S. Vassiliou

发表

Computer-aided optimization of phosphinic inhibitors of bacterial ureases.

Paulina Kosikowska, P. Kafarski, S. Vassiliou, 2010, Journal of medicinal chemistry.

Novel organophosphorus scaffolds of urease inhibitors obtained by substitution of Morita-Baylis-Hillman adducts with phosphorus nucleophiles.

Łukasz Berlicki, S. Vassiliou, Vassilis Ntatsopoulos, 2017, European journal of medicinal chemistry.

Conformational Properties of New Thiosemicarbazone and Thiocarbohydrazone Derivatives and Their Possible Targets

J. Plavec, T. Mavromoustakos, Demeter Tzeli, 2022, Molecules.

Improved Schöllkopf construction of quaternary α-amino acids: efficient enantioselective synthesis of integrin LFA-1 antagonist BIRT-377

P. A. Magriotis, S. Vassiliou, 2006 .

Phosphinic peptides, the first potent inhibitors of astacin, behave as extremely slow-binding inhibitors.

V. Dive, I. Yiallouros, W. Stöcker, 1998, The Biochemical journal.

Conformational Properties and Putative Bioactive Targets for Novel Thiosemicarbazone Derivatives

J. Plavec, T. Mavromoustakos, Demeter Tzeli, 2022, Molecules.

Novel anti-Alzheimer phenol-lipoyl hybrids: Synthesis, physico-chemical characterization, and biological evaluation.

A. Mardinoğlu, L. Marinelli, A. Di Stefano, 2019, European journal of medicinal chemistry.

Structural exploration of cinnamate-based phosphonic acids as inhibitors of bacterial ureases.

Łukasz Berlicki, S. Vassiliou, Vassilis Ntatsopoulos, 2018, European journal of medicinal chemistry.

Phosphinic acid-based enzyme inhibitors

Łukasz Berlicki, Ewelina Węglarz-Tomczak, M. Talma, 2021, Phosphorus, Sulfur, and Silicon and the Related Elements.

The M 18 Aspartyl Aminopeptidase of the Human Malaria Parasite Plasmodium falciparum *

J. Dalton, T. Spielmann, M. Dixon, 2007 .

A simple synthesis of the metabotropic receptor ligand (2S)-α-(hydroxymethyl)-glutamic acid and its Fmoc protected derivatives

P. A. Magriotis, S. Vassiliou, A. Yiotakis, 2007 .

Structure-Guided, Single-Point Modifications in the Phosphinic Dipeptide Structure Yield Highly Potent and Selective Inhibitors of Neutral Aminopeptidases

A. Joachimiak, B. Nocek, Łukasz Berlicki, 2014, Journal of medicinal chemistry.

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases.

J. Grembecka, P. Kafarski, S. Vassiliou, 2007, Bioorganic & medicinal chemistry.

Three component Kabachnik-Fields condensation leading to substituted aminomethane-P-hydroxymethylphosphonic acids as a tool for screening of bacterial urease inhibitors

Paulina Kosikowska, Łukasz Berlicki, S. Vassiliou, 2011 .

An effective one-pot synthesis of 3-benzylfurans and their potential utility as versatile precursors of 3,4-dibenzyltetrahydrofuran lignans. formal synthesis of (+/-)-burseran.

S. Vassiliou, N. Monteiro, G. Balme, 2001, The Journal of organic chemistry.

Design, synthesis, and evaluation of novel organophosphorus inhibitors of bacterial ureases.

Paulina Kosikowska, Łukasz Berlicki, P. Kafarski, 2008, Journal of medicinal chemistry.

Integrated Transition Metal Catalysed Reactions: Synthesis of Polysubstituted 4‐(Phenoxymethyl)‐3‐pyrrolines and Their Isomers by One‐Pot Coupling of Propargylamines, Vinyl Sulfones (or Nitroalkenes) and Phenols

S. Vassiliou, N. Monteiro, G. Balme, 2002 .

Protection of the Hydroxyphosphinyl Function of Phosphinic Dipeptides by Adamantyl. Application to the Solid-Phase Synthesis of Phosphinic Peptides.

