Matjaž Brvar

发表

Discovery of Mono‐ and Disubstituted 1H‐Pyrazolo[3,4]pyrimidines and 9H‐Purines as Catalytic Inhibitors of Human DNA Topoisomerase IIα

M. Filipič, T. Šolmajer, A. Perdih, 2015, ChemMedChem.

Universitet Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR 91

T. Schwartz, T. Frimurer, C. Monaco, 2022 .

Linker-switch approach towards new ATP binding site inhibitors of DNA gyrase B.

J. Ilaš, M. Anderluh, D. Kikelj, 2017, European journal of medicinal chemistry.

N-Phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATP Competitive DNA Gyrase B Inhibitors: Design, Synthesis, and Evaluation.

J. Ilaš, T. Šolmajer, T. Tomašič, 2015, Journal of medicinal chemistry.

Structure-Activity Investigations and Optimisations of Non-metabolite Agonists for the Succinate Receptor 1

T. Schwartz, T. Frimurer, Matjaž Brvar, 2018, Scientific Reports.

Discovery of the first inhibitors of bacterial enzyme D-aspartate ligase from Enterococcus faecium (Aslfm).

J. Mainardi, S. Magnet, M. Arthur, 2013, European journal of medicinal chemistry.

In silico discovery and biophysical evaluation of novel 5-(2-hydroxybenzylidene) rhodanine inhibitors of DNA gyrase B.

Roman Jerala, Andrej Perdih, Vesna Hodnik, 2012, Bioorganic & medicinal chemistry.

Structure–Activity Relationship Studies of Tetrahydroquinolone Free Fatty Acid Receptor 3 Modulators

B. Hudson, G. Milligan, A. Tobin, 2020, Journal of medicinal chemistry.

Receptor structure-based discovery of non-metabolite agonists for the succinate receptor GPR91

T. Schwartz, T. Frimurer, C. Monaco, 2017, Molecular metabolism.

Discovery of 4,5,6,7-Tetrahydrobenzo[1,2-d]thiazoles as Novel DNA Gyrase Inhibitors Targeting the ATP-Binding Site.

J. Ilaš, M. Anderluh, T. Šolmajer, 2015, Journal of medicinal chemistry.

Discovery of substituted oxadiazoles as a novel scaffold for DNA gyrase inhibitors.

J. Ilaš, T. Tomašič, D. Kikelj, 2017, European journal of medicinal chemistry.

In silico discovery of 2-amino-4-(2,4-dihydroxyphenyl)thiazoles as novel inhibitors of DNA gyrase B.

Andrej Perdih, Marko Oblak, T. Šolmajer, 2010, Bioorganic & medicinal chemistry letters.

Design, Synthesis, and Evaluation of Novel Tyrosine‐Based DNA Gyrase B Inhibitors

J. Ilaš, D. Kikelj, R. Frlan, 2017, Archiv der Pharmazie.

Structure-based discovery of substituted 4,5'-bithiazoles as novel DNA gyrase inhibitors.

D. Turk, G. Anderluh, M. Renko, 2012, Journal of medicinal chemistry.

Monocyclic 4-amino-6-(phenylamino)-1,3,5-triazines as inhibitors of human DNA topoisomerase IIα.

Andrej Perdih, Metka Filipič, M. Filipič, 2014, Bioorganic & medicinal chemistry letters.

Molecular Mechanism of Action for Allosteric Modulators and Agonists in CC-chemokine Receptor 5 (CCR5)*

T. Frimurer, M. Rosenkilde, A. Pui, 2016, The Journal of Biological Chemistry.

3‐substituted‐1H‐indazoles as Catalytic Inhibitors of the Human DNA Topoisomerase IIα

T. Šolmajer, A. Perdih, B. Pogorelčnik, 2017 .

Selective Allosteric Modulation of N-Terminally Cleaved, but Not Full Length CCL3 in CCR1.

T. Frimurer, M. Rosenkilde, T. Ulven, 2019, ACS pharmacology & translational science.

New N-phenyl-4,5-dibromopyrrolamides and N-Phenylindolamides as ATPase inhibitors of DNA gyrase.

J. Ilaš, T. Tomašič, Nace Zidar, 2016, European journal of medicinal chemistry.

Syddansk Universitet Molecular Mechanism of Action for Allosteric Modulators and Agonists in CC-chemokine Receptor 5 ( CCR 5 )

T. Frimurer, M. Rosenkilde, A. Pui, 2016 .