatives with amino acids as anti-tuberculosis agents.

V. Valcheva, G. Stavrakov, Y. Voynikov, 2014, Bioorganic & Medicinal Chemistry Letters.

CYTOTOXICITY ASSAY ON SEVERAL THEOPHYLLINE-7-ACETIC ACID AMIDES WITH AMINO ACIDS

G. Stavrakov, Y. Voynikov, G. Momekov, 2014 .

PARA-AMINOSALICYLIC ACID - BIOPHARMACEUTICAL, PHARMACO- LOGICAL, AND CLINICAL FEATURES AND RESURGENCE AS AN ANTI- TUBERCULOUS AGENT

D. Momekova, G. Stavrakov, Y. Voynikov, 2015 .

SYNTHESIS AND PHARMACOLOGICAL PROPERTIES OF GLUTAMIC ACID AMIDES: A REVIEW

G. Stavrakov, Y. Voynikov, P. Peikov, 2012 .

Galantamine-Curcumin Hybrids as Dual-Site Binding Acetylcholinesterase Inhibitors

I. Doytchinova, Z. Zhivkova, S. Konstantinov, 2020, Molecules.

Design, Synthesis, and Antimycobacterial Activity of Novel Theophylline‐7‐Acetic Acid Derivatives With Amino Acid Moieties

I. Doytchinova, S. Konstantinov, M. Atanasova, 2016, Chemical biology & drug design.

Design of novel camphane-based derivatives with antimycobacterial activity.

I. Doytchinova, V. Valcheva, G. Stavrakov, 2014, Journal of molecular graphics & modelling.

Novel hits for acetylcholinesterase inhibition derived by docking-based screening on ZINC database

Irini Doytchinova, Ivan Dimitrov, Irena Philipova, 2018, Journal of enzyme inhibition and medicinal chemistry.

Docking‐based design and synthesis of galantamine–camphane hybrids as inhibitors of acetylcholinesterase

I. Doytchinova, I. Valkova, S. Konstantinov, 2017, Chemical biology & drug design.

Galantamine derivatives with indole moiety: Docking, design, synthesis and acetylcholinesterase inhibitory activity.

I. Doytchinova, M. Atanasova, G. Stavrakov, 2015, Bioorganic & medicinal chemistry.

Cytisine as a Scaffold for ortho-Diphenylphosphinobenzenecarboxamide Ligands for Pd-Catalyzed Asymmetric Allylic Alkylation.

N. Vassilev, R. Nikolova, B. Shivachev, 2015 .

Antimycobacterial activity of chiral aminoalcohols with camphane scaffold.

I. Doytchinova, M. Stoyanova, V. Valcheva, 2014, European journal of medicinal chemistry.

Synthesis and antimycobacterial activity of novel camphane-based agents.

V. Valcheva, G. Stavrakov, I. Philipova, 2014, Bioorganic & medicinal chemistry letters.

Synthesis and absolute configuration of planar chiral ferrocenophanes by amide-directed ortho-lithiation

S. Simova, G. Stavrakov, V. Dimitrov, 2008 .

3 ANtIMYcoBActeRIAL ActIVItY oF 4-AND 3 , 4-sUBstItUteD coUMARINs

V. Angelova, V. Valcheva, G. Stavrakov, 2015 .

Ex Vivo Antioxidant and Cholinesterase Inhibiting Effects of a Novel Galantamine–Curcumin Hybrid on Scopolamine-Induced Neurotoxicity in Mice

I. Doytchinova, M. Atanasova, Rumyana Simeonova, 2022, International journal of molecular sciences.

Biochemical Studies on a Novel Potent Acetylcholinesterase Inhibitor with Dualsite Binding for Treatment of Alzheimer’s Disease

I. Doytchinova, I. Valkova, V. Vitcheva, 2021 .

In Vivo Studies on Novel Potent Acetylcholinesterase Inhibitors with Dual-site Binding for Treatment of Alzheimer’s Disease

I. Doytchinova, I. Valkova, V. Vitcheva, 2021 .

Camphane-based phosphino-carboxamide ligands as P,O-chelates in Pd-catalyzed enantioselective allylic alkylation

G. Stavrakov, I. Philipova, V. Dimitrov, 2012 .

Docking‐based design and synthesis of galantamine–camphane hybrids as inhibitors of acetylcholinesterase

I. Doytchinova, I. Valkova, S. Konstantinov, 2017, Chemical biology & drug design.

A galantamine–curcumin hybrid lacks the depressant side effect of acetylcholinesterase inhibitors

I. Doytchinova, M. Atanasova, G. Stavrakov, 2024, Biotechnology & Biotechnological Equipment.

Galantamine derivatives with indole moiety: Docking, design, synthesis and acetylcholinesterase inhibitory activity.

I. Doytchinova, M. Atanasova, G. Stavrakov, 2015, Bioorganic & medicinal chemistry.