V. Dive, S. Vassiliou, A. Yiotakis, 1996, The Journal of organic chemistry.

Mapping the pathway toward thiophosphinic pseudopeptides. Synthesis of suitably protected PG-Phe-Ψ[P(S)(OX)CH2]-Gly-OY analogues as thiophosphinyl dipeptide isosters (TDI), a comparative study for selective deprotection and further elongation.

S. Vassiliou, Eirini Tzouma, 2013, The Journal of organic chemistry.

Phosphinic peptide inhibitors as tools in the study of the function of zinc metallopeptidases.

V. Dive, P. Cuniasse, D. Georgiadis, 2000, Biochemical Society transactions.

A convenient method to synthesize phosphinic peptides containing an aspartyl or glutamyl aminophosphinic acid. Use of the phenyl group as the carboxyl synthon

V. Dive, D. Georgiadis, S. Vassiliou, 1999 .

Structure of astacin with a transition-state analogue inhibitor

W. Bode, V. Dive, I. Yiallouros, 1996, Nature Structural Biology.

RXP 407, a phosphinic peptide, is a potent inhibitor of angiotensin I converting enzyme able to differentiate between its two active sites.

P Corvol, P Cuniasse, A Yiotakis, 1999, Proceedings of the National Academy of Sciences of the United States of America.

Phosphinic pseudo-tripeptides as potent inhibitors of matrix metalloproteinases: a structure-activity study.

P. Basset, F. Beau, V. Dive, 1999, Journal of medicinal chemistry.

Cyclic peptides with a phosphinic bond as potent inhibitors of a zinc bacterial collagenase.

V. Dive, P. Cuniasse, I. Raynal, 1994, Journal of medicinal chemistry.

RXP 407, a selective inhibitor of the N-domain of angiotensin I-converting enzyme, blocks in vivo the degradation of hemoregulatory peptide acetyl-Ser-Asp-Lys-Pro with no effect on angiotensin I hydrolysis.

P Corvol, A Yiotakis, V Dive, 2001, The Journal of pharmacology and experimental therapeutics.

Rational Design and Synthesis of AT1R Antagonists

T. Mavromoustakos, A. Tzakos, S. Vassiliou, 2021, Molecules.

Discovery of potent and selective inhibitors of human aminopeptidases ERAP1 and ERAP2 by screening libraries of phosphorus-containing amino acid and dipeptide analogues.

Ewelina Węglarz-Tomczak, Stamatia Vassiliou, Artur Mucha, 2016, Bioorganic & medicinal chemistry letters.

Structure assignment, conformational properties and discovery of potential targets of the Ugi cinnamic adduct NGI25

T. Mavromoustakos, Demeter Tzeli, S. Vassiliou, 2021, Journal of biomolecular structure & dynamics.

Covalent Inhibition of Bacterial Urease by Bifunctional Catechol-Based Phosphonates and Phosphinates.

Łukasz Berlicki, S. Vassiliou, A. Grabowiecka, 2020, Journal of medicinal chemistry.

Catechol-based inhibitors of bacterial urease.

Łukasz Berlicki, S. Vassiliou, Katarzyna Macegoniuk, 2019, Bioorganic & medicinal chemistry letters.

The M18 Aspartyl Aminopeptidase of the Human Malaria Parasite Plasmodium falciparum*

J. Dalton, T. Spielmann, M. Dixon, 2007, Journal of Biological Chemistry.

Thiocarbohydrazone and Chalcone-Derived 3,4-Dihydropyrimidinethione as Lipid Peroxidation and Soybean Lipoxygenase Inhibitors

D. Hadjipavlou-Litina, J. Plavec, T. Mavromoustakos, 2023, ACS omega.

Thiophosphinic Acids: Historic Overview and Recent Advances in Their Synthesis and Applications

S. Vassiliou, 2011 .

Rapid and Efficient Microwave-Assisted Hydrophosphinylation of Unactivated Alkenes with H-Phosphinic Acids without Added Metal or Radical Initiator

S. Vassiliou, Panagiota Troupa, Georgia Katsiouleri, 2015, Synlett : Accounts and Rapid Communications in Synthetic Organic Chemistry.

Efficient enantioselective synthesis of orthogonally protected (R)-α-alkylserines compatible with the solid phase peptide synthesis

P. A. Magriotis, S. Vassiliou, A. Yiotakis, 2006 .