M. Robba

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A New and Efficient Synthesis of 4-Arylimidazolidin-2-ones

S. Rault, P. Dallemagne, M. Robba, 1991 .

A New and Efficient Synthesis of 4-Arylimidazolidin-2-ones.

S. Rault, P. Dallemagne, M. Robba, 1991 .

Synthesis of new thienocyclopenta[3,2‐d]‐oxazole and thiazole derivatives

S. Rault, M. Boulouard, P. Dallemagne, 1993 .

Synthesis and evaluation of the CNS activity of new 4-alkoxyphenylimidazolidin-2-ones.

S. Rault, M. Boulouard, O. Renault, 1998, Chemical & pharmaceutical bulletin.

Design, Synthesis and Antiviral Activity of New Pyridinone Derivatives

R. Bureau, A. Aubertin, A. Kirn, 1997 .

Comparative molecular field analysis of CCK-B antagonists

S. Rault, R. Bureau, M. Robba, 1994 .

Comparative molecular field analysis of CCK-A antagonists using field fit as alignment technique

S. Rault, R. Bureau, M. Robba, 1993 .

Novel selective and partial agonists of 5-HT3 receptors. Part 1. Synthesis and biological evaluation of piperazinopyrrolothienopyrazines.

P Delagrange, M. Hamon, B. Guardiola-Lemaitre, 1996, Journal of medicinal chemistry.

Thiaisatoic anhydrides: Efficient synthesis under microwave heating conditions and study of their reactivity

S. Rault, F. Fabis, M. Robba, 1998 .

Comparative Molecular Field Analysis of Chlorophenols. application in Ecotoxicology

S. Rault, R. Bureau, F. Briens, 1994 .

Synthesis, Crystal Structure and Interaction With DNA of N,N′-(Butane-1,4-Diyl)Bis(Guanidinium) Tetrachloroplatinate (II)

C. Bailly, G. Morgant, N. Dung, 1998, Metal-based drugs.

Highly Potent and Selective Ligands for a New Class H3 of Histamine Receptor

J. Schwartz, J. Arrang, J. Lecomte, 1988, Investigative radiology.

Synthesis and antiviral study of dihydrothieno and thianopyrimidine diones acyclic nucleosides as potential anti-HIV agents

M. Robba, J. Renault, D. Ladurée, 1994 .

Synthesis of thieno[3,2-d]pyrimidine-2,4-diones cyclic and acyclic nucleosides as potential anti HIV agents

M. Robba, F. Jourdan, D. Ladurée, 1994 .

Effect of cetiedil analogs on acetylcholine and choline fluxes in synaptosomes and vesicles.

M. Robba, M. Diebler, M. Israël, 1989, European journal of pharmacology.

Synthesis and antiviral study of cyclopentano [d] pyrimidine-2,4-diones and octahydroquinazoline-2,4-diones acyclic nucleosides as potential anti-HIV agents

M. Robba, J. Renault, D. Ladurée, 1994 .

New arylhexahydropyrimidinediones: Synthesis, benzodiazepine receptor affinity and anticonvulsant activity

S. Rault, M. Boulouard, P. Dallemagne, 1996 .

Pyrrolothieno[1,4]diazepines Part 1 : Synthesis and Study of the Reaction Pathway

S. Rault, M. Boulouard, P. Dallemagne, 1995 .

Synthesis and evaluation of antileukemic activity of 5-thienyl- or 5-(2-furyl)-2,3-dihydro-6,7-bis(hydroxymethyl)-1H-pyrrolizine bis(alkylcarbamates) and derivatives.

G. Mathé, J. Lancelot, M. Robba, 1989, Journal of Medicinal Chemistry.

[SYNTHESIS OF THIAZOLES AND ISOTHIAZOLES. STUDY OF THEIR ACTION ON TRICHOMONAS VAGINALIS AND CANDIDA ALBICANS].

