Shital Tondlekar

Discovery of 2-((2-chloro-6-fluorophenyl)amino)-N-(3-fluoro-5-(trifluoromethyl)phenyl)-1-methyl-7,8-dihydro-1H-[1,4]dioxino[2',3':3,4]benzo[1,2-d]imidazole-5-carboxamide as potent, selective and efficacious microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitor.

Neelima Khairatkar-Joshi, G. Gudi, S. Jadhav, 2016, Bioorganic & medicinal chemistry letters.

Alleviating CYP and hERG liabilities by structure optimization of dihydrofuran-fused tricyclic benzo[d]imidazole series - Potent, selective and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-2.

Neelima Khairatkar-Joshi, G. Gudi, S. Jadhav, 2018, Bioorganic & medicinal chemistry letters.

Discovery of 5-(2-chloro-4'-(1H-imidazol-1-yl)-[1,1'-biphenyl]-4-yl)-1H-tetrazole as potent and orally efficacious S-nitrosoglutathione reductase (GSNOR) inhibitors for the potential treatment of COPD.

Neelima Khairatkar-Joshi, Daisy M Shah, G. Gudi, 2018, Bioorganic & medicinal chemistry letters.

Discovery of furan and dihydrofuran-fused tricyclic benzo[d]imidazole derivatives as potent and orally efficacious microsomal prostaglandin E synthase-1 (mPGES-1) inhibitors: Part-1.

Neelima Khairatkar-Joshi, G. Gudi, S. Jadhav, 2017, Bioorganic & medicinal chemistry letters.

A Novel and One-Pot Synthesis of 6-arylpyrimidin-4-ol

L. Gharat, Shital Tondlekar, J. M. Gajera, 2008 .

Tricyclic 4,4-dimethyl-3,4-dihydrochromeno[3,4-d]imidazole derivatives as microsomal prostaglandin E2 synthase-1 (mPGES-1) inhibitors: SAR and in vivo efficacy in hyperalgesia pain model.

Neelima Khairatkar-Joshi, G. Gudi, S. Jadhav, 2017, Bioorganic & medicinal chemistry letters.