Qiu-Qin He

发表

Chiral resolution, absolute configuration assignment and biological activity of racemic diarylpyrimidine CH(OH)-DAPY as potent nonnucleoside HIV-1 reverse transcriptase inhibitors.

E. De Clercq, C. Pannecouque, Xiaodong Ma, 2012, European journal of medicinal chemistry.

Synthesis and biological evaluation of DAPY-DPEs hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase.

E. De Clercq, C. Pannecouque, D. Daelemans, 2015, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of new conformationally restricted S-DABO hybrids as non-nucleoside inhibitors of HIV-1 reverse transcriptase

C. Pannecouque, J. Balzarini, E. Clercq, 2014 .

An efficient enantioselective synthesis of florfenicol via a vanadium-catalyzed asymmetric epoxidation

Fangjun Xiong, Fener Chen, Qiu-Qin He, 2011 .

Asymmetric synthesis of the HMG-CoA reductase inhibitor atorvastatin calcium: an organocatalytic anhydride desymmetrization and cyanide-free side chain elongation approach.

Fangjun Xiong, Fener Chen, Xiaofei Chen, 2014, The Journal of organic chemistry.

An efficient enantioselective synthesis of florfenicol via asymmetric aziridination

C. Zheng, Fener Chen, Qiu-Qin He, 2011 .

Synthesis and Anti‐HIV Activity of Aryl‐2‐[(4‐cyanophenyl)amino]‐4‐pyrimidinone hydrazones as Potent Non‐nucleoside Reverse Transcriptase Inhibitors

C. Pannecouque, Xiaodong Ma, J. Balzarini, 2011, ChemMedChem.

Design, synthesis and biological evaluation of cycloalkyl arylpyrimidines (CAPYs) as HIV-1 NNRTIs.

C. Pannecouque, Xiaodong Ma, J. Balzarini, 2011, Bioorganic & medicinal chemistry.

Synthesis, structure-activity relationships, and docking studies of N-phenylarylformamide derivatives (PAFAs) as non-nucleoside HIV reverse transcriptase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Liu-meng Yang, 2012, European journal of medicinal chemistry.

Synthesis and structure-activity relationship of novel diarylpyrimidines with hydromethyl linker (CH(OH)-DAPYs) as HIV-1 NNRTIs.

E. De Clercq, C. Pannecouque, Xiaodong Ma, 2011, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of (±)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Liu-meng Yang, 2011, Bioorganic & medicinal chemistry.

Synthesis and biological activity of naphthyl-substituted (B-ring) benzophenone derivatives as novel non-nucleoside HIV-1 reverse transcriptase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Liu-meng Yang, 2011, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of naphthyl phenyl ethers (NPEs) as novel nonnucleoside HIV-1 reverse transcriptase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Liu-meng Yang, 2011, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of HQCAs with aryl or benzyl substituents on N-1 position as potential HIV-1 integrase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Liu-meng Yang, 2011, Bioorganic & medicinal chemistry.

Structural modifications of quinolone-3-carboxylic acids with anti-HIV activity.

Yong-tang Zheng, Liu-meng Yang, Fener Chen, 2011, Bioorganic & medicinal chemistry.

Organocatalytic asymmetric [3 + 3] annulations of 3-carboxamide oxindoles with β,γ-unsaturated α-keto esters: facile access to chiral spiro-δ-lactam oxindoles

Dan Yang, Lin-Hai Jing, Qiu-Qin He, 2023, Organic Chemistry Frontiers.

Organocatalytic asymmetric synthesis of trans -configured trispirooxindoles through a cascade Michael-cyclization reaction

Lin-Hai Jing, Qiu-Qin He, Chaoling Wu, 2016 .

Hybrid diarylbenzopyrimidine non-nucleoside reverse transcriptase inhibitors as promising new leads for improved anti-HIV-1 chemotherapy.

E. De Clercq, C. Pannecouque, J. Balzarini, 2010, Bioorganic & medicinal chemistry.

Synthesis and anti-HIV activity of 2-naphthyl substituted DAPY analogues as non-nucleoside reverse transcriptase inhibitors.

C. Pannecouque, J. Balzarini, E. Clercq, 2010, Bioorganic & medicinal chemistry.

Synthetic studies on statins. Part 1: a short and cyanide-free synthesis of atorvastatin calcium via an enantioselective aldol strategy

Fangjun Xiong, Fener Chen, Xiaofei Chen, 2013 .

An Efficient EnantioselectiveSynthesis of Florfenicol Based on Sharpless Asymmetric Dihydroxylation

C. Zheng, Fener Chen, Qiu-Qin He, 2012 .

Towards new C6-rigid S-DABO HIV-1 reverse transcriptase inhibitors: synthesis, biological investigation and molecular modeling studies.

E. De Clercq, C. Pannecouque, J. Balzarini, 2013, Bioorganic & Medicinal Chemistry.

Synthesis and biological evaluation of 5-fluoroquinolone-3-carboxylic acids as potential HIV-1 integrase inhibitors

Yong-tang Zheng, Liu-meng Yang, Fen‐er Chen, 2013, Journal of enzyme inhibition and medicinal chemistry.

Development of an Efficient Process for the Decomposition of the Borate Complexes Formed during the Large-Scale Synthesis of (S)-1,2,4-Butanetriol

Fangjun Xiong, Qiu-Qin He, Fener Chen, 2013 .

Structural modifications of CH(OH)-DAPYs as new HIV-1 non-nucleoside reverse transcriptase inhibitors.

Christophe Pannecouque, E. De Clercq, C. Pannecouque, 2014, Bioorganic & medicinal chemistry.

Anti-HIV diarylpyrimidine-quinolone hybrids and their mode of action.

E. De Clercq, C. Pannecouque, D. Daelemans, 2015, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of CHX-DAPYs as HIV-1 non-nucleoside reverse transcriptase inhibitors.

Christophe Pannecouque, E. De Clercq, C. Pannecouque, 2014, Bioorganic & medicinal chemistry.

Synthesis and biological evaluation of (±)-benzhydrol derivatives as potent non-nucleoside HIV-1 reverse transcriptase inhibitors.

Xiaodong Ma, Yong-tang Zheng, Fener Chen, 2011, Bioorganic & medicinal chemistry.