M. Robba, R. Moreau, 1964, Annales Pharmaceutiques Françaises.

Synthesis of Trans-thienyl-3-ethoxycarbonyl-2,3-dihydro[1,5]benzothiazepin-4(5h)-ones

C. Saturnino, J. Lancelot, P. D. Caprariis, 1992 .

A novel synthesis of methyl cis-(3-thienyl)glycidate with 2-aminothiophenol and the synthesis of [1,5]benzothiazepine derivatives

S. Rault, C. Saturnino, J. Lancelot, 1992 .

A NOVEL SYNTHESIS OF 2,3-DIHYDRO[1,5]BENZOTHIAZEPIN-4(5H)-ONES

J. Lancelot, P. D. Caprariis, M. Robba, 1992 .

[1]Benzothienopyrimidines. II. Study of the electrophilic substitutions of [1]benzothieno[3,2-d]pyrimidine and [1]benzothieno[3,2-d]pyrimidin-4-(3H)one

S. Rault, H. El-Kashef, M. Robba, 1980 .

Synthesis and pharmacological activities of some 2,3,4,5-tetrahydro[1,5]benzo[f]thiazepines.

S. Rault, C. Saturnino, G. de Martino, 1997, Farmaco.

Preparation of 2,3-Dihydro [1,5] Benzothiazepines and 2,3-Dihydro [1,5] Benzodiazepines

C. Saturnino, J. Lancelot, M. Robba, 1991 .

Amoebicidal efficiencies of various diamidines against two strains of Acanthamoeba polyphaga

C. Saturnino, M. Robba, J. Lancelot, 1995, Antimicrobial agents and chemotherapy.

New synthesis of isopiperitenol, previously isolated from species of Cymbopogon

J. Guillon, M. Robba, J. Rioult, 2000 .

Cyclisation de l'acide amino-3 (thienyl-3)-3 propionique en aminocyclopentathiophenes

S. Rault, M. Robba, K. Hassan, 1986 .

Pyrido [2, 3-h] pyrrolo [1, 2-a] quinoxalines

S. Rault, J. Lancelot, M. Robba, 1983 .

Synthesis of N-1β-D-Arabinofuranosyl and N-1-2′-Deoxy-β-D-erythro-pentofuranosyl Thieno [3,2-d] Pyrimidine Nucleosides

M. Robba, C. Fossey, D. Ladurée, 1994 .

Synthesis of phenylpyrrolylpyrroles. Part II

S. Rault, M. Robba, H. Dumoulin, 1996 .

Novel and selective partial agonists of 5-HT3 receptors. 2. Synthesis and biological evaluation of piperazinopyridopyrrolopyrazines, piperazinopyrroloquinoxalines, and piperazinopyridopyrroloquinoxalines.

P Delagrange, M. Hamon, P. Renard, 1997, Journal of medicinal chemistry.

Efficient synthesis of 6H-pyrido [3,2-b] carbazole derivatives from 3-amino-1,4-dimethyl carbazole

S. Rault, J. Lancelot, M. Robba, 1987 .

Synthesis and Anti-HSV-1 Activity of New 3-Amino-3-Arylpropionic Acid Esters

S. Rault, J. Boustie, P. Dallemagne, 1996 .

FIRST SYNTHESIS OF 4-AMINO-4,5-DIHYDRO-1-PHENYLCYCLOPENTA[ b]PYRROL-6(1H)-ONES

S. Rault, P. Dallemagne, F. Fabis, 1994 .

Effective cerebral antihypoxic activity of new aminocyclopentanones

S. Rault, P. Dallemagne, M. Robba, 1992 .

One-Pot Cyclization of Alkoxy-3-aminoindan-1-ones.

S. Rault, P. Dallemagne, M. Robba, 1991 .

Cyclisation of 3-Amino-3-[thienyl-3]-propionic Acid to Aminocyclopentathiophenes.

S. Rault, P. Dallemagne, M. Robba, 1986 .

Amide derivatives with H1-antihistaminic effect.

C. Saturnino, G. de Martino, M. Robba, 1998, Pharmaceutica acta Helvetiae.

Synthesis of [1]benzothieno[2,3‐e]pyrrolo[1,2a]pyrazines and related compounds

S. Rault, J. Lancelot, H. El-Kashef, 1986 .

(1)BENZOTHIENOPYRIMIDINES. I. STUDY OF 3H-BENZOTHIENO(3,2-D)PYRIMID-4-ONE

H. El-Kashef, M. Robba, P. Touzot, 1981 .

THIENOPYRIMIDINES PART 7, REACTION OF THE 4-HYDRAZINOTHIENO(2,3-D)PYRIMIDINES

J. Lecomte, M. Robba, M. D. Sevricourt, 1975 .

Synthesis of cyclic and acyclic nucleoside analogues having a thiophene or dihydrothiophene ring fused to the d side of an uracil

M. Robba, F. Jourdan, J. Renault, 1995 .

SYNTHESIS OF 5'-HALO-2',3'-LYXO-EPOXY AND 2',3'-UNSATURATED THIENO 3,2-D PYRIMIDINE NUCLEOSIDES

M. Robba, C. Fossey, D. Ladurée, 1995 .

Synthesis of some pyrimido[4′,5′:4,5]thieno[2,3-b]quinolines and related heterocycles

S. Rault, A. El-Dean, H. El-Kashef, 1996 .

13C Nmr study of 1,2,4-triazino[4,5-b]indazole derivatives

J. Lancelot, M. Robba, A. Rabaron, 1979 .

Synthesis of new phenylpyrrolylpyrroles

S. Rault, M. Robba, H. Dumoulin, 1995 .

Pyrrolothienopyrimidines. Part 2. Synthesis of 4-Aminopyrrolo[1,2-a]thieno[3,2-e](and[2,3-e]) Pyrimidines.

S. Rault, J. Lancelot, M. Robba, 1986 .

PYRIDO(2,3-H)PYRROLO(1,2-A)QUINOXALINES

S. Rault, J. Lancelot, M. Robba, 1984 .

Synthesis of 1-(β-D-ribofuranosyl)thieno[3,2-d] pyrimidine-2,4-dione and 4-substituted derivatives

M. Robba, C. Fossey, H. Landelle, 1993 .

A convenient route to 6-aminocyclopenta[c]thiophen-4-one derivatives

S. Rault, M. Boulouard, P. Dallemagne, 1987 .

Synthesis of Benzofuro[3,2-f]pythalazine Derivatives

M. Robba, D. Ladurée, E. Chenu, 1991 .

[1]Benzofuro[2,3‐d]pyridazine III. Etude de la dichloro‐1,4 benzofuropyridazine

M. Robba, M. D. Sevricourt, 1978 .

A NEW EFFICIENT SYNTHESIS OF 3-AMINO-1-PHENYLPYRROLE

S. Rault, P. Dallemagne, F. Fabis, 1995 .

Highly potent and selective ligands for histamine H3-receptors

J. Schwartz, J. Arrang, J. Lecomte, 1987, Nature.

Applicability of CoMFA in ecotoxicology: a critical study on chlorophenols.

S. Rault, R. Bureau, F. Briens, 1995, Ecotoxicology and environmental safety.

Synthesis of Cone, Partial-Cone, and 1,3-Alternate 25,27-Bis[1-(2-ethyl)hexyl]- and 25,27-Bis[1-(2-tert-butoxy)ethyl]calix[4]arene-crown-6 Conformers as Potential Selective Cesium Extractants.

J. Leger, C. Jarry, P. Sonnet, 2001 .

A convenient synthesis of new aminopyrroloindoles via an imminium salt

S. Rault, M. Robba, A. Godard, 1985 .

Ètude des reactions de nitration de l'acetamido‐3 ethyl‐9 carbazole

M. Robba, J. Lancelot, J. Gazengel, 1981 .

A Convenient Rearrangement of 1-Phenylpyrrole-2-carboxaldehydes into Their 3-Isomers

S. Rault, P. Dallemagne, F. Fabis, 1994 .

Synthesis of Acyclic Thieno[3,2-d]Pyrimidine Nucleosides and Azido Derivatives as Potential Anti-HIV Agents

M. Robba, C. Fossey, D. Ladurée, 1994 .

Pyrrolothieno[1,4]diazepines part III: Synthesis of amino, hydrazino and mercapto derivatives

S. Rault, M. Boulouard, P. Dallemagne, 1996 .

Pyrrolothieno(1,4)diazepines. Part 1. Synthesis and Study of the Reaction Pathway.

S. Rault, M. Boulouard, P. Dallemagne, 1995 .

Sequence-selective binding to DNA of bis(amidinophenoxy)alkanes related to propamidine and pentamidine.

M. Waring, C. Bailly, C. Saturnino, 1997, The Biochemical journal.

Tetrachloroplatinates et tetrachloropalladates de N,N'(alkane-dyl)bis(guanidinium) leur preparation et leur application en therapeutique

G. Morgant, M. Robba, J. Lancelot, 1996 .

In vitro cytotoxicity of carbazole derivatives. V. 9-Halogeno-substituted 5,11-dimethyl-6H-pyrido[3,2-b]carbazoles

C. Saturnino, P. Gauduchon, F. Sichel, 1997 .

Pyrrolo [1,2-a] thieno [3,2-f] 1,4-diazepines. Novel synthesis and X-ray analysis

S. Rault, M. Robba, M. D. Sevricourt, 1979 .

Synthesis and salidiuretic activity of 2,3-dihydro-8-(1-pyrrolyl)-1,2,4-triazolo[4,3-a]pyridines and 5,6-dihydro-4H-pyrido[2,3-c]pyrrolo[1,2-e]-1,2,5-triazepines.

J. Imbs, M. Barthelmebs, M. Robba, 1991, Chemical & pharmaceutical bulletin.

Novel fused triheterocyclic systems. Synthesis of 6H-pyrido[2,3-c]pyrrolo[1,2-e]-1,2,5-triazepines

J. Lancelot, M. Robba, D. Ladurée, 1985 .

Thiaisatoic Anhydrides: Efficient Synthesis under Microwave Heating Conditions and Study of Their Reactivity.

S. Rault, F. Fabis, M. Robba, 1998 .

Pyrrolothieno[1,4]diazepines: Synthesis of alkoxy derivatives

S. Rault, M. Boulouard, P. Dallemagne, 1995 .

Pyrrolo [1', 2' : 1, 2] pyrazino [6, 5-b] carbazoles

S. Rault, J. Lancelot, M. Robba, 1983 .

Synthesis of 4‐amino[1] benzofuro[3,2‐g] cinnolines

M. Robba, D. Ladurée, D. Florentin, 1980 .

Thiazolo [4,5-d] pyridazine—III

M. Robba, Y. Guen, 1971 .

In vitro cytotoxicity of carbazole derivatives IV. 5,11-Dimethyl-6H-pyrido[3,2-b]carbazoles substituted on the pyridine ring

S. Rault, P. Gauduchon, M. Robba, 1993 .

In vitro effects of Celiptium and MR 14504 on mature rat Leydig cell testosterone production

S. Rault, S. Carreau, M. Robba, 1997, Cell Biology and Toxicology.

Synthesis of 4-Aminothieno[2,3-c]pyrid-7-one from 4-Aminocyclopenta[b]thiophen-6-one

S. Rault, P. Dallemagne, M. Robba, 1988 .

Benzo (1) thieno[2,3-d]pyridazines—II

M. Robba, G. Doré, M. Bonhomme, 1972 .

Comparison of the Effects of Vesamicol and of Cetiedil Analogues on Acetylcholine Release and Vesicular Acetylcholine Transport

M. Robba, M. Israël, M. Diebler, 1991 .

Pyridazino [4,5-b] carbazole : Synthese et Etude des Spectres de Resonance Magnetique Nucleaire

J. Lancelot, M. Robba, H. Landelle, 1984 .

Mutagenicity of nitro- and amino-substituted carbazoles in Salmonella typhimurium. II. Ortho-aminonitro derivatives of 9H-carbazole.

C. Mercier, S. Chemtob, P. Gauduchon, 1995, Mutation research.

Mutagenicity of nitro- and amino-substituted carbazoles in Salmonella typhimurium. I. Monosubstituted derivatives of 9H-carbazole.

S. Rault, C. Saturnino, P. Gauduchon, 1993, Mutation research.

Pyrrolo[2,1-c][1,4]benzodiazepines : A mild conversion of thiolactam into amidine.

S. Rault, M. Robba, M. Foloppe, 1992 .

Pyrrolo[2,1-c][1,4]benzodiazepines: synthesis of N-substituted amidines

S. Rault, M. Robba, I. Rault, 1993 .

THIAZOLO4,3-C1,4BENZODIAZEPINES. II. SYNTHESIS OF FUSEDATRIAZOLO, TETRAZOLO AND OXADIAZOLO DERIVATIVES

S. Rault, M. Boulouard, M. Robba, 1996 .

Thiazolo[4,3-c][1,4]benzodiazepines. I. Synthesis of amidine derivatives

S. Rault, M. Boulouard, M. Robba, 1995 .

Original and quick access to 4-phenyl-6H-pyrrolo[1,2-a]thieno [3,2-f][1,4]diazepines

S. Rault, P. Sonnet, M. Robba, 1995 .

Pyrrolo[1,2-a][1,4] benzodiazepines : An original three-step synthesis from anthranilonitrile.

S. Rault, M. Robba, I. Rault, 1993 .

Pyrrolo(2,1-c)(1,4)benzodiazepines: A Mild Conversion of Thiolactam into Amidine.

S. Rault, M. Robba, M. Foloppe, 1992 .

New access to 4‐phenyl‐6H‐pyrrolo[1,2‐a]thieno[3,2‐f]‐[1,4]diazepines

S. Rault, P. Sonnet, M. Robba, 1996 .

DNA-binding properties of pyrrolo[2,1-c][1,4]benzodiazepine N10-C11 amidines

S. Rault, T. C. Jenkins, D. Thurston, 1996 .

Pyrrolo(2,1‐c)(1,4)benzodiazepines: Synthesis of N‐Substituted Amidines.

S. Rault, M. Robba, I. Rault, 1993 .

Pyrrolo(1,2-a)(1,4)benzodiazepines: An Original Three-Step Synthesis from Anthranilonitrile.

S. Rault, M. Robba, I. Rault, 1993 .

ORIGINAL AND QUICK ACESS TO 4-PHENYL-6H-PYRROLO1,2-ATHIENO 3,2-F1,4 DIAZEPINES

S. Rault, P. Sonnet, M. Robba, 1995 .

Pyrrolo[1,2-a]thieno[3,2-f][1,4]diazepines: new 4H and 4H-5,6-dihydro derivatives

S. Rault, M. Robba, I. Rault, 1994 .

Pyrrolo[1,2-a]thieno[3,2-f][1,4]diazepines: An Efficient Synthesis

S. Rault, M. Robba, I. Rault, 1993 .

Thiazolo(4,3-c) (1,4)benzodiazepines. Part 2. Synthesis of Fused(a) triazolo, Tetrazolo and Oxadiazolo Derivatives.

S. Rault, M. Boulouard, M. Robba, 2010 .

Thiazolo(4,3‐c) (1,4)Benzodiazepines. Part 1. Synthesis of Amidine Derivatives.

S. Rault, M. Boulouard, M. Robba, 1996 .

New Access to 4‐Phenyl‐6H‐pyrrolo(1,2‐a)thieno(3,2‐f)(1,4)diazepines.

S. Rault, P. Sonnet, M. Robba, 1996 .

A new rearrangement under microwave heating conditions: synthesis of cyclopenta[b][1,4]benzodiazepines and tetrahydrodibenzo[b,fl[1,4]diazepines.

S. Rault, M. Robba, Alain-Claude Gillard, 1995 .

Pyrrolothienopyrazines. IV. Synthese de derives de 1′amino-5 pyrrolo[1,2-a]thieno[2,3-e]pyrazine

S. Rault, J. Lancelot, M. Robba, 1987 .

Synthesis of Tetracyclic Systems: A Convenient Route to [1]Benzothieno [2,3-e]pyrrolo[1,2-a]pyrazine and [1]Benzofuro[2,3-e]pyrrolo[1,2-a]pyrazine Derivatives

S. Rault, M. Robba, M. D. Sevricourt, 1981 .

Pyrrolothienopyrazines. Part 4. Synthesis of Derivatives of 5-Aminopyrrolo(1,2-a)thieno(2,3-e)pyrazine.

S. Rault, J. Lancelot, M. Robba, 1987 .

New Condensed Triheterocyclic Systems; Pyrrolothienopyrimidines.

S. Rault, M. Robba, M. D. Sevricourt, 1980 .

In Vivo Nitric Oxide Synthase Inhibitors Can Be Deprived of This Activity: Unexpected Influence of the Tetrachloroplatinate(II) Counteranion. Crystal Structures of Bis(S-Methyl-Isothiouronium)-N,N′-Bis(3-Guanidinopropyl)Piperazinium and Hexamidinium Tetrachloroplatinates(II) Salts

G. Morgant, P. Prognon, M. Roch-Arveiller, 1998, Metal-based drugs.

Benzofuro[2,3-d]pyridazines IV. Etude de la chloro-4 benzofuropyridazine†

M. Robba, A. Godard, M. D. Sevricourt, 1978 .

[1] Benzofuro [2,3‐d] pyridazines II. Etude des benzofuropyridazones

M. Robba, M. D. Sevricourt, 1977 .

Matrix-Assisted Laser Desorption and Ionization Mass Spectrometry and Its Applications in Chemistry

K. Seff, A. K. Dutta, M. Robba, 1990, CHIMIA.

Synthesis and cytotoxic activity against L1210 leukemia of new aminocyclopenta[c]thiophenones.

S. Rault, F. Carreiras, P. Gauduchon, 1994, Chemical & pharmaceutical bulletin.

Synthesis and Cytotoxic Activity Against L1210 Leukemia of New Aminocyclopenta(c)thiophenones (IV).

S. Rault, F. Carreiras, P. Gauduchon, 1995 .

The Third Histamine Receptor

J. Schwartz, J. Arrang, J. Lecomte, 1989 .

SYNTHESIS, CHARACTERIZATION, AND CRYSTAL STRUCTURE OF THE ISOSTRUCTURAL N,N'-(OCTANE-1,8-DIYL)BIS(GUANIDINIUM) TETRACHLOROPLATINATE (II) AND PALLADATE (II) : ANTIAMEBIC EFFECTS STUDY

G. Morgant, N. Dung, M. Robba, 1997 .

Synthesis and study of the stability of 3b,4,4a-5-tetrahydrothieno[2',3':5,4]cyclopenta[2,3-b]aziridine derivatives

D. Maume, S. Rault, P. Dallemagne, 1987 .

Synthesis and Study of the Stability of 3b,4,4a,5‐Tetrahydrothieno‐(2′,3′:5,4)cyclopenta(2,3‐b)aziridine Derivatives.

D. Maume, S. Rault, P. Dallemagne, 1987 .

Complexation d'un agent trichomonacide (ténonitrozole) par l'acétate de rhodium: Structure cristalline du tétrakis(μ‐acétato)‐bis[5‐nitro‐2‐(2‐thénoylamino)‐1,3‐thiazole]dirhodium(II) dichlorométhane

N. Dung, M. Robba, B. Viossat, 1991 .

Comparative molecular field analysis of CCK-A antagonists using field-fit as an alignment technique. A convenient guide to design new CCK-A ligands

Ronan Bureau, Sylvain Rault, Juan Carlos Pilo, 1992, J. Comput. Aided Mol. Des..

Novel selective and partial agonists of 5-HT3 receptors. Part 1. Synthesis and biological evaluation of piperazinopyrrolothienopyrazines.

Sylvain Rault, Philippe Delagrange, M. Hamon, 1996, Journal of medicinal chemistry.